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1-{4-[(3-phenylpropyl)amino]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
N-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2,2-diethyl-4-[5-(methoxymethyl)-1,3,4-oxadiazole-2-carbonyl]morpholine
4-{[methyl(prop-2-en-1-yl)amino]methyl}-N-(1-methyl-1H-indazol-3-yl)benzamide
3-(3,5-dimethoxyphenyl)-5-[(2-methoxyethyl)sulfamoyl]benzoic acid
1-(2-chloroprop-2-en-1-yl)-6,7-dimethoxy-3-(morpholin-4-ylmethyl)-1,2-dihydroquinolin-2-one
1,3-dimethyl-2,6-dioxo-N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-1,2,3,6-tetrahydropyrimidine-4-carboxamide
N-cyclopropyl-1-[1-(4-methyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
5-({2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}methyl)-N,N-dimethylfuran-2-carboxamide
4-(naphthalen-1-ylmethyl)-3-{2-oxo-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethyl}piperazin-2-one
1-[(3S,4R)-1-[(4-methanesulfonylphenyl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
3-{[3-(2-hydroxyethyl)-4-(thiophen-2-ylmethyl)piperazin-1-yl]methyl}phenol
(furan-2-ylmethyl)(methyl){[1-(2-methylpropyl)-2-phenylmethanesulfonyl-1H-imidazol-5-yl]methyl}amine
1-methyl-N-[2-(4-methylphenyl)ethyl]-3-propyl-1H-pyrazole-5-carboxamide
2-[4-({[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl](methyl)amino}methyl)phenoxy]propanoic acid
4-(2-hydroxypropan-2-yl)-N-(3-phenyl-1,2,4-thiadiazol-5-yl)piperidine-1-carboxamide
N-[(4-hydroxy-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}azepan-4-yl)methyl]-3-methoxypropanamide
3-butyl-1-methyl-4-(1-methyl-3-phenyl-1H-pyrazole-5-carbonyl)piperazin-2-one
3-[7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decane-2-carbonyl]-N,N-dimethylaniline
4-{4-[(3-methylphenyl)methyl]piperazin-1-yl}-4-oxobutane-1-sulfonamide
N-(2-{4-[(4-phenylpiperidin-1-yl)methyl]phenoxy}propyl)-4-sulfamoylbenzamide
2-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carbonitrile
2-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
{4-benzyl-1-[2-methyl-6-(1H-pyrazol-1-yl)pyrimidin-4-yl]piperidin-4-yl}methanol
2-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}benzonitrile
3-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-1-(6-methoxypyridin-3-yl)urea
(1S,5R)-6-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-3-(pyridin-3-yl)propanamide
5-(2-fluorophenoxymethyl)-N-[2-(4-methyl-1H-pyrazol-1-yl)propyl]-1H-pyrazole-3-carboxamide
N-{2-[(3S,4R)-3-cyclopropyl-4-(dimethylamino)pyrrolidin-1-yl]-2-oxoethyl}methanesulfonamide
1-{[2-(4-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(1,3-thiazol-2-yl)piperidine
N-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
5-[(3S,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidine-1-carbonyl]-1,2-oxazol-3-ol
2-[3-({methyl[2-(pyridin-3-yl)ethyl]amino}methyl)phenyl]-6-(oxolan-2-yl)-3,4-dihydropyrimidin-4-one
N-ethyl-2-[3-(pyridin-4-yl)azetidin-1-yl]pyrimidin-4-amine
4-(1,3-dimethyl-4-{[3-(4-methylphenoxymethyl)piperidin-1-yl]methyl}-1H-pyrazol-5-yl)morpholine
5-chloro-2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-[2-(1,3-thiazol-4-yl)ethyl]benzamide
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-[(5-methylthiophen-2-yl)methyl]pyrimidin-2-amine
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5-(hydroxymethyl)furan-2-carboxamide
2-acetyl-8-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-{[4-(methylsulfanyl)phenyl]methyl}-2-(2-oxopyrrolidin-1-yl)-N-propylacetamide
N-{3-[2-(3-hydroxypropyl)-1H-1,3-benzodiazol-1-yl]phenyl}acetamide
2,3-dimethyl-6-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine-1-carbonyl}quinoxaline
(4aS,8aR)-6-[(2-ethylpyrimidin-5-yl)methyl]-1-(2-phenylethyl)-decahydro-1,6-naphthyridin-2-one
2-(3-fluorophenyl)-N-({7-[(2-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)acetamide
2-({1-[(4-fluorophenyl)methyl]piperidin-4-yl}oxy)-4-methoxy-N-(2-methoxyethyl)benzamide
3,5-dimethyl-1-{1-[5-(phenoxymethyl)-1H-pyrazole-3-carbonyl]pyrrolidin-3-yl}-1H-pyrazole
(1R,2S,6R,7S)-4-(5-methyl-1H-indazole-3-carbonyl)-4-azatricyclo[5.2.2.02,6]undecane
4-[4-(4-ethoxyphenyl)-1H-imidazol-2-yl]-2-methoxyphenol