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N,N-dimethyl-2-({1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidin-3-yl}formamido)acetamide
{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}({[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
2-ethoxy-5-{[4-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyridine
6-(cyclopropylmethoxy)-1-[(3-methoxyphenyl)methyl]-4-[3-(pyrazin-2-yl)propanoyl]-1,4-diazepan-2-one
6-[1-(2,1,3-benzothiadiazol-5-ylmethyl)piperidin-3-yl]-2-methylpyrimidin-4-ol
N-{[1-(4-methoxyphenyl)cyclopentyl]methyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
3-(2,4-dimethoxybenzoyl)-1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidine
({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)[(3-methylquinoxalin-2-yl)methyl]amine
N-(2-chloropyridin-3-yl)-4-(thian-4-yl)piperazine-1-carboxamide
N-tert-butyl-4-[5-(2-methylbenzamido)-1H-pyrazol-1-yl]piperidine-1-carboxamide
1-[3-(hydroxymethyl)-3-(2-phenoxyethyl)piperidin-1-yl]-3-phenylprop-2-yn-1-one
2-{4-[5-chloro-2-(piperidine-1-carbonyl)phenoxy]piperidin-1-yl}acetic acid
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-(2-oxo-1,2-dihydropyridin-1-yl)acetamide
5-(2,4-difluorophenoxymethyl)-N-[2-(propan-2-yloxy)ethyl]-1,2-oxazole-3-carboxamide
1'-(4-chlorophenyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-methanesulfonyl-2-({4-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H-1,2,3-triazol-1-yl}methyl)morpholine
(2S)-N-{2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfanyl]phenyl}-2-(methoxymethyl)pyrrolidine-1-carboxamide
4-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-6-(propan-2-yl)pyrimidine
(7-chloro-5-{thieno[2,3-d]pyrimidin-4-yl}-2,3-dihydro-1-benzofuran-2-yl)methanamine
1-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-2-{8-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
7-(propan-2-yl)-N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-4-methylpyridine-3-carboxamide
2-(4-fluorophenoxymethyl)-N-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1,3-oxazole-4-carboxamide
2-amino-4-(2-chloro-4-hydroxyphenyl)-6-(6-methoxypyridin-3-yl)pyridine-3-carbonitrile
6-(2-fluoro-4-methoxyphenyl)-7-methyl-8-oxo-N-(1,3-thiazol-2-ylmethyl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
(1S,5R)-3-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(propan-2-yl)-9-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}acetyl)-2,9-diazaspiro[5.5]undecan-3-one
4-methyl-N-[2-(2-oxoimidazolidin-1-yl)ethyl]-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
N-methyl-2-(pyridin-4-yl)-N-(quinolin-8-ylmethyl)acetamide
4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-[(2E)-3-phenylprop-2-en-1-yl]piperidine
1-(3-methoxyphenyl)-6-methyl-4-[5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carbonyl]piperazin-2-one
[2-(1H-1,3-benzodiazol-2-yl)ethyl][(1-ethyl-1H-imidazol-2-yl)methyl]methylamine
1-[(3-phenoxyphenyl)methyl]-3-(1H-pyrazol-5-yl)piperidine
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-[(2-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-methyl-4-(pyrrolidine-1-carbonyl)-6-(thiophene-2-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-4-methyl-N-(oxolan-2-ylmethyl)-1,3-thiazole-5-carboxamide
1-[4-(1-hydroxy-3-phenylpropyl)piperidin-1-yl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)propan-1-one
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-(dicyclopropylmethyl)-N-methyl-1,3-oxazole-4-carboxamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]benzamide
2-(6-chloro-2H-1,3-benzodioxol-5-yl)-8-methoxy-5-(1H-pyrazol-3-ylmethyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
2-{5-cyclopropyl-4-[4-(piperidin-1-yl)piperidine-1-carbonyl]-1H-pyrazol-1-yl}-4-(3-methoxyphenyl)pyrimidine
methyl 3-benzamido-1-(oxolan-2-ylmethyl)-5-[(thiophen-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[1-(2,6-dimethylphenoxy)propan-2-yl]-2-[methyl(piperidin-4-yl)amino]acetamide
1-[2-(methylamino)-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-6-yl]-2-(1H-pyrazol-1-yl)butan-1-one
1-[2-(dimethylamino)ethyl]-4-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine-1-carbonyl}pyrrolidin-2-one
(3R,4R)-4-(2-methoxyethyl)-3-methyl-1-[2-(methylamino)pyrimidine-5-carbonyl]piperidin-4-ol
4-[(6-fluoroquinolin-2-yl)methyl]-1-(4-methoxyphenyl)-3-methylpiperazin-2-one
N-[(2-methoxyphenyl)methyl]-2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
1-methyl-1'-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
2-(2-methoxyphenyl)-5-(quinoxalin-5-ylmethyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine