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({5-[1-(3-ethoxybenzoyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
5-[2-(4-chlorophenyl)ethyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
(2R,3S,6R)-5-(cyclobutylmethyl)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-[(4-methoxyphenyl)methyl]-3-(1-methylpiperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)methylamine
N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-2-(phenylamino)pyrimidine-5-carboxamide
2-(1H-pyrazol-1-yl)-1-[2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]butan-1-one
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(oxan-4-yl)pyrrolidin-3-yl]-1-methyl-2-oxo-1,2-dihydropyridine-4-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
2-({2-[4-(methylsulfanyl)phenyl]-1H-imidazol-1-yl}methyl)pyridine
1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-4-(pyrrolidine-1-sulfonyl)piperazine
N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]-1H-pyrrole-3-carboxamide
5-(1H-indol-1-ylmethyl)-N-[1-(thiophen-3-yl)propan-2-yl]-1H-pyrazole-3-carboxamide
5-[3-(1H-1,2,4-triazol-1-yl)propyl]-1-[4-(trifluoromethoxy)phenyl]-1H-1,2,4-triazole
(2S,4S)-4-(benzylamino)-1-[(2-chlorophenyl)methyl]-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
(2,3-dihydro-1-benzofuran-5-ylmethyl)({1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
5-methyl-N-[2-(morpholin-4-yl)ethyl]-6-(pyrrolidine-1-carbonyl)thieno[2,3-d]pyrimidin-4-amine
4-cyclopropyl-6-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
1-[(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
2-methyl-6-[(3-phenylcyclobutyl)amino]heptan-2-ol
5-{1-[3-(5-methylfuran-2-yl)benzoyl]pyrrolidin-2-yl}-3-(propan-2-yl)-1,2,4-oxadiazole
(3S,4R)-1-(cyclopentylcarbamoyl)-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
7-methyl-2-{4-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]butanoyl}-2,7-diazaspiro[4.5]decan-6-one
4-benzyl-3-ethyl-1-(2-methyl-6-oxo-1,6-dihydropyrimidine-5-carbonyl)-1,4-diazepan-5-one
1-{3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
3-methyl-7-{[3-(4-methylphenyl)-1,2-oxazol-5-yl]methyl}-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
1-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(pyridin-2-yl)ethan-1-one
(3S,4R)-N,N-dimethyl-1-[2-(morpholin-4-yl)pyrimidine-5-carbonyl]-4-propylpyrrolidin-3-amine
4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[3-(methylsulfanyl)propyl]piperidine
4-(2,2-difluoro-2H-1,3-benzodioxol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
1-(methoxymethyl)-N-[(4-methylphenyl)(pyridin-4-yl)methyl]cyclobutane-1-carboxamide
(2R,4R)-4-hydroxy-N-[4-methyl-3-(3-methylbenzamido)phenyl]pyrrolidine-2-carboxamide
(1R,5R)-6-(cyclobutylmethyl)-3-(naphthalene-1-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]cyclopropan-1-amine
N-cyclobutyl-2-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
N-(4-{[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]methyl}phenyl)acetamide
5-fluoro-2-(1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidin-2-yl)-1H-1,3-benzodiazole
ethyl 4-{6-[(2-phenyl-1,3-thiazol-5-yl)methyl]-6-azaspiro[2.5]octane-1-carbonyl}piperazine-1-carboxylate
N-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-1-[2-(4-chlorophenyl)ethyl]-6-oxopiperidine-3-carboxamide
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-methyl-N-(1,2-oxazol-3-ylmethyl)acetamide
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-3-(4H-1,2,4-triazol-4-yl)propanamide
2-({[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}(methyl)amino)-N-methylacetamide
1-cyclopentanecarbonyl-N-[1-(4-propyl-4H-1,2,4-triazol-3-yl)ethyl]piperidine-4-carboxamide
2-[5-(dimethoxy-1,3,5-triazin-2-yl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(5-methylpyridine-2-carbonyl)pyrrolidin-3-yl]methanol
3-(2-methylpropyl)-N-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}-1,2-oxazole-5-carboxamide
N-[2-(benzylsulfanyl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
2-{2-[(4-benzylpiperazin-1-yl)methyl]-1,3-oxazole-4-carbonyl}-1,2,3,4-tetrahydroisoquinoline
methyl({[5-(oxan-2-yl)furan-2-yl]methyl})(thiophen-3-ylmethyl)amine
1-(3-{[3-(naphthalene-1-carbonyl)piperidin-1-yl]methyl}phenyl)ethan-1-one