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5-ethyl-N-methyl-N-[(1-methylpiperidin-2-yl)methyl]pyrimidin-2-amine
N-methyl-9-oxo-N-[1-(pyrimidin-4-yl)ethyl]-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraene-10-carboxamide
2-hydroxy-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
1-methyl-6-(pyridin-4-yl)-N-[1-(1,3-thiazol-2-yl)propyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-benzyl-N3-ethyl-N5-[(3-fluorophenyl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
3-methoxy-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-4-[(1-methylpiperidin-4-yl)oxy]benzamide
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-(1H-indol-4-ylmethyl)acetamide
methyl 6-({4-[(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}methyl)pyridine-2-carboxylate
6-{1-[(1-ethyl-1H-indol-4-yl)methyl]piperidin-4-yl}-2-methylpyrimidin-4-ol
{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}(1,4-dioxan-2-ylmethyl)amine
butyl N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}carbamate
1-(1,3-thiazole-4-carbonyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
3-(1-methyl-1H-pyrazol-4-yl)-1-{3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}propan-1-one
3-methyl-7-{2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]acetyl}-1-oxa-3,7-diazaspiro[4.5]decan-2-one
3-[2-(3-methoxyphenyl)pyrrolidine-1-carbonyl]-1-methyl-1,4-dihydroquinolin-4-one
4-methyl-N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]-2-oxopentanamide
2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}-1-[3-(4-phenylbenzoyl)piperidin-1-yl]ethan-1-one
2-(benzyloxy)-1-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]ethan-1-one
N-[2-(pyrrolidine-1-sulfonyl)ethyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-amine
1-{3-[(dimethylamino)methyl]-3-hydroxypiperidin-1-yl}-2-(pyridin-4-yl)ethan-1-one
methyl 1-methoxy-2-oxo-8-[(3-phenoxyphenyl)methyl]-1,8-diazaspiro[4.5]decane-4-carboxylate
4-hydroxy-1-[6-(morpholin-4-yl)pyrimidin-4-yl]piperidine-4-carboxylic acid
4-{3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}-1λ6-thiane-1,1-dione
4-[({2H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}(methyl)amino)methyl]-2,6-dimethylphenyl acetate
(3R,4S)-1-(2,6-difluoro-3-methylbenzoyl)-3,4-dimethylpiperidin-4-ol
7,8-dimethyl-2-(2-methylpyrimidin-5-yl)-4-(pyrrolidine-1-carbonyl)quinoline
8-chloro-4-(cyclopropylmethyl)-2-ethyl-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[3-(furan-2-yl)-3-phenylpropyl]-1H-1,2,3-triazole-5-carboxamide
4-benzyl-1-(3-ethoxypropanoyl)-3-ethyl-1,4-diazepan-5-one
3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-[(4-fluorophenyl)methyl]-N-(prop-2-en-1-yl)propanamide
3-methyl-5-[1-(2-phenylethyl)-1H-1,2,3-triazol-4-yl]-1,2,4-oxadiazole
3-[(2-fluorophenyl)formamido]-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]propanamide
(2E)-1-{3-[4-(2-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-3-(pyridin-2-yl)prop-2-en-1-one
N,2,2,6,6-pentamethyl-N-[6-(morpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperidin-4-amine
3,3-dimethyl-1-[(5-{[2-(propylamino)pyrimidin-5-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]urea
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-2-propyl-1,3-thiazole-4-carboxamide
N-[2-(2-chloro-6-fluorophenyl)ethyl]-1-cyclopentyl-5-oxopyrrolidine-3-carboxamide
(3R,5S)-N-[3-(dimethylamino)propyl]-5-(3-fluorophenoxymethyl)-1-(naphthalen-2-ylmethyl)piperidine-3-carboxamide
(3S,4R)-1-[(3-hydroxy-4-methoxyphenyl)methyl]-4-phenylpyrrolidine-3-carboxylic acid
7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-4-cyclohexanecarbonyl-9-(oxolan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-propyl-5-{[4-(pyrrolidine-1-sulfonyl)piperazin-1-yl]methyl}pyrimidin-2-amine
N-[(1R,3S)-3-[(4-chlorophenyl)carbamoyl]cyclopentyl]-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
3-methoxy-2-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyridin-4-amine
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-2,6-dimethylpyrimidine-4-carboxamide
(2R,6R)-6-methyl-1-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
(1R,2R,6S,7S)-4-[6-(morpholin-4-yl)pyrimidin-4-yl]-4-azatricyclo[5.2.1.02,6]decane
2-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-N-methylpyridine-4-carboxamide
N-[(5-methoxy-1H-indol-2-yl)methyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
2-(4-{[7-methyl-2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}phenoxy)ethan-1-ol
1-[1-(3-cyanopyridin-2-yl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide