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1-[(3-{furo[3,2-c]pyridin-4-yloxy}-5-methylphenyl)methyl]pyrrolidine
2,5-dimethyl-3-(4-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazin-1-yl)pyrazine
[(5-tert-butyl-1H-pyrazol-3-yl)methyl](2-methoxyethyl)[(4-methylphenyl)methyl]amine
9-[(4-acetyl-1-methyl-1H-pyrrol-2-yl)methyl]-2-cyclopentyl-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(2S)-3-(4-hydroxyphenyl)-2-{[2-oxo-6-(propan-2-yl)-1,2-dihydropyridin-3-yl]formamido}propanamide
1-[2-(3-phenylpropyl)morpholin-4-yl]-3-(1H-pyrazol-4-yl)propan-1-one
1-cycloheptanecarbonyl-4-(4-propyl-1H-1,2,3-triazol-1-yl)piperidine
N-[(2R,3R)-1'-(1H-indole-6-carbonyl)-2-(pyridin-2-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
4-(3,4-difluorobenzoyl)-5-methyl-1-(4-methylphenyl)piperazin-2-one
3-(azepane-1-sulfonyl)-5-(2,3-dimethoxyphenyl)benzoic acid
methyl 2-[(oxolan-2-ylmethyl)sulfamoyl]-6-(pentan-3-yl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-{4-[4-chloro-2-(2-ethyl-2,5-dihydro-1H-pyrrole-1-carbonyl)phenoxy]piperidin-1-yl}ethan-1-one
ethyl 1-(1-methyl-2-oxo-1,2-dihydroquinolin-4-yl)-5-({methyl[1-(trimethyl-1H-pyrazol-4-yl)ethyl]amino}methyl)-1H-pyrazole-4-carboxylate
1-(4-{4-[1-propyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]piperazin-1-yl}phenyl)ethan-1-one
N-(4-fluoro-2-methylphenyl)-3-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperidin-3-yl]propanamide
4-phenyl-N-[1-(pyridin-3-yl)propan-2-yl]butanamide
2-chloro-4-[3-cyclopropyl-1-(3-methylpyridin-2-yl)-1H-1,2,4-triazol-5-yl]phenol
1-{2-[4-(2-methoxyphenoxy)piperidin-1-yl]-2-oxoethyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
3-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenol
N-[(2R)-oxolan-2-ylmethyl]-5-[4-(2-phenylethyl)piperidine-1-carbonyl]pyridin-2-amine
1-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)-3-(pyrazin-2-yl)propan-1-one
3-{1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl}-N-(3-methylphenyl)propanamide
3-(3-phenyl-1,2,4-oxadiazol-5-yl)-1-(5,6,7,8-tetrahydro-1,6-naphthyridin-6-yl)propan-1-one
2-(4-{[5-(3-chlorophenyl)furan-2-yl]methyl}piperazin-1-yl)pyrimidine
N,3,5-trimethyl-N-{[3-(1-methyl-1,2,5,6-tetrahydropyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,2-oxazole-4-carboxamide
8-methyl-5-(pyrimidin-5-yl)quinoline
N-[1-(4-fluorophenyl)-2-methylpropan-2-yl]imidazo[1,2-a]pyridine-6-carboxamide
N-(2-ethylphenyl)-3-[4-(piperidin-3-yl)-1H-1,2,3-triazol-1-yl]propanamide
methyl 2-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]acetate
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-2-(2-oxopyrrolidin-1-yl)propanamide
8-[3-(morpholin-4-yl)propanoyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]-N-(oxan-4-yl)pyrimidin-2-amine
N-[(4-methylpyridin-2-yl)methyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
3-{[1-(1H-imidazole-5-carbonyl)piperidin-4-yl]oxy}pyridine
methyl (2S,4S,5R)-1,2-dimethyl-5-(2-methylphenyl)-4-[(pyridin-3-ylmethyl)carbamoyl]pyrrolidine-2-carboxylate
N-ethyl-2-(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)acetamide
1-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
(1R,6S)-N-(1H-1,2,3-benzotriazol-5-yl)-9-methyl-3,9-diazabicyclo[4.2.1]nonane-3-carboxamide
6-[6-(methylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]-N-(propan-2-yl)pyridazin-3-amine
(4aS,7aR)-1-[2-(dimethylamino)acetyl]-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(4aS,8aS)-2-[2-(2-methoxy-4-methylphenoxy)ethyl]-decahydro-2,7-naphthyridin-4a-ol
3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-1-[2-(2-phenylethyl)piperidin-1-yl]propan-1-one
N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]-4-oxo-4-phenylbutanamide
(3S,4S)-4-propyl-1-[3-(1H-pyrazol-1-yl)propyl]pyrrolidine-3-carboxylic acid
1-{2-[(propan-2-yl)amino]pyrimidine-5-carbonyl}azetidin-3-ol
1-[3-(dimethylamino)propanoyl]-3-(3-methylbut-2-en-1-yl)piperidine-3-carboxylic acid
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-2-propyl-1,3-thiazole-4-carboxamide
2-({3-[4-(2,6-difluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)-4-methoxyphenol
3-chloro-4-[(1-cyclooctylpiperidin-4-yl)oxy]-N-(2-methoxyethyl)benzamide