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4-ethyl-5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-1,3-thiazol-2-amine
[(5-ethylpyridin-2-yl)methyl](methyl){[1-(2-methylpropyl)-2-(oxolan-2-ylmethanesulfonyl)-1H-imidazol-5-yl]methyl}amine
2-{5-[2-(dimethylamino)propyl]-3-(2-methoxyethyl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
ethyl 2-(1-{[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-2-yl)acetate
1-cyclopentanecarbonyl-N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]piperidine-4-carboxamide
N-(2-methoxyethyl)-1-{1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]piperidin-4-yl}piperidine-3-carboxamide
1-{5-cyclopropyl-1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}-N,N-dimethylpyrrolidin-3-amine
(1s,4s)-4-({methyl[2-(2-methylpiperidin-1-yl)ethyl]amino}methyl)cyclohexan-1-amine
1-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-4-(1-propyl-1H-imidazol-2-yl)-1H-1,2,3-triazole
N-(1-{1-[(3-chlorophenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methoxy-2-phenylacetamide
(3R,4R)-1-[(2-methylpyrimidin-5-yl)methyl]-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-3-ol
5-{3,9-diazaspiro[5.5]undecane-3-carbonyl}-4,6-dimethyl-2H-pyran-2-one
N-(1-{1-[(3-methylquinoxalin-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)oxolane-3-carboxamide
2-(2-methyl-1,3-thiazol-4-yl)-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}acetamide
N-[(3R,4S)-4-cyclopropyl-1-{2-[(2-methoxyethyl)(methyl)amino]acetyl}pyrrolidin-3-yl]methanesulfonamide
N,7-dimethyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]pyrazolo[1,5-a]pyrimidine-6-carboxamide
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-1H-pyrrole-2-carboxamide
1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N-[2-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
4-[2-(4-hydroxyphenyl)acetyl]-5-methyl-1-(4-methylphenyl)piperazin-2-one
3-{2-[3-(2-ethylphenoxy)azetidin-1-yl]-2-oxoethyl}-3,4-dihydroquinazolin-4-one
1-(cyclohex-3-en-1-ylmethyl)-3-[4-(2,5-difluorophenyl)-1H-pyrazol-5-yl]piperidine
1-[6-(2-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-N-ethylpyrrolidine-3-carboxamide
2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-[(3-ethoxyphenyl)methyl]-N-(prop-2-en-1-yl)acetamide
2-cyclopentyl-9-[2-(1H-imidazol-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
6-[3-(5-chloro-2-methoxyphenyl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]-1,3,3-trimethyl-6-azabicyclo[3.2.1]octane
4-[4-(3-chlorophenyl)-3-oxopiperazine-1-carbonyl]-1,2-dihydroquinolin-2-one
7-[2-(oxan-2-ylmethoxy)acetyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-3-phenyl-1,2-oxazole-4-carboxamide
2-(furan-2-yl)-1-[3-(4-methylphenyl)-1H-pyrazole-5-carbonyl]azepane
5-(hydroxymethyl)-N-[4-(4-methylbenzamido)phenyl]furan-2-carboxamide
N-methyl-2-{4-oxo-6-propyl-3H,4H-thieno[2,3-d]pyrimidin-3-yl}acetamide
9-(5-ethyl-1,3-oxazole-4-carbonyl)-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
2-(adamantan-1-yl)-1-[2-(1H-pyrazol-1-ylmethyl)pyrrolidin-1-yl]ethan-1-one
(3R,4S)-1-[4-(difluoromethoxy)benzoyl]-4-propylpyrrolidin-3-amine
2-(3-hydroxypropyl)-9-(2-methyl-2-phenylpropanoyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(2-fluoro-4-methylphenyl)-2-[4-(4-hydroxybutyl)piperazin-1-yl]acetic acid
3-(1-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperidine-3-carbonyl)pyridine
(4aS,7aR)-1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-amino-1-[(6-ethoxypyridin-3-yl)methyl]pyrrolidine-3-carboxylic acid
5-[3-({7-cyclopropanecarbonyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}amino)propyl]-1,3,4-thiadiazol-2-amine
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]amine
3-(1-cyclohexanecarbonylpiperidin-4-yl)-N-(3-methylphenyl)propanamide
2-(4-fluorophenoxymethyl)-N-methyl-N-(pyridin-2-ylmethyl)-1,3-oxazole-4-carboxamide
1-benzyl-N3-ethyl-N5-[(1R)-1-(4-methoxyphenyl)ethyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-[(4-ethoxyphenyl)methyl]-N-(2-methoxyethyl)-[1,2,4]triazolo[4,3-a]pyridine-7-carboxamide
N2,N2,N4,N4-tetramethyl-7-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
N-[1-(cyclohexylmethyl)piperidin-3-yl]-2-methoxybenzamide
2-(4-{[4-(methylsulfanyl)phenyl]methyl}-1-(propan-2-yl)piperazin-2-yl)ethan-1-ol
N-cyclopentyl-2-methyl-7-(oxane-2-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
5-(3-fluorophenoxymethyl)-N-methyl-N-[1-(thiophen-2-yl)ethyl]-1H-pyrazole-3-carboxamide