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N-ethyl-4-hydroxy-N-[(3-methoxyphenyl)methyl]-2-(phenoxymethyl)pyrimidine-5-carboxamide
3-methoxy-1-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
ethyl 4-{2-[3-(2-methoxyphenyl)-1-methyl-2,5-dioxopyrrolidin-3-yl]acetyl}piperazine-1-carboxylate
(3S,4R)-4-(hydroxymethyl)-1-(2-methyl-5-propylpyrimidin-4-yl)piperidin-3-ol
2-(butylsulfanyl)-6-[3-(morpholin-4-yl)azetidin-1-yl]pyrimidin-4-amine
N-[1-(morpholin-4-yl)propan-2-yl]-3-(pyrrolidine-1-carbonyl)benzene-1-sulfonamide
N-[(2R,3R)-2-ethoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylbenzamide
(1S,3R)-3-amino-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}cyclopentane-1-carboxamide
2-[4-(morpholine-4-carbonyl)pyridin-2-yl]-2,7-diazaspiro[4.5]decan-6-one
1-(1,3-dihydro-2-benzofuran-5-yl)-3-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}urea
2-({4-[(2-ethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)-6-methoxyphenol
N-{7-methoxy-2-oxo-4-[2-(trifluoromethyl)phenyl]-1,2,3,4-tetrahydroquinolin-6-yl}propanamide
methyl({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)[2-(oxan-2-yl)ethyl]amine
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-ethoxypropan-1-one
dimethyl(2-{4-[4-(1H-pyrazol-1-yl)benzoyl]morpholin-2-yl}ethyl)amine
5-propyl-1'-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-methyl-N-[2-phenyl-1-(1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)ethyl]thiophene-3-carboxamide
({2,4-dimethyl-5-[(4-methylpiperazin-1-yl)methyl]phenyl}methyl)(methyl)[(2-methyl-1,3-thiazol-4-yl)methyl]amine
(3R)-N-[3-(pyridin-3-yloxy)propyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
4-(1H-imidazol-1-ylmethyl)-1-(quinolin-4-ylmethyl)piperidin-4-ol
7-(cyclohexylmethyl)-2-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-2,7-diazaspiro[4.5]decane
(2S)-2-amino-N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4-(methylsulfanyl)butanamide
2-[3-({4-[(2-ethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenoxy]ethan-1-ol
2-(1-cyclohexyl-4-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}piperazin-2-yl)ethan-1-ol
4-(2-{4-[4-methoxy-3-(prop-2-en-1-yl)phenyl]-1H-1,2,3-triazol-1-yl}ethyl)morpholine
3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-methyl-N-(quinoxalin-2-ylmethyl)propanamide
N-cyclohexyl-N-methyl-3-[({[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}amino)methyl]pyridin-2-amine
2-methyl-4-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
2-methoxy-5-{[methyl({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amino]methyl}phenol
N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-2-[(prop-2-en-1-yl)amino]benzamide
3-[({2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}amino)methyl]pyrrolidin-3-ol
2-methoxy-5-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridine
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-({[(5-methyl-1H-pyrazol-3-yl)methyl]amino}methyl)piperidin-2-one
1-[(3-chloro-5-fluoro-4-methoxyphenyl)methyl]-4-(pyridin-4-ylmethyl)-1,4-diazepane
N-methyl-3-{methyl[2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}propanamide
2-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)morpholine
1-(2-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-oxoethyl)imidazolidine-2,4-dione
(3S,4S)-1-[4-(3-hydroxy-3-methylbutyl)benzoyl]-4-(propan-2-yloxy)pyrrolidin-3-ol
N-{[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}-N-methyl-1,2,3,4-tetrahydronaphthalen-1-amine
9-(cyclopropylmethyl)-1-methyl-4-(3-methyl-1H-pyrazole-5-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
N2-{5H,6H,7H,8H,9H,10H,11H-cycloocta[b]indol-2-ylmethyl}pyrrolidine-1,2-dicarboxamide
2-{[1-benzyl-3-(pyrrolidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-4-phenyl-1,3-thiazole
N-[2-(1H-imidazol-4-yl)ethyl]-2-(morpholin-4-yl)pyrimidine-5-carboxamide
2-cyclopropanecarbonyl-7-[(2,3-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-[(5-fluoro-2-methylphenyl)methyl]-2-(methoxymethyl)-1-methyl-5-(2-phenylacetamido)-1H-1,3-benzodiazole-7-carboxamide
5,6-dimethyl-3-[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidine-1-carbonyl]-1,2-dihydropyridin-2-one
1-(2-{1-[2-(3-methoxyphenyl)acetyl]piperidin-2-yl}ethyl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
(1S,5R)-6-methyl-3-{[4-(1,2-oxazol-5-yl)thiophen-2-yl]sulfonyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[3-(1H-imidazol-2-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-6-(4-fluorophenyl)-N-methylimidazo[2,1-b][1,3]thiazole-3-carboxamide