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N-(4-{[(3S,4S)-3-hydroxy-4-(3-methoxyphenyl)piperidin-1-yl]methyl}phenyl)acetamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]pyrrolidin-3-yl]pyrazine-2-carboxamide
3-(5-tert-butyl-1,3,4-thiadiazol-2-yl)-1-[(1-cyclopentyl-5-oxopyrrolidin-3-yl)methyl]urea
8-{[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-1-oxa-8-azaspiro[4.6]undecan-9-one
3-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-N,N-dimethylpyrazin-2-amine
(1r,4r)-4-[(4,6-dimethylpyrimidin-2-yl)amino]cyclohexan-1-ol
N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(2,5-dioxoimidazolidin-1-yl)acetamide
8-(4-chloro-1-methyl-1H-indole-2-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
3-ethyl-8-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
9-(2-chlorophenyl)-N-(2-methoxyethyl)-N,15-dimethyl-13-oxo-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide
1-(cyclohexylmethyl)-4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
5-cyclobutanecarbonyl-1'-[(3-methylphenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2,3-difluoro-N-[2-(1H-pyrazol-4-yl)ethyl]benzamide
2,3-dimethyl-7-{3-[5-(4-methylphenyl)pyrimidin-4-yl]piperidine-1-carbonyl}-1H-indole
1-[(2-fluorophenyl)methyl]-3-hydroxy-3-{[(pyridin-2-ylmethyl)amino]methyl}piperidin-2-one
1-methyl-2-{1-[4-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]-1H-imidazol-2-yl}-1H-1,3-benzodiazole
(4aS,7aR)-1-(3-hydroxypyridine-2-carbonyl)-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-2,2-bis(prop-2-en-1-yl)piperidine
1-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
3-[2-methoxy-5-(pyrrolidin-1-ylmethyl)phenoxy]-N,N-dimethylpyrazin-2-amine
4-[3-oxo-3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
5-[(2-oxo-1,2,3,4-tetrahydroquinolin-1-yl)methyl]-1,2,4-oxadiazole-3-carboxamide
2-{[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-4-methoxy-3,5-dimethylpyridine
N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]-2-(1H-pyrazol-1-yl)benzamide
2-(2-chloro-4-fluorophenyl)-1-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-ethyl-2-{4-[(3-phenoxyphenyl)methyl]morpholin-3-yl}acetamide
1-[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-3-(thiophen-2-yl)propan-1-one
3-methyl-1-[1-(6-{[(1-methyl-1H-pyrazol-4-yl)methyl]amino}pyridine-3-carbonyl)piperidin-3-yl]butan-1-one
3-[(3S,4R)-1-[(4-chlorophenyl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-N-(2-methoxyphenyl)propanamide
1-[(4aR,8aS)-6-(5-acetylthiophene-3-carbonyl)-decahydro-1,6-naphthyridin-1-yl]-2-(phenylsulfanyl)ethan-1-one
5-methyl-4-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]-1-(2-methylphenyl)piperazin-2-one
1-{3-[(4-fluorophenyl)amino]piperidin-1-yl}-3-phenylpropan-1-one
N,N,4-trimethyl-6-[4-({2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}amino)piperidin-1-yl]pyrimidin-2-amine
2-amino-6-[4-(dimethylamino)phenyl]pyrimidin-4-ol
N-[2-(5-cyano-2-methyl-1H-indol-3-yl)ethyl]-4-hydroxy-1-methylpiperidine-4-carboxamide
2-(dimethylamino)-N-ethyl-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}benzamide
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-2-(1H-pyrazol-1-yl)acetamide
3-(2-{2-[4-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}ethyl)-1,3-oxazinan-2-one
1-(4-chlorophenyl)-5-methyl-4-(3-methylbenzoyl)piperazin-2-one
(2E)-3-(2-chlorophenyl)-N-(2-{4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)prop-2-enamide
2-({4-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]-2-oxo-1-(2-phenylethyl)-1,4-diazepan-6-yl}oxy)-N,N-diethylacetamide
3-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-3-methyl-1-[3-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]urea
N-[(1-hydroxycyclohexyl)methyl]-4-methylpyrimidine-5-carboxamide
2-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]quinoline-4-carboxylic acid
N-[2-(3-ethyl-1,2,4-oxadiazol-5-yl)phenyl]-2-(3-methyl-1,2-oxazol-5-yl)pyrrolidine-1-carboxamide
3-(3,4-dimethoxyphenyl)-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]propanamide
2-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(3-methylphenyl)methyl]acetamide
4-(3-chloro-4-hydroxybenzoyl)-1-(2-methoxyphenyl)piperazin-2-one