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3-methyl-5-[1-(1,3-thiazol-2-ylmethyl)pyrrolidin-2-yl]-1H-1,2,4-triazole
7-methyl-2-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzoyl]-2,7-diazaspiro[4.5]decan-6-one
N-[3-(3-fluorophenyl)phenyl]-1-[(2-hydroxy-6-methoxyphenyl)methyl]piperidine-4-carboxamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-3-(pyridin-2-yl)-3-(pyridin-4-yl)propanamide
(1R,5S)-8-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3,8-diazabicyclo[3.2.1]octane
4-{4-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-4-methylphenyl]phenyl}piperidin-4-ol
1-cyclohexyl-4-(2-methyl-1,3-thiazole-4-carbonyl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
3-methyl-8-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-cyclopropyl-1-[4-(furan-2-yl)pyrimidin-2-yl]-N-[phenyl(pyridin-4-yl)methyl]-1H-pyrazole-4-carboxamide
({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)(isoquinolin-5-ylmethyl)methylamine
(1S,5R)-3-(6-aminopyridine-3-carbonyl)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-7-one
3-(3-methoxyphenyl)-N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-1H-pyrazole-5-carboxamide
2-{4-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1-methylpiperazin-2-yl}ethan-1-ol
1-(4-{4-[(1-ethyl-1H-1,2,3-triazol-4-yl)amino]piperidin-1-yl}phenyl)-3-methylimidazolidin-2-one
3-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-6-oxo-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
(3S,4S)-4-cyclopropyl-1-[4-(4-methylpiperazin-1-yl)benzoyl]pyrrolidine-3-carboxylic acid
5-({3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}methyl)-N-methyl-1,2,4-oxadiazole-3-carboxamide
2-{[5-fluoro-4-(morpholin-4-yl)pyrimidin-2-yl]amino}-N-(2-fluoro-4-methylphenyl)acetamide
1-(2,3-dihydro-1-benzofuran-5-ylmethyl)-N-[4-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
5-propyl-3-[2-(pyridin-2-yl)ethyl]-5-[1-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
N-[5-(1-benzothiophen-7-yl)pyridin-2-yl]methanesulfonamide
1-{3,9-diazaspiro[5.5]undecan-3-yl}-2-(4-ethylpiperazin-1-yl)ethan-1-one
1-[1-(dimethyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]-4-(2-methylphenyl)piperazine
3-methyl-4-(1-{[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl)-1,2,5-oxadiazole
2-({3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}methyl)-3,4-dimethoxypyridine
N-(4-methylphenyl)-N-{[3-(propan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]methyl}methanesulfonamide
3-hydroxy-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-(pyridin-4-ylmethyl)pyridine-2-carboxamide
(3S,4S)-3-hydroxy-N-[3-(methylsulfanyl)phenyl]-4-(propan-2-yloxy)pyrrolidine-1-carboxamide
4-[1-cyclohexyl-5-(5-methyl-1,2-oxazol-3-yl)-1H-1,2,4-triazol-3-yl]benzamide
2-(2-phenylethyl)-8-[2-(pyrrolidin-1-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
N-(2-methoxyethyl)-6,6-dimethyl-5-oxo-N-(pyridin-3-ylmethyl)thiomorpholine-3-carboxamide
2-(2-chloro-6-fluorophenyl)-1-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]ethan-1-one
N-[(2-ethyl-5-fluoro-3-methyl-1H-indol-7-yl)methyl]-2-methyloxane-2-carboxamide
3-methoxy-1-[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-one
(7-chloro-5-{furo[3,2-c]pyridin-4-yl}-2,3-dihydro-1-benzofuran-2-yl)methanamine
N-[1-(5-{[(4-methoxyphenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)-2-phenylethyl]-2-methylpropanamide
3-[(4aS,8aR)-4a-(hydroxymethyl)-decahydro-1,6-naphthyridine-6-carbonyl]-4-fluorobenzene-1-sulfonamide
(1S,6R)-9-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
1-[2-(furan-2-yl)azepan-1-yl]-2-{8-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
N-(oxan-4-yl)-5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
1-ethyl-N-(furan-2-ylmethyl)-N-methyl-5-(morpholin-4-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-{[5-(4-methylphenyl)-1,2-oxazol-3-yl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-[(2-chloro-6-fluorophenyl)methyl]-7-(pyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
7-(2-hydroxyethyl)-2-(2-methanesulfonylethyl)-2,7-diazaspiro[4.5]decan-6-one
N-[5-(methoxymethyl)-1,3,4-thiadiazol-2-yl]-2-{4-[(pyrimidin-2-yl)amino]piperidin-1-yl}acetamide
4-[(2-{[(dimethylcarbamoyl)amino]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl)methyl]benzoic acid
6,8-dimethyl-3-(2,2,6,6-tetramethylpiperidin-4-yl)-3,4-dihydroquinazolin-4-one