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2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-1-[3-methyl-4-(propan-2-yl)piperazin-1-yl]ethan-1-one
3-(4-cyano-2-fluorophenyl)-1-[(1S,2S)-2-hydroxycyclohexyl]urea
(3R,9aR)-3-(2-methylpropyl)-8-[4-(trifluoromethoxy)benzoyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-cyclohexyl-N-(oxolan-2-ylmethyl)-N-propyl-1,3-benzoxazole-6-carboxamide
1-[1-ethyl-3-(4-phenylpiperazine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-methoxy-2-phenylethan-1-one
2-(ethylamino)-N-methyl-N-[(4-phenoxyphenyl)methyl]pyrimidine-5-carboxamide
5-methoxy-2-{[(1S,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}-4H-pyran-4-one
1-[(2S,4R)-1-[(2-methoxynaphthalen-1-yl)methyl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carbonyl]azepane
1-({2-[({5-methylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]phenyl}methyl)pyrrolidin-2-one
1-ethyl-3-(pyrrolidine-1-carbonyl)-5-(thiomorpholin-4-yl)-4,5,6,7-tetrahydro-1H-indazole
N-[(3R,4S)-1-[2-amino-6-(4-methylpiperazin-1-yl)pyrimidin-4-yl]-4-cyclopropylpyrrolidin-3-yl]acetamide
2-(1-ethylpiperidin-4-yl)-1-[2-(1,3-thiazol-2-yl)piperidin-1-yl]ethan-1-one
N-ethyl-5-{[(4-methoxynaphthalen-1-yl)oxy]methyl}-N-[2-(1H-pyrazol-1-yl)ethyl]-1,2-oxazole-3-carboxamide
3-methyl-N-[(1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}pyrrolidin-3-yl)methyl]-1H-pyrazole-5-carboxamide
2-(4-fluoro-2-methoxyphenyl)-4-{1-[(1-methyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-yl}pyridine
2-({[(3R,4R)-1-[(3,5-dichloro-2-methoxyphenyl)methyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)-3-(pyridine-2-carbonyl)piperidine-1-carboxamide
6-cyano-N-{3-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}pyridine-3-carboxamide
N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}quinoline-4-carboxamide
5-(3,5-dimethyl-4-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-1H-pyrazol-1-yl)-1H-1,2,3,4-tetrazole
5-{[(2S)-4-methyl-2-phenylpiperazin-1-yl]methyl}-2-(piperidin-1-yl)pyrimidine
N-{2-[(2-chlorophenyl)formamido]ethyl}-3-(2,5-dioxoimidazolidin-4-yl)propanamide
2,3,5-trimethyl-N-[1-(6-methylpyridin-2-yl)propan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine
2-(2-{[1-(1-methyl-1H-pyrazol-5-yl)propyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
4-(2-fluorophenoxy)-1-(1H-imidazole-2-carbonyl)piperidine-4-carboxylic acid
5-{1-[(4-chlorophenyl)methyl]piperidin-4-yl}-3-(2-methoxyethyl)-5-[(3-methoxyphenyl)methyl]imidazolidine-2,4-dione
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-(dimethyl-1H-1,2,4-triazol-3-yl)-4-[2-oxo-2-(piperidin-1-yl)ethyl]piperazine-1-carboxamide
7-methyl-3-[(5-methylthiophen-2-yl)methyl]-3,7,11-triazaspiro[5.6]dodecan-12-one
3-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)-4,6-dimethyl-1,2-dihydropyridin-2-one
N-[(dimethyl-1,3-thiazol-2-yl)methyl]-5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
8-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
(1S,4S)-2-(3-chloro-4-methoxyphenyl)-5-(2-cyclopentylacetyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
(3R,5S)-N-cyclohexyl-5-[(pyridin-3-yloxy)methyl]piperidine-3-carboxamide
(1S,5R)-6-(cyclopropylmethyl)-3-[1-(pyridine-2-carbonyl)piperidin-4-yl]-3,6-diazabicyclo[3.2.2]nonane
2-(1-methyl-1H-pyrrol-2-yl)-2-oxo-N-[(1R,3S)-3-(thiomorpholine-4-carbonyl)cyclopentyl]acetamide
N-[(5-chloro-1H-indol-2-yl)methyl]-4-methyl-1,3-oxazole-5-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-3-yl)-4-[(2-hydroxyethyl)(methyl)amino]benzamide
1-(4-{2-[9-methoxy-7-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-oxoethyl}phenyl)imidazolidin-2-one
pyridin-3-yl(4-{[4-(trifluoromethyl)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methanol
(1R,7S)-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-4-oxo-3-[4-(propan-2-yl)phenyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
3-(3-methoxyphenyl)-4-{3-methylimidazo[1,5-a]pyridin-1-yl}-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
[(3R,4R)-4-(azepan-1-ylmethyl)-1-[1-(methoxymethyl)cyclobutanecarbonyl]pyrrolidin-3-yl]methanol
N-methyl-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}pyrimidin-4-amine
N-(pyridin-2-ylmethyl)-3-[(1-{spiro[2.3]hexane-1-carbonyl}piperidin-4-yl)oxy]benzamide
9-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
2-{1-[(2-chloro-4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}acetamide
1-[4-(benzyloxy)piperidin-1-yl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
2-[3-(pyridin-4-yl)azetidin-1-yl]-6-(pyrrolidine-1-carbonyl)pyrazine
N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-1-[(4-methylphenyl)amino]cyclopentane-1-carboxamide