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2-(3-fluorophenyl)-1-(1-methyl-1H-pyrrole-2-carbonyl)piperidine
1-[3-(thiophene-2-carbonyl)piperidin-1-yl]-2-(trimethyl-1H-pyrazol-1-yl)ethan-1-one
N-(1-{1-[(4-fluoro-3-methoxyphenyl)methyl]piperidin-4-yl}-2-(3-methoxyphenyl)ethyl)-N-methylfuran-2-carboxamide
{4-[(3-fluorophenyl)methyl]-1-methanesulfonylpiperidin-4-yl}methanol
4-(7-{spiro[2.3]hexane-1-carbonyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl)thiomorpholine
N-{[1-(ethoxymethyl)cyclobutyl]methyl}-4-methyl-2-(pyridin-3-yl)pyrimidine-5-carboxamide
1-{2-oxo-2-[(1S,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethyl}-1,2-dihydropyridin-2-one
4-(2,2-diphenylethyl)-3-[2-oxo-2-(thiomorpholin-4-yl)ethyl]piperazin-2-one
3,3-dimethyl-1-{2-oxo-2-[3-oxo-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-8-yl]ethyl}urea
1-(cyclohexylmethyl)-3-(oxolan-3-yl)-5-(1H-pyrazol-4-yl)-1H-1,2,4-triazole
4-(4-fluoro-2-methylphenoxy)-1-[3-(methylsulfanyl)butyl]piperidine-4-carboxylic acid
(2S,4R)-4-amino-1-{[5-(2-cyanophenyl)furan-2-yl]methyl}-N-ethylpyrrolidine-2-carboxamide
(4aS,7aR)-1-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[4-(2-chloro-4-fluorophenyl)-1H-pyrazol-1-yl]propanamide
1-ethyl-5-methyl-N-[1-(1-methyl-1H-imidazol-2-yl)butyl]-1H-pyrazole-4-carboxamide
N2,N2-dimethyl-N5-{2-methyl-[1,2,4]triazolo[1,5-a]pyridin-8-yl}-4H,5H,6H,7H-thieno[3,2-c]pyridine-2,5-dicarboxamide
2-(1,3-thiazol-2-yl)-N-(1,3,6-trimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)pyrrolidine-1-carboxamide
3-[1-(1-hydroxypropan-2-yl)-1H-imidazol-2-yl]benzonitrile
N-{[4-(1H-1,3-benzodiazol-2-yl)cyclohexyl]methyl}-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
5-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]-4-(propan-2-yl)-1,2,3-thiadiazole
4-(2,5-dimethoxyphenyl)-2-({[(4-methoxyphenyl)methyl]amino}methyl)phenol
N-[2-(propan-2-yl)-2H-1,2,3-triazol-4-yl]-2-{3-[3-(pyrrolidin-1-yl)phenyl]-1H-pyrazol-1-yl}acetamide
1-(1-methyl-5-phenyl-1H-pyrrole-2-carbonyl)-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
N-(2-hydroxyethyl)-2,7-dimethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]imidazo[1,2-a]pyridine-3-carboxamide
6-methyl-3-[3-(morpholin-4-ylmethyl)phenyl]pyridin-2-amine
8-[(3-chloro-5-fluoro-4-methoxyphenyl)methyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
4-cyclopentyl-9-methoxy-7-(4-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(5-fluoro-2-methylphenyl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)acetamide
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-methyl-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
(8aS)-2-[2-(phenylsulfanyl)ethyl]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
2-[(2-amino-6-ethyl-5-methylpyrimidin-4-yl)amino]-1-(thiophen-2-yl)ethan-1-ol
ethyl 3-benzyl-1-(3,4-dimethoxybenzenesulfonyl)piperidine-3-carboxylate
(3R)-1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-3-ol
(4aR,7aS)-N,N-dimethyl-6,6-dioxo-4-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
3-[4-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperazin-1-yl]-1-azabicyclo[2.2.2]octane
3-[(3S,7S,8aS)-3-ethyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-chloro-2-methylphenyl)urea
4-(2H-1,3-benzodioxol-4-ylmethyl)-7-chloro-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-{2-[2-(4-fluorophenyl)azetidin-1-yl]-2-oxoethyl}piperidine-4-carboxamide
ethyl 2-[3-(2-{[(2-fluorophenyl)methyl]carbamoyl}ethyl)piperidin-1-yl]pyridine-3-carboxylate
1-[(4-fluorophenyl)methyl]-5-[(4-methanesulfonylphenyl)methyl]-1H-1,2,4-triazole
1-(6-methyl-1,3-benzothiazol-2-yl)-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N-[3-(4-methoxyphenyl)propyl]-6-[(oxan-3-yl)amino]pyridine-3-carboxamide
1-[1-ethyl-5-(3-fluoro-4-methoxybenzoyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-4-phenylpiperazine
N-ethyl-8-methyl-N-(pentan-2-yl)-2-(pyrimidin-5-yl)quinoline-4-carboxamide
3-[2-(dimethylsulfamoyl)ethyl]-1-[3-fluoro-4-(trifluoromethyl)phenyl]urea
N-[3-(3-methyl-2,5-dioxoimidazolidin-1-yl)phenyl]-2-(pyridin-2-yl)pyrrolidine-1-carboxamide
1-{6-[4-(4-chlorophenoxy)piperidin-1-yl]pyridin-2-yl}ethan-1-ol
3-(1H-pyrazol-1-yl)-1-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}-4-(pyrimidin-2-yl)-1,4-diazepane
N-(3-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-3-oxopropyl)-4-fluorobenzamide