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(1S,5R)-3-(oxan-4-yl)-6-(3-phenyl-1,2-oxazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-[(3-chloro-2,6-difluorophenyl)methyl]-8-methyl-octahydro-1H-pyrazino[1,2-a]piperazine
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)pyrimidin-2-amine
dimethyl({2-[6-(piperidin-1-yl)pyrimidin-4-yl]phenyl}methyl)amine
1-methyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-3-phenyl-1H-pyrazole-5-carboxamide
7-(2-phenylethyl)-2-(pyridine-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
5-(azepane-1-carbonyl)-1-(butan-2-yl)-N-[(3-fluorophenyl)methyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
N-{2-[(2-butyl-6-methylpyrimidin-4-yl)amino]ethyl}-2,7-dioxo-1,3-diazepane-4-carboxamide
ethyl 4-[1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperazine-1-carboxylate
2-[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]-1,3-thiazole-4-carboxamide
N-benzyl-2-(2,6-dioxo-1,3-diazinan-1-yl)-N-(1,3-thiazol-2-ylmethyl)acetamide
7-[(4-methoxy-3-methylphenyl)methyl]-3-(oxolan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
N-{2-[4-(3-methylbut-2-en-1-yl)morpholin-2-yl]ethyl}cyclobutanecarboxamide
N-{[(2S,4S)-4-fluoro-1-(propane-2-sulfonyl)pyrrolidin-2-yl]methyl}morpholine-4-sulfonamide
1-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(propan-2-yl)urea
5-{1-[(2,4-difluorophenyl)methyl]-4-hydroxypiperidin-4-yl}-N-(4-methoxyphenyl)-1-benzofuran-2-carboxamide
4-[2-(4-methoxyphenoxymethyl)-1,3-oxazole-4-carbonyl]piperazine-1-sulfonamide
(3R,4R)-4-amino-1-({5-[(4-methylphenyl)sulfanyl]furan-2-yl}methyl)piperidin-3-ol
4-(3-ethyl-1,2,4-oxadiazol-5-yl)-1-(pyridin-2-ylmethyl)pyrrolidin-2-one
5-fluoro-2-{1-[(5-methyl-1,2-oxazol-3-yl)methyl]piperidin-4-yl}-1H-1,3-benzodiazole
3-amino-N-methyl-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1H-1,2,4-triazole-5-carboxamide
1-[4-(2-phenoxyethyl)piperazine-1-carbonyl]-6-azaspiro[2.5]octane
5-phenyl-4-[1-(pyridine-4-carbonyl)piperidin-4-yl]-2-(trifluoromethyl)pyrimidine
(2S,4R)-4-amino-1-(2-{[(4-fluorophenyl)methyl](methyl)amino}acetyl)-N-methylpyrrolidine-2-carboxamide
N-(2-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-oxoethyl)methanesulfonamide
N-[2-(morpholine-4-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]pyridine-4-carboxamide
(2R,3R,6R)-5-(2H-1,3-benzodioxole-5-carbonyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
3-(1-methyl-1H-imidazol-4-yl)-5-[4-(1H-1,2,4-triazol-5-yl)phenyl]-1,2,4-oxadiazole
3-{2-[4-(1,3-benzoxazol-2-yl)piperidin-1-yl]-2-oxoethyl}-1,3-diazinane-2,4-dione
(2S)-2-({[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}amino)propanamide
ethyl 1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylate
1-methyl-4-({5-[3-(5-methylthiophen-2-yl)-1H-pyrazol-5-yl]-1,2,4-oxadiazol-3-yl}methyl)piperazine
1-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl}-3-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]propan-1-one
5-{1-[5-(1,5-dimethyl-1H-pyrazol-4-yl)-1,2-oxazole-3-carbonyl]pyrrolidin-2-yl}-3-(propan-2-yl)-1,2,4-oxadiazole
2-hydroxy-4-methyl-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)benzamide
2-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-3-yl]pyridine-3-carbonitrile
2-(3-phenylpropyl)-4-(1H-pyrazole-4-carbonyl)morpholine
5-ethyl-2,3-dimethyl-N-[3-(morpholin-4-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-[3-(tert-butylcarbamoyl)-2-methylphenyl]-3-methylfuran-2-carboxamide
N-(1H-1,2,3-benzotriazol-5-yl)-2-methyl-4-[(3-methylphenyl)methyl]-3-oxopiperazine-1-carboxamide
(1H-imidazol-2-ylmethyl)(methyl){[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}amine
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carboxamide
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-[3-(5-methoxy-1-benzofuran-3-yl)-1H-pyrazol-1-yl]acetamide
({1-[(2-fluorophenyl)methyl]-2-(propane-2-sulfonyl)-1H-imidazol-5-yl}methyl)(methyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
(3S,4R)-4-(2-methoxyphenyl)-1-(1,2,5-trimethyl-1H-pyrrole-3-carbonyl)pyrrolidine-3-carboxylic acid
N-(3-methoxypropyl)-5-methyl-4-[(prop-2-en-1-yl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
N-[(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
3-(1,3-benzothiazol-2-ylmethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one