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(1R,5R)-6-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane
5-[2-(methylsulfanyl)benzoyl]-3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
N-methyl-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-N-(thian-4-yl)butanamide
1-methyl-5-{2-[2-(naphthalen-1-yl)pyrimidin-5-yl]-1H-imidazol-1-yl}piperidin-2-one
N-[(3S,5S)-5-{[(1R)-1-(4-methoxyphenyl)ethyl]carbamoyl}-1-methylpyrrolidin-3-yl]morpholine-4-carboxamide
9-{[5-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
6-ethyl-N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)propyl]-2-methylquinoline-4-carboxamide
3-(3,4-dimethylphenyl)-1-methyl-1-[1-(pyrimidin-4-yl)ethyl]urea
1-methyl-5-{[3-(2-methylpropyl)pyrrolidin-1-yl]methyl}-1H-imidazole
2-oxo-6-phenyl-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]-1,2-dihydropyridine-3-carboxamide
{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}[1-(1H-1,2,4-triazol-5-yl)ethyl]amine
9-(2-methoxypyridine-4-carbonyl)-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecane
3-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]-1-(4-methylpiperidin-1-yl)propan-1-one
N-(2,4-dimethylphenyl)-3-[(3-methyl-4,5-dihydro-1,2-oxazol-5-yl)formamido]propanamide
(2R,3R,6R)-5-[(4-methyl-1H-imidazol-5-yl)methyl]-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(4-methylpyridine-3-carbonyl)spiro[azepane-4,2'-chromene]
N-[(2,3-difluoro-4-methoxyphenyl)methyl]-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
1-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)-3-phenylpiperazine
1-(pyrrolidin-1-yl)-3-{1-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]piperidin-4-yl}propan-1-one
N-{[2-(morpholin-4-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)-2-(thiophen-3-yl)acetamide
6-hydroxy-N-{3-[(trifluoromethyl)sulfanyl]phenyl}-1,4-oxazepane-4-carboxamide
2-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-5-(piperidine-1-carbonyl)pyridine
1-benzyl-5-(butylamino)-N-ethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-methyl-3-[(2-{2-methyl-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}acetamido)methyl]benzoic acid
5-(2-fluorophenyl)-N-[2-(4H-1,2,4-triazol-4-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-[4-(1H-pyrazol-1-yl)phenyl]-1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperidine-4-carboxamide
N-[4-chloro-2-(trifluoromethyl)phenyl]-2-oxo-1,3-dioxa-8-azaspiro[4.5]decane-8-carboxamide
N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-2-(1H-1,2,4-triazol-1-yl)acetamide
3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]urea
1-{[4-(1H-imidazol-1-yl)phenyl]methyl}-2-(5-methyl-1,2-oxazol-3-yl)piperidine
1-{1-[(4-methyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
2-{4-[3-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)propanoyl]piperazin-1-yl}-N-ethylacetamide
2-[2-(3-hydroxypiperidin-1-yl)ethyl]-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(4aS,8aS)-2-(6-aminopyrimidin-4-yl)-7-(1-methylcyclopentanecarbonyl)-decahydro-2,7-naphthyridin-4a-ol
N-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
1-[2-(4,6-dimethoxypyrimidin-2-yl)ethyl]pyrrolidin-2-one
(1R,5R)-6-{2-[(3-methoxyphenyl)sulfanyl]acetyl}-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-(1-cyanocyclopentyl)-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-N-propylpiperidine-1-carboxamide
2-[1-(cyclohexylmethyl)-4-[(2,4,5-trimethoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
2-{4-[3-(piperidine-1-carbonyl)pyridin-2-yl]phenyl}acetic acid
N-({2-methoxy-5-oxo-6-[2-(pyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3,3-dimethylbutanamide
N-[3-(4-fluorophenyl)phenyl]-1-(4-methyl-1,3-oxazole-5-carbonyl)piperidine-3-carboxamide
(2S,4R)-4-(4-{[2-(4-fluorophenyl)acetamido]methyl}-1H-1,2,3-triazol-1-yl)-N-methylpyrrolidine-2-carboxamide
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-3-[5-(thiophen-3-yl)-1,3,4-oxadiazol-2-yl]propanamide
methyl (2S,4R)-1-[(4-hydroxyphenyl)methyl]-4-(2-phenylbenzamido)pyrrolidine-2-carboxylate
2-(dimethylamino)-2-(2-methylphenyl)-N-{[1-(piperidin-1-yl)cyclopentyl]methyl}acetamide
3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-(4-fluoro-3-methylbenzoyl)piperidine
[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]({[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
8-(1,2,3,4-tetrahydroquinoline-8-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione