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N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}-2-(2-oxopiperidin-1-yl)acetamide
3-[1-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-3-yl]-N-[(3-methoxyphenyl)methyl]propanamide
1-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethan-1-one
1'-(4-methyl-1H-pyrrole-2-carbonyl)-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
(3S,4S)-1-(4-cyclopentylpyrimidin-2-yl)-4-(piperidin-1-yl)pyrrolidin-3-ol
3-[2-(4-methoxyphenyl)ethyl]-5-methyl-5-{1-[2-(phenylsulfanyl)acetyl]piperidin-4-yl}imidazolidine-2,4-dione
2-({4-[4-(5-methylpyrimidin-2-yl)phenyl]-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)acetic acid
3-{2-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]-2-oxoethyl}-1-methylimidazolidine-2,4-dione
5-[(5,6-dimethyl-1H-1,3-benzodiazol-1-yl)methyl]-N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]-1H-pyrazole-3-carboxamide
2-butyl-N-[2-(7-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-1,3-benzoxazole-5-carboxamide
4-fluoro-N-{2-[(6-fluoro-2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)formamido]ethyl}benzamide
2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1H-1,3-benzodiazole
3-(3-methyl-1H-1,2,4-triazol-5-yl)-1-(5-phenoxyfuran-2-carbonyl)piperidine
3-(1-methyl-1H-pyrazol-5-yl)-1-{3-[3-(4-methylpiperazin-1-yl)-3-oxopropyl]piperidin-1-yl}propan-1-one
N-(2-fluoropyridin-3-yl)-3-(3-methylphenyl)piperidine-1-carboxamide
2-amino-6-cyclobutyl-4-{5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}pyridine-3-carbonitrile
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-3-cyano-N-methylbenzamide
N-(2-{7-[(5-ethylfuran-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-phenoxyacetamide
2-(1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperidin-3-yl)-1,3-benzothiazole
(4aR,8aR)-2-methanesulfonyl-7-(1,2,5-trimethyl-1H-pyrrole-3-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-cyclopropyl-1-(pyridin-2-ylmethyl)pyrrolidine-2-carboxamide
2-amino-7-(pyrazine-2-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-(diethylamino)-3-[2-methoxy-4-({methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}methyl)phenoxy]propan-2-ol
2-[3-(5-fluoro-2-methoxyphenyl)-1H-indazol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-4-[(2-methoxyphenyl)methyl]-9-(oxolan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-hydroxy-2-(1H-1,2,4-triazol-1-ylmethyl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]pyrimidine-5-carboxamide
1-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-[ethyl(methyl)amino]ethan-1-one
N-cycloheptyl-1-[2-(trifluoromethyl)pyrimidin-4-yl]piperidine-4-carboxamide
5-ethyl-N4-{1-[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]ethyl}pyrimidine-2,4-diamine
2-{[3-(aminomethyl)pyrrolidin-1-yl]methyl}-4-tert-butylphenol
5-{1-[2-(cyclohex-1-en-1-yl)ethyl]-1H-imidazol-2-yl}pyrimidin-2-amine
1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-N-[4-(pyridin-3-yloxy)phenyl]piperidine-4-carboxamide
1-(2-methoxyphenyl)-5-methyl-4-[3-(1H-1,2,4-triazol-1-yl)propanoyl]piperazin-2-one
(3R,4R)-1-{[2-(5-methylfuran-2-yl)phenyl]methyl}-4-(morpholin-4-yl)piperidin-3-ol
1-{4-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-4-oxobutyl}pyrrolidin-2-one
5-{2-[1-tert-butyl-3-(2-methyl-1,3-thiazol-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}-4,6-dimethylpyrimidin-2-ol
5-[2-(3-ethoxyphenoxy)ethyl]-3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
4-(2-methoxyphenoxy)-1-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidine
1-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]-2-[2-(thiophen-2-yl)ethyl]piperidine
4-({2-[2-(3-methylpiperidin-1-yl)ethoxy]phenyl}methyl)-1λ6-thiomorpholine-1,1-dione
N-[2-methoxy-4-(quinolin-8-yl)phenyl]acetamide
5-(2-fluorophenoxymethyl)-N-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]-1H-pyrazole-3-carboxamide
1-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]-4-(1H-pyrazol-1-ylmethyl)piperidine
3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-{2-[2-(trifluoromethyl)phenyl]ethyl}propanamide
8-(oxolan-3-ylmethyl)-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
5-(3,4-dimethylphenoxymethyl)-N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1,2-oxazole-3-carboxamide
5-[(6-ethoxyquinolin-2-yl)methyl]-N-methyl-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-(4-chloro-2-methoxyphenoxymethyl)-3-[3-(methoxymethyl)pyrrolidine-1-carbonyl]-1,2-oxazole
1-(adamantan-1-yl)-4-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperazine