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1-(4-ethylpiperazin-1-yl)-3-[1-(3-methylthiophene-2-carbonyl)piperidin-4-yl]propan-1-one
4,6-dimethyl-2-oxo-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]-1,2-dihydropyridine-3-carboxamide
2-(2,3-dihydro-1H-indol-1-yl)-1-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidin-1-yl]ethan-1-one
2-(2,3-dihydro-1H-inden-1-yl)-N-[1-(morpholine-4-carbonyl)piperidin-4-yl]acetamide
3-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}-1-[3-(1H-imidazol-2-yl)piperidin-1-yl]propan-1-one
[(3R,4R)-1-(5-chloro-2-fluorobenzoyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
4-(2,3-dihydro-1H-inden-2-yl)-11-{[(3,4-dimethoxyphenyl)methyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
3-[(dimethyl-1,2-oxazol-4-yl)methyl]-1-[3-(3-ethyl-1,2,4-oxadiazol-5-yl)phenyl]-3-methylurea
4-benzyl-1-[2-(morpholin-4-yl)ethyl]-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-cyclopropyl-1-[1-(8-fluoroquinoline-2-carbonyl)piperidin-4-yl]piperidine-4-carboxamide
2-[3-(3-methoxyphenoxy)azetidin-1-yl]-N-(1,3-thiazol-2-yl)propanamide
1-(2,4-dimethylquinoline-7-carbonyl)azetidin-3-ol
2-({[(3R,4R)-4-(hydroxymethyl)-1-[(pentafluorophenyl)methyl]pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-[(4-hydroxy-3-methoxyphenyl)methyl]pyrazolo[1,5-a]pyridine-7-carboxamide
2-ethyl-8-{1H-pyrrolo[2,3-b]pyridine-2-carbonyl}-2,8-diazaspiro[5.5]undecan-3-one
(1S,6R)-3-{[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
N-(furan-2-ylmethyl)-N-(1-hydroxybutan-2-yl)-4-methyl-3,4-dihydro-2H-1,4-benzoxazine-7-carboxamide
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-5-fluoro-4-(morpholin-4-yl)pyrimidin-2-amine
2-chloro-4-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidine-1-carbonyl]phenol
2-[(4-chlorophenyl)methyl]-4-{4-[(4-methoxy-3-methylphenyl)methyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
(4aS,8aR)-1-butyl-6-{[3-(morpholin-4-yl)phenyl]methyl}-decahydro-1,6-naphthyridin-2-one
2-[3-methyl-5-({1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}methyl)-1H-1,2,4-triazol-1-yl]acetic acid
1-[(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinolin-2-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
1-[3-(furan-2-yl)-3-phenylpropanoyl]-4-hydroxypiperidine-4-carboxylic acid
1-{2-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]-2-oxoethyl}-3,3-dimethylurea
4-(3-hydroxy-3-methylbutyl)-N-(5-oxo-1-propylpyrrolidin-3-yl)benzamide
(2R,6S)-4-(1-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)-2,6-dimethylmorpholine
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}({[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl})amine
5,6-dimethyl-N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
2-(2-methoxyphenoxy)-N-[1-(3-phenylpropyl)piperidin-3-yl]acetamide
(3S,4S)-1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-4-(3-methoxyphenyl)piperidin-3-ol
5-({3-[2-(4-fluorophenyl)piperidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)-2-methylpyridine
1-(2-oxo-2-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethyl)piperidin-2-one
2-(5-fluoro-2-methylphenyl)-1-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
3-(3-hydroxy-3-methylbutyl)-N-[1-(1-methyl-1H-pyrazol-4-yl)propyl]benzamide
2-methyl-N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-2,8-diazaspiro[4.5]decane-3-carboxamide
N-[(3R,4S)-1-(carbamoylmethyl)-4-(propan-2-yl)pyrrolidin-3-yl]-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-2-(phenylamino)pyrimidine-5-carboxamide
2-({[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(thiophen-2-ylmethyl)amino)ethan-1-ol
3-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-6-methyl-4H-pyrido[1,2-a]pyrimidin-4-one
N-[2-(1H-imidazol-1-yl)ethyl]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4-{[2-(ethylamino)pyrimidin-5-yl]methyl}-1-(2-phenylethyl)piperazin-2-one
(2S,4R)-1-benzyl-4-{[(9-ethyl-9H-carbazol-3-yl)methyl]amino}-N-methylpyrrolidine-2-carboxamide
N-{1-[1-(5-ethyl-2-methylpyrimidin-4-yl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopentanecarboxamide
3-fluoro-N-{1-[1-(2-hydroxyacetyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
N-{[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}oxan-4-amine
N-cyclopropyl-3-{1-[(4-acetamidophenyl)methyl]piperidin-4-yl}propanamide
4-benzyl-1-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)-3-ethyl-1,4-diazepan-5-one
1-(oxolane-3-carbonyl)-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
1-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]-2-(pyrimidin-2-ylsulfanyl)ethan-1-one