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2-(3-acetyl-1H-indol-1-yl)-N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]butanamide
5-(2,5-dihydro-1H-pyrrole-2-carbonyl)-N-[2-(dimethylamino)ethyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
5-ethyl-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-1,2-oxazole-3-carboxamide
N-(2-methoxyethyl)-2-(3-methyl-1H-pyrazole-5-carbonyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
3-(3-methoxyphenyl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1H-pyrazole-4-carboxamide
1-[1'-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[2-(1,3-thiazol-2-yl)ethyl]benzamide
methyl (2S,4R)-1-[(3-hydroxyphenyl)methyl]-4-(2-phenylquinoline-4-amido)pyrrolidine-2-carboxylate
5-(2,4-difluorophenoxymethyl)-N-ethyl-N-(oxolan-2-ylmethyl)-1,2-oxazole-3-carboxamide
3-({6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}methyl)pyrrolidin-3-ol
1'-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
8-[(2S)-3-hydroxy-2-(methylamino)propanoyl]-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
9-(2-methoxyethyl)-1-methyl-4-[(1-propyl-1H-imidazol-2-yl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2,5-dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
1-(azepan-1-yl)-3-{3-[(cyclobutylamino)methyl]phenoxy}propan-2-ol
5-tert-butyl-4-{[(1S,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}furan-2-carboxamide
3-methyl-1-propyl-N-[2-(pyridin-4-yl)ethyl]-1H-pyrazole-4-carboxamide
5-{3-[2-(2,3-dimethoxyphenyl)-1H-imidazol-1-yl]phenyl}-1,3-oxazole
2-ethyl-9-[(4-methoxy-2-methylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
methyl 3-acetamido-5-{[(4-fluorophenyl)methyl]amino}-1-[2-(4-methoxyphenyl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
5-{[(5-chloropyridin-3-yl)oxy]methyl}-N-[(4-ethylphenyl)methyl]-N-methyl-1,2-oxazole-3-carboxamide
N-(1,3-benzothiazol-2-ylmethyl)-N-methyl-3-(1H-pyrazol-1-ylmethyl)benzamide
2-[1-(3,5-difluorophenyl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
7-[(2,3-dimethyl-1H-indol-7-yl)methyl]-2,3-dimethyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
1-(4-{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-1,4-diazepan-1-yl)ethan-1-one
3-({[1-({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-3-yl]oxy}methyl)pyridine
N-[3-(furan-2-yl)-3-phenylpropyl]-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-cyclopropyl-1-[(1s,4s)-4-(2-fluorobenzenesulfonamido)cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
7-[(2-fluorophenyl)methyl]-2-(4-methyl-1,3-oxazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
{3-[5-(2-fluorophenyl)-1,2,4-oxadiazol-3-yl]propyl}dimethylamine
1-[(3-methylphenyl)methyl]-4-(oxolane-3-carbonyl)piperazine
1-{1-[(2-methyl-1H-imidazol-4-yl)methyl]piperidin-4-yl}-N-(2-phenylethyl)piperidine-4-carboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-3-ol
1-(3-cyanopyridin-2-yl)-N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]piperidine-3-carboxamide
2-(carbamoylamino)-N-[(1S,3S)-3-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}cyclopentyl]acetamide
2-(3,4,5-trifluorobenzoyl)-2,7-diazaspiro[4.5]decane
4-methyl-3-[(5-{[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]methyl}furan-2-yl)sulfanyl]-4H-1,2,4-triazole
6-{[7-(hydroxymethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}-1,4-oxazepan-6-ol
(3S)-4-[6-(cyclopentylamino)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]-1-ethyl-3-methylpiperazin-2-one
1-[(2,5-dimethoxyphenyl)methyl]-3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)urea
1-[(2,4-dimethylphenyl)methyl]-4-methyl-1,4-diazepan-5-one
5-(2-methoxyphenoxymethyl)-N-(piperidin-4-yl)-1H-pyrazole-3-carboxamide
N-{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
2-[3-benzyl-3-(hydroxymethyl)piperidin-1-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
4-{[5-(2,2-dimethylpropyl)-4-phenyl-1H-imidazol-1-yl]methyl}-1-methylpiperidin-4-ol
5-chloro-N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-N,3-dimethyl-1H-indole-2-carboxamide
3-[(3S,7S,8aS)-1,4-dioxo-3-propyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-phenylurea
2-{[(3,5-dimethylphenyl)methyl]sulfanyl}-1-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidin-1-yl]ethan-1-one
ethyl 4-[2-(pyridin-4-yl)pyrimidine-5-carbonyl]piperazine-1-carboxylate
[5-(1-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-1H-imidazol-2-yl)furan-2-yl]methanol