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3-({1-methyl-2-oxo-1,2-dihydrospiro[indole-3,4'-piperidine]-1'-yl}carbonyl)piperidine-1-carboxamide
4-[2-(5-methylfuran-2-yl)propyl]-1-{[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}-1H-1,2,3-triazole
5-cyclopropyl-N-ethyl-1-{8-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-N-(pyridin-4-ylmethyl)-1H-pyrazole-4-carboxamide
N-[(2-chloropyridin-3-yl)methyl]-N-methyl-4-(1H-1,2,4-triazol-3-yl)benzamide
1-[1-(1-{3-fluoro-7-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-4-yl)ethyl]-4-methylpiperazine
3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}piperidine
N'-[2-(propan-2-yl)phenyl]-N-(3-propoxypropyl)butanediamide
4-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
(1R,5S,6R)-3-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-3-azabicyclo[3.1.0]hexane-6-carboxylic acid
N-(4-fluoro-3-methylphenyl)-6-hydroxy-1,4-oxazepane-4-carboxamide
3-(3,4-difluorophenyl)-N,N-dimethyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-sulfonamide
7-chloro-4-[2-(2-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-tert-butyl-3-{[2-(4-fluorophenyl)azetidin-1-yl]methyl}-1H-pyrazole
2-(dimethylamino)-2-(4-fluorophenyl)-1-[3-(2-methoxyphenoxy)azetidin-1-yl]ethan-1-one
N-[(3R,4S)-1-(2-methanesulfonylethyl)-4-propylpyrrolidin-3-yl]pyridazine-3-carboxamide
N-[(1-methanesulfonylpiperidin-3-yl)methyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
N-[(2S)-4-methyl-1-oxo-1-{4-[(4-propyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}pentan-2-yl]acetamide
2-(4,6-dimethyl-1-benzofuran-3-yl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]ethan-1-one
1-(1H-imidazole-2-carbonyl)-2-methyl-4-(4-methylphenyl)piperazine
3-(4-fluorophenyl)-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-1H-pyrazole-5-carboxamide
4-[4-(4-methoxyphenyl)-2-methyl-3-oxopiperazin-1-yl]-4-oxobutane-1-sulfonamide
(3aR,5R,6S,7aS)-2-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-octahydro-1H-isoindole-5,6-diol
(2S,4S)-1-[(5-chloro-2-hydroxyphenyl)methyl]-4-[(4-fluorophenyl)sulfanyl]-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]pyrrolidine-2-carboxamide
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}acetamide
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
2-{4-[3-(2-hydroxyphenyl)-1H-pyrazole-5-carbonyl]piperazin-1-yl}benzonitrile
N-[2-(4-fluorophenyl)-2-(piperidin-1-yl)ethyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1-[(2-chlorophenyl)methyl]-N-methyl-N-(1-methylpyrrolidin-3-yl)-1H-1,2,3-triazole-4-carboxamide
(1S,5R)-6-(pyridin-2-ylmethyl)-3-(quinoxalin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-tert-butyl-2-[4-(1,2,3,4-tetrahydroisoquinoline-2-sulfonyl)morpholin-3-yl]acetamide
5-(hydroxymethyl)-2-methyl-4-({[(5-methyl-1,2,4-oxadiazol-3-yl)methyl](propan-2-yl)amino}methyl)pyridin-3-ol
N-(1-{5-[(cyclohexylmethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}-2-phenylethyl)-3,4,5-trimethoxybenzamide
1-{2-[(1R,3S,5S)-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octan-8-yl]-2-oxoethyl}imidazolidin-2-one
(2E)-N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-3-(pyridin-3-yl)prop-2-enamide
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-N-{[4-(trifluoromethyl)phenyl]methyl}propanamide
[1-(4-{1-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-1H-1,2,3-triazol-4-yl}phenyl)ethyl]dimethylamine
4-[(dimethylamino)methyl]-1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}azepan-4-ol
4-[2-(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)-1H-imidazol-1-yl]-1-ethylpyrrolidin-2-one
3-{[benzyl(methyl)amino]methyl}-7-methoxy-1,2-dihydroquinolin-2-one
N-{[7-(5-acetyl-2-fluorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,3,6-trifluorobenzamide
N-ethyl-2-(furan-2-yl)-2-oxo-N-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
3-(1-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}pyrrolidin-2-yl)pyridine
2-[(3S,4R)-4-amino-3-methoxypiperidin-1-yl]-6-phenylpyridine-3-carboxylic acid
1-{2-[(2-chlorophenyl)methyl]morpholin-4-yl}-2-(pyridin-4-yl)ethan-1-one
3-(2-benzyl-1,3-thiazole-4-carbonyl)-7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepine
{4-[2-(pyridin-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]morpholin-2-yl}methanamine
1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-3-{[4-(4-ethylpiperazin-1-yl)piperidin-1-yl]methyl}-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-2-one
9-[2-(4-chlorophenyl)-2-hydroxyacetyl]-2-cyclopropyl-2,9-diazaspiro[5.5]undecan-3-one
5-methyl-N-[2-(1-methylpiperidin-3-yl)ethyl]-1-(pyridin-2-yl)-1H-pyrazole-4-carboxamide
5-{2-[(pyridin-3-ylmethyl)amino]ethyl}-1-{[4-(trifluoromethyl)phenyl]methyl}pyrrolidin-2-one