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2-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)pyridine-3-carboxamide
5-(2,6-difluorophenoxymethyl)-N-[1-(1-phenyl-1H-pyrazol-4-yl)ethyl]-1,2-oxazole-3-carboxamide
(2S,4S)-4-amino-N-methyl-1-[1-(trifluoromethyl)cyclopropanecarbonyl]pyrrolidine-2-carboxamide
N-[2-(4-methoxyphenyl)ethyl]-8-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
5,5-dimethyl-1-{2-oxo-2-[3-(pyridin-3-yl)azetidin-1-yl]ethyl}imidazolidine-2,4-dione
6-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-2,3,4,5-tetrahydropyridazin-3-one
methyl 1-(2-methoxyethyl)-5-[(2-methylpropyl)amino]-3-(3-phenylpropanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[(5-amino-1,3,4-thiadiazol-2-yl)(phenyl)methyl]-2-(2-methyl-1,3-thiazol-4-yl)acetamide
2-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]pyridine-3-carbonitrile
6-[3-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]-2,3-dimethyl-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
5,7-dimethyl-N-[1-(propan-2-yl)cyclopropyl]pyrido[2,3-d]pyrimidin-4-amine
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
5-(2-fluorophenoxymethyl)-N-{[1-(hydroxymethyl)cyclobutyl]methyl}-N-methyl-1H-pyrazole-3-carboxamide
2-benzyl-5-[4-(propan-2-yl)benzoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine
2-ethyl-9-(2-hydroxyethyl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
6-ethyl-1,5-dimethyl-3-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
N-cyclohexyl-5-(pyrrolidin-1-ylmethyl)-N-(thiophen-3-ylmethyl)furan-2-carboxamide
N-[1-methyl-4-(propan-2-yloxy)-1H-indazol-3-yl]-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
1,6-dimethyl-N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-methyl-6-[1-(3-phenyl-1,2-oxazole-4-carbonyl)piperidin-3-yl]pyrimidin-4-ol
2-[2-(1-{2-[(2-ethyl-6-methylpyridin-3-yl)oxy]acetyl}piperidin-4-yl)-1H-imidazol-1-yl]acetamide
N-methyl-5-{[(trimethylpyrimidin-4-yl)amino]methyl}-1,2,4-oxadiazole-3-carboxamide
3-{4-[4-methoxy-3-(methoxymethyl)phenyl]-1H-1,2,3-triazol-1-yl}propane-1,2-diol
1-{1-[(7-hydroxyquinolin-3-yl)methyl]piperidin-4-yl}pyrrolidin-2-one
2-[1-(thiophen-3-ylmethyl)-4-[(2,3,6-trifluorophenyl)methyl]piperazin-2-yl]ethan-1-ol
(4aS,8aR)-1-(2-aminoethyl)-6-(quinolin-2-yl)-decahydro-1,6-naphthyridin-2-one
1-[(2-methoxyphenyl)methyl]-4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-{4H,5H,6H,7H,8H-cyclohepta[b]thiophene-2-carbonyl}-N-phenylpiperidin-3-amine
(3S,4S)-4-cyclopropyl-1-(2-methyl-1H-1,3-benzodiazole-5-carbonyl)pyrrolidine-3-carboxylic acid
N-[5-oxo-1-(propan-2-yl)pyrrolidin-3-yl]-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
(3S,4S)-1-(morpholine-4-sulfonyl)-4-(naphthalen-2-yl)piperidin-3-ol
2,N4-dimethyl-N4-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]pyrimidine-4,6-diamine
N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-1-propanoylpiperidine-3-carboxamide
2-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]-5-[4-(prop-2-en-1-yloxy)phenyl]-2H-1,2,3,4-tetrazole
(2S,4S)-4-[4-({[(5-fluoro-2-methylphenyl)carbamoyl]amino}methyl)-1H-1,2,3-triazol-1-yl]pyrrolidine-2-carboxylic acid
methyl[(4-{2-[4-(oxolane-2-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl](quinolin-6-ylmethyl)amine
1-[3-(1,3-benzoxazol-2-yl)piperidin-1-yl]-2-(pyridin-3-yl)ethane-1,2-dione
5-(2-chloro-4-methoxyphenoxymethyl)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-1H-pyrazole-3-carboxamide
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-N-methyl-3-(2-methylphenyl)-3-phenylpropanamide
8-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]-1-[(2-fluorophenyl)methoxy]-1,8-diazaspiro[4.5]decan-2-one
1-(2,3-dimethylphenyl)-N-[(2-methyl-1,3-thiazol-4-yl)methyl]piperidin-4-amine
1-{2-[1-(2,3-dihydro-1H-inden-2-yl)-3-ethyl-1H-1,2,4-triazol-5-yl]ethyl}-6-methyl-1,2-dihydropyridin-2-one
1-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
8-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]-1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-methoxy-4-[(1E)-3-{4-[2-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}prop-1-en-1-yl]phenol
2-(1-{[1-(3-methylphenyl)-1H-imidazol-2-yl]methyl}piperidin-3-yl)-1,2,3,4-tetrahydroisoquinoline
2-[(3S)-3-hydroxypyrrolidin-1-yl]-N,1-dimethyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-1H-1,3-benzodiazole-5-carboxamide
N-methyl-N-{3-[(4-methylphenyl)sulfanyl]propyl}morpholine-2-carboxamide
8-(1H-1,3-benzodiazol-2-ylmethyl)-1-methyl-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione