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4-benzyl-1-cyclopropanecarbonyl-3-ethyl-1,4-diazepan-5-one
2-[7-(1-benzothiophen-3-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-methylacetamide
4-{[5-(4-methyl-1H-imidazol-5-yl)-1,2,4-oxadiazol-3-yl]methyl}-1-propylpiperidine
N-{2-[2-(pyridin-3-yl)-1,3-thiazol-4-yl]ethyl}-3,4-dihydro-2H-1-benzopyran-6-carboxamide
N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-N-methyl-1-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
3-[5-(2,3-dihydro-1-benzofuran-2-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
3-methyl-N-[1-(1-{[4-(pyrimidin-2-yloxy)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]butanamide
N-[2-(4-methoxyphenyl)ethyl]-4-methyl-N-[(1-methylpiperidin-4-yl)methyl]-1,3-oxazole-5-carboxamide
1-[(2-methylphenyl)methyl]-N-[3-(pyridin-3-yloxy)propyl]-1H-1,2,3-triazole-4-carboxamide
4-ethyl-3-({1-[(3-fluorophenyl)methyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-methyl-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
1-cyclobutyl-3-(2,4-dimethoxybenzoyl)piperidine
1-(5-chloropyridin-2-yl)-4-[2-(1H-1,2,4-triazol-3-yl)benzoyl]piperazine
4-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-1-butylpiperazin-2-one
4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(4-methylphenyl)methyl]piperidine
1-methyl-9-{[1-(4-methylpyridin-2-yl)-1H-pyrrol-2-yl]methyl}-1,4,9-triazaspiro[5.5]undecan-5-one
N-[3-(2-methoxyphenyl)propyl]-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[(1-methyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-yl]-3-hydroxypyridine-2-carboxamide
2-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-1,3-benzoxazole
5-(3-benzyl-1,2,4-oxadiazol-5-yl)-N-methyl-N-(pyridin-3-ylmethyl)pyridin-2-amine
(2,1,3-benzoxadiazol-4-ylmethyl)(methyl)[1-(pyridin-4-yl)ethyl]amine
1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)-4-propylpiperazine
1-[2-(1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)ethyl]pyrrolidin-2-one
2-(oxolan-2-ylmethyl)-8-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-2,8-diazaspiro[4.5]decan-3-one
3-(1-methyl-1H-imidazole-2-carbonyl)-1-[3-(thiophen-2-yl)-1H-pyrazole-4-carbonyl]piperidine
N-[(6-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridin-3-yl)methyl]acetamide
2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]-N-[3-(pyridin-3-yl)propyl]acetamide
N5-[(4-fluorophenyl)methyl]-N3-methyl-N3-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-(pyridin-2-ylmethyl)-1-(quinoxaline-6-carbonyl)piperidine-4-carboxamide
3-chloro-N-[2-(dimethylamino)ethyl]-4-({1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}oxy)benzamide
2-[4-hydroxy-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidine-1-carbonyl]-6-methyl-4H-pyran-4-one
N-cyclopentyl-2-(2-methyl-1,3-thiazol-4-yl)-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)acetamide
2-(1H-1,3-benzodiazol-1-yl)-1-{7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}ethan-1-one
N-(2-methoxyethyl)-4-methyl-3-{[(6-methylpyridin-3-yl)carbamoyl]methyl}-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
5-(methoxymethyl)-N-(1-{7-[(3-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)furan-2-carboxamide
6-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrole-1-sulfonyl]-1,2,3,4-tetrahydroquinolin-2-one
N4-[(dimethyl-1,3-thiazol-2-yl)methyl]-6-methylpyrimidine-2,4-diamine
3-(pyrimidin-5-yl)-5-(pyrrolidine-1-sulfonyl)benzoic acid
5-[3-(4-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-1H-1,3-benzodiazole
(2S,4R)-4-amino-1-(4-ethenylbenzoyl)-N-methylpyrrolidine-2-carboxamide
4-{[3-(2-hydroxyethyl)-4-(3-methylbut-2-en-1-yl)piperazin-1-yl]methyl}-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
methyl 4-[6-amino-5-cyano-4-(4-methyl-1H-imidazol-5-yl)pyridin-2-yl]benzoate
N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
N-[1-(2,6-dimethylphenoxy)propan-2-yl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-5-(morpholin-4-ylmethyl)furan-3-carboxamide
2-[2-(3-methoxyphenyl)ethyl]-4-[4-(pyrazine-2-carbonyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
5-[(isoquinolin-5-yloxy)methyl]-N-[1-(1,3-thiazol-2-yl)ethyl]-1,2-oxazole-3-carboxamide
1-(2-{imidazo[1,2-a]pyridin-6-ylformamido}ethyl)piperidine-3-carboxamide
2-methyl-6-[4-(5-methylpyrimidin-4-yl)piperidine-1-carbonyl]-4H-pyran-4-one
6-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pyrazine-2-carboxamide