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2-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)morpholine
1-(2,3-dihydro-1H-inden-2-yl)-4-[(1,4-dithiepan-6-yl)amino]pyrrolidin-2-one
6-(azepane-1-carbonyl)-2-[(4-methoxyphenyl)methyl]-1,3-benzoxazole
methyl[(3-methylpyrazin-2-yl)methyl][(3-phenyl-1H-pyrazol-5-yl)methyl]amine
2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-[2-(methylsulfanyl)ethyl]-1,3-oxazole-4-carboxamide
[(3R,4R)-1-{[6-(dimethylamino)pyridin-3-yl]methyl}-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}pyrrolidin-3-yl]methanol
3-[1-(5-cyclopropyl-1,3,4-oxadiazol-2-yl)piperidine-3-carbonyl]pyridine
3-fluoro-N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)benzamide
N-(2-methoxyethyl)-3-pentanamido-N-(1,3-thiazol-2-ylmethyl)benzamide
N-{[4-(2-methylpropyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}pyridine-2-carboxamide
1-(2-chlorophenyl)-4-(5-methoxy-1H-indazole-3-carbonyl)piperazin-2-one
2-(4-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)pyrimidine
N-[3-(3-chlorophenyl)phenyl]-1-(pyridine-3-carbonyl)piperidine-4-carboxamide
methyl 3-acetamido-1-[2-(4-methoxyphenyl)ethyl]-5-{[(4-methylphenyl)methyl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-{4-[(3-methoxyphenyl)methyl]piperazin-1-yl}-2-{[3-(pyridin-3-yl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]sulfanyl}ethan-1-one
1-[1-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]-4-[3-(trifluoromethyl)phenyl]piperazine
1-cyclohexyl-N3-methyl-N5-[2-(7-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
3-[3-(2,5-dimethoxyphenyl)phenyl]-1-(2-fluoroethyl)-1H-pyrazole
10-methoxy-5-(piperidin-3-yl)-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
N-cyclopropyl-2-{[1-methyl-3-(2-methylpropyl)-1H-pyrazol-5-yl]formamido}acetamide
1-(3,4-dihydro-2H-1-benzopyran-3-yl)-2-(2-ethoxyphenyl)-1H-imidazole
4-{[1-(3-chloro-4-fluorophenyl)-5-(pyrrolidin-3-yl)-1H-1,2,4-triazol-3-yl]methyl}-1-methylpiperidine
2-[4-({4-[2-(2-methylphenyl)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperazin-1-yl]ethan-1-ol
[(2S,6S)-4-(dimethyl-1,3-thiazol-2-yl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
5-(2-methylphenyl)-3-[4-(pyridin-2-yl)piperazin-1-yl]-1,2,4-triazine
4-ethyl-1-{2-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonan-3-yl]-2-oxoethyl}-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(2-hydroxyethyl)-N-methyl-1-{1-[(2-methyl-1H-indol-3-yl)methyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[2-(5-methylfuran-2-yl)ethyl]benzamide
9-[2-(propan-2-yloxy)acetyl]-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-[4-(2-methoxypyridine-3-carbonyl)-1-(2-methylpropyl)piperazin-2-yl]ethan-1-ol
3-[(3R,7S,8aS)-3-(hydroxymethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2-fluorophenyl)urea
ethyl 1-(2-{1-cyclopropyl-2,5-dioxo-3-[3-(trifluoromethyl)phenyl]pyrrolidin-3-yl}acetyl)piperidine-2-carboxylate
4-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-8-thia-4,6-diazatricyclo[7.5.0.02,7]tetradeca-1(9),2(7),5-trien-3-one
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)-2-(2-methyl-1,3-thiazol-4-yl)acetamide
2-({4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)-3-methylpyridine
2-[1-(2,2-dimethylpropyl)-4-[(2,4,5-trimethoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
(2E)-N-[(3,4-dimethoxyphenyl)methyl]-3-(3-fluorophenyl)-N-(pyridin-3-ylmethyl)prop-2-enamide
N-benzyl-N-methyl-1-(1,2,3-thiadiazole-4-carbonyl)piperidin-3-amine
1-amino-N-({2-[4-(2-methoxyphenyl)piperazin-1-yl]pyridin-3-yl}methyl)cyclopropane-1-carboxamide
N-({1-[3-(5-amino-1H-1,2,4-triazol-3-yl)propanoyl]piperidin-4-yl}methyl)acetamide
(3aS,7aR)-5-methyl-2-phenylmethanesulfonyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
4-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-1-(4-methylphenyl)piperazin-2-one
1,5-dimethyl-4-{[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-1H-pyrrole-2-carbonitrile
N-[3-(methylamino)propyl]-2-(1H-1,2,4-triazol-3-yl)benzamide
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-{[3-(1H-1,2,4-triazol-1-yl)phenyl]methyl}pyrimidin-2-amine
5-methyl-1-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-5-phenylpiperidin-2-one
N-{[1-(2,1,3-benzoxadiazol-5-ylmethyl)pyrrolidin-3-yl]methyl}pyridine-2-carboxamide
N-[(3R,4S)-1-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
1-cyclopentyl-4-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}piperazine
4-[1-({[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}amino)ethyl]hepta-1,6-dien-4-ol