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(3R,5S)-1-benzyl-N3-(2,3-dihydro-1H-inden-5-yl)-N5-[(3-fluorophenyl)methyl]piperidine-3,5-dicarboxamide
2-(dimethylamino)-1-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]-2-(3-methylphenyl)ethan-1-one
5-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1-(2-methylphenyl)-1H-1,2,4-triazole
2,5,6-trimethyl-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}pyrimidin-4-amine
1-butanoyl-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-2-carboxamide
2-{[1-(4-methoxyphenyl)-3-(2-methyl-1,3-thiazol-4-yl)-1H-1,2,4-triazol-5-yl]methyl}morpholine
6-(2-methylpropyl)-2-oxo-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-1,2-dihydropyrimidine-4-carboxamide
N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]-5-[(methylsulfanyl)methyl]furan-2-carboxamide
4-(6-methyl-2-propylpyrimidin-4-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
2-{[(4S,4aS,8aS)-4-hydroxy-4-phenyl-decahydroquinolin-1-yl]methyl}-5-methoxy-4H-pyran-4-one
4-{[4-(3-hydroxypiperidin-1-yl)piperidin-1-yl]methyl}-1-methyl-1H-pyrrole-2-carbonitrile
4-[4-(2,5,7-trimethylquinoline-4-carbonyl)piperazin-1-yl]phenol
4-{3-[9-methoxy-7-(4-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]butyl}phenol
N-[2-(furan-2-yl)ethyl]-2-[4-(propan-2-yl)morpholin-2-yl]acetamide
N-(2-{4-[(6-methylpyridin-2-yl)methyl]morpholin-2-yl}ethyl)benzamide
3-(2-methyl-1H-imidazol-1-yl)-6-(2,4,6-trimethylphenyl)pyridazine
N,N-diethyl-1-[6-fluoro-2-(1-methyl-1H-pyrazol-4-yl)quinoline-4-carbonyl]pyrrolidin-3-amine
N-{2-[2-(3-chloro-5-fluorophenyl)-1H-imidazol-1-yl]ethyl}pyridine-4-carboxamide
1-({4-methyl-5-[1-(pyrimidin-2-yl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
3-(azocan-1-yl)-N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]propanamide
(3aR,6aR)-2-(cyclobutylmethyl)-5-(3-cyclopropylpropanoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(1,4-diazepane-1-sulfonyl)-N-(3-ethoxypropyl)benzamide
2-(1H-indazol-1-yl)-N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}acetamide
1-(4-chlorophenyl)-4-{1,3-dimethyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1H-pyrazole
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-(4,5,6,7-tetrahydro-2H-indazol-3-yl)propanamide
4-[2-(dimethylamino)-2-(2-fluorophenyl)acetyl]piperazine-1-sulfonamide
1-(3-methoxypyrazin-2-yl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-[3-oxo-3-(4-phenylazepan-1-yl)propyl]pyrrolidin-2-one
1-(pentan-3-yl)-4-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
methyl 4-[(2-cyclopropyl-1,3-benzoxazol-6-yl)formamido]butanoate
1-(4-{[3-(dimethyl-1,2-oxazol-4-yl)propyl]amino}-2-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
(1R,5R)-6-benzyl-3-(3-phenyl-1H-pyrazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-{[1-(4-methylpiperazin-1-yl)cyclohexyl]methyl}-1-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
3-methoxy-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
N,N-dimethyl-4-[3-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]piperidine-1-carboxamide
2-(1-{5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carbonyl}piperidin-3-yl)-4-methyl-1H-1,3-benzodiazole
(2S,4S)-4-acetamido-N,N-diethyl-1-{[2-(methylsulfanyl)phenyl]methyl}pyrrolidine-2-carboxamide
(1S,5R)-N-{3-[(2-methylprop-2-en-1-yl)oxy]phenyl}-10-oxo-3,9-diazabicyclo[3.3.2]decane-3-carboxamide
N-(2-methoxyethyl)-2-(4-methyl-1H-imidazole-2-carbonyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
[3-(cyclopropylmethyl)-1-(1,2,3,4-tetrahydroquinoline-8-carbonyl)piperidin-3-yl]methanol
1-[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propan-1-one
2-[1-(5-methyl-1,3-oxazole-4-carbonyl)piperidin-2-yl]pyridine
3-(3-tert-butyl-1-methyl-1H-pyrazol-5-yl)-1-[3-(1H-1,2,3-triazol-1-yl)propyl]urea
5-{1-[(dimethyl-1,2-oxazol-4-yl)methyl]pyrrolidin-2-yl}-N-(2-methylpropyl)thiophene-2-carboxamide
{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
[(1,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)(thiophen-3-ylmethyl)amine
1-[1'-(4-fluoro-3-methylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
5-(2-methylphenyl)-N-[3-(1H-pyrazol-1-yl)propyl]-1,2,4-triazin-3-amine
6-cyclopentyl-N-[2-methoxy-1-(pyridin-2-yl)ethyl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-(3-phenylpropyl)-4-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-1,4-diazepane