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ethyl 2-{[5-({[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]amino}methyl)pyrimidin-2-yl](methyl)amino}acetate
5-benzyl-4-(2-hydroxyacetyl)-1-(2-methylphenyl)piperazin-2-one
N-[2-(furan-2-ylmethyl)-3-hydroxypropyl]-3-(1H-pyrazol-4-yl)benzamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]ethan-1-one
methyl (2S,4R)-1-[(2,4-dimethoxyphenyl)methyl]-4-[3-(4-fluorophenyl)benzamido]pyrrolidine-2-carboxylate
1-[1-(6-methyl-2-propylpyrimidin-4-yl)piperidin-4-yl]-3-phenylpyrrolidin-3-ol
N-(1,3-benzoxazol-2-ylmethyl)-2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
N-benzyl-2-cyclopropyl-N-[(4-methyl-1,3-thiazol-5-yl)methyl]-1,3-benzoxazole-6-carboxamide
N-[1-(2-amino-9H-purin-6-yl)piperidin-4-yl]methanesulfonamide
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-6-methoxypyrimidin-4-amine
2-methyl-N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]-6-oxo-1,6-dihydropyrimidine-5-carboxamide
1-cyclopentanecarbonyl-N-[(2-ethoxy-3-methoxyphenyl)methyl]piperidine-4-carboxamide
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)-2-methyl-1H-pyrrole-3-carboxamide
N-[1-(7-{[3-(4-chlorophenoxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]furan-2-carboxamide
2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(3-hydroxy-2,2-dimethylpropyl)acetamide
N,N-dimethyl-2-{[2-(1H-pyrazol-1-yl)butanamido]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
1-ethyl-3-(7-fluoro-1-methyl-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-6-methyl-1,2-dihydropyridin-2-one
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-(2-methyl-1H-1,3-benzodiazol-5-yl)acetamide
3-({[1-(hydroxymethyl)cyclobutyl]methyl}sulfamoyl)-N-(pyrrolidin-3-yl)benzamide
5-(1H-indol-1-ylmethyl)-N-[2-methyl-2-(morpholin-4-yl)propyl]-1H-pyrazole-3-carboxamide
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyloxan-4-amine
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(pyridine-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-{imidazo[1,2-a]pyridin-2-yl}propanamide
N-[(6-{pyrazolo[1,5-a]pyridin-7-yl}pyridin-3-yl)methyl]acetamide
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N-methyl-6-oxo-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
4-[(5-cyclobutyl-1,3,4-oxadiazol-2-yl)amino]-N-cyclohexylpiperidine-1-carboxamide
N-({3-[2-(dimethylamino)ethoxy]phenyl}methyl)-2,3-dimethyl-N-(pyridin-2-ylmethyl)-1H-indole-7-carboxamide
N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)oxane-4-carboxamide
2-{5-[2-(furan-2-yl)azepane-1-carbonyl]-1H-pyrazol-3-yl}phenol
6-methyl-N4-[3-methyl-1-(pyridin-3-yl)butyl]pyrimidine-2,4-diamine
1-[2-(4-fluorophenoxy)ethyl]-4-(5-methylpyridin-2-yl)piperidin-4-ol
1-[5-(2,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-4-(2-methoxyethoxy)piperidine
1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]ethan-1-one
naphthalen-1-yl (7S,9aR)-7-benzyl-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-1-(morpholin-4-yl)ethan-1-one
1-(2H-1,3-benzodioxol-5-ylmethyl)-3-[5-(benzylsulfanyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
4-[4-(4-chlorophenoxy)piperidine-1-carbonyl]-1-ethyl-1,2-dihydropyridin-2-one
N-[1-(2-methoxyethyl)-7-(4-methylpiperidine-1-carbonyl)-1H-1,3-benzodiazol-5-yl]cyclohexanecarboxamide
1-(3-cyanophenyl)-3-({1-[(4-methyl-1H-imidazol-5-yl)methyl]pyrrolidin-3-yl}methyl)urea
2-[3-benzyl-1-(2-methoxyphenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-(2-hydroxyethyl)-N-methylacetamide
diethyl({4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-5-phenylfuran-2-yl}methyl)amine
4-{[5-(1-cyclobutanecarbonylpiperidin-4-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}morpholine
6-[2-fluoro-3-(pyrrolidin-1-ylmethyl)phenoxy]pyridine-3-carboxamide
2-[2-(1-{2-[methyl(pyridin-3-ylmethyl)amino]acetyl}piperidin-4-yl)-1H-imidazol-1-yl]acetamide
3-methyl-N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}-1-propyl-1H-pyrazole-4-carboxamide
4-{1-[2-(cyclohexylcarbamoyl)ethyl]piperidin-3-yl}benzoic acid
[(1-cyclohexylpiperidin-3-yl)methyl]({[3-(1H-pyrazol-1-yl)phenyl]methyl})(pyridin-3-ylmethyl)amine
2-benzyl-4-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-3-methyl-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]benzamide
(2S,4R)-4-amino-1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-N-(propan-2-yl)pyrrolidine-2-carboxamide