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1-(4-fluoro-3-methylbenzoyl)-3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
2-(3-methoxypropanoyl)-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
(2E)-3-(pyridin-4-yl)-N-{[7-(1,3-thiazol-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}prop-2-enamide
2-(naphthalen-2-yloxy)-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}propanamide
1-[4-methyl-2-(4-methylpiperazin-1-yl)pyrimidine-5-carbonyl]azepan-4-amine
4-[2-(4-fluorophenyl)ethyl]-11-{methyl[(4-methyl-1,3-thiazol-2-yl)methyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
{[1-butyl-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}dimethylamine
5-(1-benzylpyrrolidin-2-yl)-3-cyclopropyl-1H-1,2,4-triazole
(4aR,7aS)-1-(1H-imidazol-2-ylmethyl)-4-(3-methylbut-2-enoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-({7-chloro-5-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-3-acetamidopropanamide
N-{[6-(3-chlorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-2-cyclopentyl-N-(2-methoxyethyl)acetamide
1-(1-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}ethyl)-1H-1,3-benzodiazole
3-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-1-(2,2,4,4-tetrafluoro-2,4-dihydro-1,3-benzodioxin-6-yl)urea
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-[(4-ethylphenyl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-2-(pyrrolidin-1-yl)-5,6,7,8-tetrahydroquinazoline-4-carboxamide
N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-2-(2-methoxyethyl)-N-methyl-1,3-benzoxazole-6-carboxamide
4-{4-[2-(3-fluorophenyl)acetamido]-1H-pyrazol-1-yl}-N-[3-(1H-pyrazol-1-yl)propyl]benzamide
5-(4-chlorophenyl)-N-[(1R)-1-(4-methoxyphenyl)ethyl]-1,2,4-triazin-3-amine
3-cyclopropyl-5-[3-(2-methylphenoxy)azetidine-1-carbonyl]-1H-pyrazole
2-(butylsulfanyl)-6-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}pyrimidin-4-amine
2-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-N-methylpyridine-3-carboxamide
2-{3-[(pyridin-3-yl)amino]propyl}-2,9-diazaspiro[5.5]undecan-3-one
7-fluoro-2-methyl-4-[(3R)-3-methylpiperazine-1-carbonyl]quinoline
2-(4-methyl-1,2,5-oxadiazol-3-yl)-1-[3-(3-methyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]ethan-1-one
4-(3-chlorophenyl)-3-[(propan-2-yloxy)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
3-({[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}(2-methoxyethyl)amino)-2,2-dimethylpropan-1-ol
(3R,4R)-3-cyclobutyl-4-methyl-1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)pyrrolidin-3-ol
1-{3-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-3-(2-methoxyphenyl)propan-1-one
N-benzyl-N-methyl-2-[({[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}amino)methyl]-2,3-dihydro-1H-inden-2-amine
2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-N-[3-(1H-1,2,3-triazol-1-yl)propyl]-1H-1,3-benzodiazole-5-carboxamide
1-{4-fluoro-2-[1-(thiophen-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]phenyl}-1H-pyrazole
(2-{4-[3-(2-chlorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-oxoethyl)urea
(3S,9aR)-8-[(5-chlorothiophen-2-yl)methyl]-3-(1H-indol-3-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-methyl-4-{2-[4-(methylsulfanyl)phenyl]ethyl}piperazine
5-({[3-(cyclohexylsulfanyl)propyl]carbamoyl}amino)-2-fluorobenzamide
3-benzoyl-1-(3-benzyl-1,2-oxazole-5-carbonyl)piperidine
1-(8-fluoro-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-3-methyl-3-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)urea
(1s,4s)-4-({methyl[3-(oxolan-2-yl)propyl]amino}methyl)cyclohexan-1-amine
(1R,5R)-6-[3-(2-fluorophenyl)-1H-pyrazole-5-carbonyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
methyl (2S,4S)-4-[2-(ethylamino)-4-methyl-1,3-thiazole-5-amido]-1-methylpyrrolidine-2-carboxylate
1-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]-2-{[(3,5-dimethylphenyl)methyl]sulfanyl}ethan-1-one
6-cyclopropyl-N-[cyclopropyl(3-methylpyridin-2-yl)methyl]pyrimidin-4-amine
methyl 2-({[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}(methyl)amino)acetate
[(3R,5R)-1-[6-(methoxymethyl)pyrimidin-4-yl]-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]methanol
(3S,4S)-3,4-dihydroxy-N-[4-(propan-2-yl)phenyl]piperidine-1-carboxamide
1-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]-2-(propan-2-yloxy)ethan-1-one
9-({2-[(propan-2-yl)amino]pyrimidin-5-yl}methyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
2-(1-{1-[(1r,4r)-4-methylcyclohexanecarbonyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)propan-2-ol
3-(5-methyl-1H-1,2,4-triazol-3-yl)-1-[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propan-1-one