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N-[(5-chloro-3-methyl-2-phenyl-1H-indol-7-yl)methyl]-1-ethyl-1H-pyrazole-5-carboxamide
5-(4-methyl-1,4-diazepan-1-yl)-2-[2-(morpholin-4-yl)ethyl]-2,3-dihydropyridazin-3-one
N-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl}-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
N-(2-methoxyethyl)-N-methyl-6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N6-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N5,N5-dimethyl-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[2-(6-methylpyridin-2-yl)ethyl]piperidine-3-carboxamide
1-[(3-{[3-(3-methylphenoxy)azetidin-1-yl]methyl}phenyl)methyl]-1H-pyrazole
4-(1-{4-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]phenyl}-1H-imidazol-2-yl)-2-(propan-2-yl)pyrimidine
3-benzyl-1-methyl-8-(thian-4-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-methoxy-N-({1-[(6-methylpyridin-2-yl)methyl]piperidin-3-yl}methyl)benzene-1-sulfonamide
1-(carbamoylmethyl)-N-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxamide
3-(benzyloxy)-1-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
4-(4-chlorophenyl)-N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}butanamide
methyl[(4-methyl-1H-imidazol-5-yl)methyl][(3-phenyl-1H-pyrazol-5-yl)methyl]amine
3-(benzyloxy)-1-{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
methyl (1S,3S,3aR,6aS)-5-ethyl-3-(4-hydroxyphenyl)-4,6-dioxo-1-phenyl-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
2-(3-fluoro-4-methoxybenzenesulfonyl)-2,8-diazaspiro[4.5]decane
6-[(dimethyl-1,2-oxazol-4-yl)methoxy]-1-[(3-methoxyphenyl)methyl]-4-[(4-methyl-1H-imidazol-5-yl)methyl]-1,4-diazepan-2-one
N-ethyl-1-[6-(4-ethylphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]pyrrolidine-3-carboxamide
ethyl 2-({[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}(methyl)amino)acetate
2-[({1-[(2,3-difluoro-6-methoxyphenyl)methyl]piperidin-4-yl}oxy)methyl]pyridine
2-[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]pyrimidin-4-amine
1-[3-fluoro-5-(trifluoromethyl)phenyl]-3-methyl-3-[2-(methylsulfanyl)ethyl]urea
2-{2-[2-(hydroxymethyl)-2,5-dihydro-1H-pyrrol-1-yl]-2-oxoethyl}-4-methyl-1,2-dihydrophthalazin-1-one
3-{3-[methyl(2-methylpropyl)amino]propyl}-8-[(2R)-pyrrolidine-2-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}quinoline-6-carboxamide
(1R,5R)-N,N-dimethyl-6-[2-(methylamino)pyridine-4-carbonyl]-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
1-(2-methylphenyl)-4-(1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperidin-3-yl)piperazine
N-({3-[(3-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)-2,3,4,9-tetrahydro-1H-carbazole-1-carboxamide
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-6-(2-methylpropyl)-2-oxo-1,2-dihydropyrimidine-4-carboxamide
1-[4-(dimethylamino)-5-methylpyrimidin-2-yl]-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-{[(3,4-difluorophenyl)methyl]amino}-1-(propan-2-yl)pyrrolidine-2-carboxamide
N3-(1,3-benzothiazol-2-ylmethyl)-1-cyclohexyl-N5-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
5-methyl-N-[2-(6-oxo-3-phenyl-1,4,5,6-tetrahydropyridazin-1-yl)ethyl]imidazo[1,2-a]pyridine-2-carboxamide
2-{2-[4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]pyrimidin-4-yl}pyridine-4-carboxylic acid
9-methoxy-4-[(4-methoxy-2,3-dimethylphenyl)methyl]-7-(6-methoxypyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-{1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]piperidin-4-yl}pyridine
4-{[2-(dimethylamino)ethyl]amino}-N-(2,2-dimethyloxan-4-yl)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
N,N-diethyl-1-[5-(3-fluorophenyl)-1,2,4-triazin-3-yl]pyrrolidin-3-amine
[1-(2-chloro-6-fluoro-3-methylbenzoyl)-3-(prop-2-en-1-yl)piperidin-3-yl]methanol
N-({5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}methyl)oxolane-2-carboxamide
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-1H-pyrazole-4-sulfonamide
1-[4-({[2-(4,6-dimethylpyrimidin-2-yl)ethyl]amino}methyl)-2-methoxyphenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
ethyl 2-[7-(2-cyclohexylacetyl)-2,7-diazaspiro[4.5]decan-2-yl]acetate
1-(difluoromethyl)-N-(2-methylpropyl)-N-(thiophen-3-ylmethyl)-1H-pyrazole-5-carboxamide
methyl 4-{[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}benzoate
N-ethyl-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-2-(naphthalen-1-yl)acetamide
N-[(2,4-dimethylphenyl)(pyridin-3-yl)methyl]-1H-1,2,4-triazole-5-carboxamide
({4-[3-cyclopropyl-1-(2-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]-1,3-thiazol-2-yl}methyl)dimethylamine
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N,1-dimethylpiperidine-4-carboxamide