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4-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-1-(3,5-dimethylphenyl)piperazin-2-one
4-fluoro-N-(2-{5-[(2-methoxyethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}ethyl)benzamide
1-(3-chlorophenyl)-4-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine
5-methoxy-3-({2-[2-(morpholin-4-yl)ethyl]piperidin-1-yl}methyl)-1H-indazole
4-chloro-N,N-diethyl-3-[3-(1-methylpiperidin-3-yl)propanamido]benzamide
4-({[5-fluoro-7-(4-fluoro-3-methylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}carbamoyl)pyridin-1-ium-1-olate
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-1-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
methyl({[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}){[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}amine
N-[2-(ethanesulfonyl)ethyl]-5-(2-methylpropyl)-1,2-oxazole-3-carboxamide
1-[6-(2-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-4-(2-methoxyethyl)piperazine
N-({7-[3-(2-methoxyphenyl)propanoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)furan-2-carboxamide
5-{4-[3-(morpholine-4-carbonyl)piperidin-1-yl]piperidine-1-carbonyl}pyrazin-2-ol
N-{2-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]-2-oxoethyl}methanesulfonamide
3-(4-acetyl-6-hydroxy-1,4-diazepan-1-yl)-N-(1,3-thiazol-2-yl)propanamide
ethyl 1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1H-imidazole-2-carboxylate
4-[(3aS,6aS)-octahydropyrrolo[3,4-b]pyrrol-5-yl]-1-{6-methylthieno[2,3-d]pyrimidin-4-yl}piperidine
2-cyclopentyl-9-[(4-ethylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
(3S,4R)-3-benzyl-1-[(5-ethylpyridin-2-yl)methyl]-4-methylpiperidin-4-ol
3-{2-[4-(3-methoxyphenyl)-3-oxopiperazin-1-yl]-2-oxoethyl}-1λ6-thiolane-1,1-dione
N-methyl-1-(6-methyl-2-propylpyrimidin-4-yl)-N-[3-(1H-pyrazol-1-yl)propyl]piperidin-4-amine
2-methoxy-6-[(4-{1-[(2-methoxyethyl)(pyridin-2-ylmethyl)amino]-2-phenylethyl}piperidin-1-yl)methyl]phenol
2-(propylsulfanyl)-1-[(1S,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
4-fluoro-N-(3-{9-methyl-3,9-diazaspiro[5.6]dodecan-3-yl}-3-oxopropyl)benzamide
2-(dimethylamino)-N-(2,4-dimethylphenyl)-4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carboxamide
N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-(2-phenylethyl)piperidin-3-amine
5-phenyl-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1,3,4-thiadiazol-2-amine
5-(2-methoxyethyl)-3-(4H-1,2,4-triazol-4-ylmethyl)-1,2,4-oxadiazole
9-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-[3-(1H-imidazol-1-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
N-{1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperidin-4-yl}pyridin-2-amine
{[1-(cyclohexylmethyl)-2-cyclopropylmethanesulfonyl-1H-imidazol-5-yl]methyl}(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
2-(dimethylamino)-8-[2-(2-methylphenyl)pyrimidin-5-yl]-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
3,6-dimethyl-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-1-benzofuran-2-carboxamide
N,N-dimethyl-2-{[4-(1H-1,2,3,4-tetrazol-1-yl)butanamido]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
N-(1-hydroxybutan-2-yl)-6-methyl-2-oxo-N-(pyridin-3-ylmethyl)-1,2-dihydropyridine-3-carboxamide
2-[(3-methoxyphenyl)methyl]-4-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}morpholine
N-[2-(5-methyl-4-{[2-(5-phenyl-4H-1,2,4-triazol-3-yl)acetamido]methyl}-1,3-oxazol-2-yl)phenyl]benzamide
(1S,5R)-6-(2-methoxyethyl)-3-[(4-phenylphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[3-chloro-4-(ethylcarbamoyl)phenyl]-4-(pyridin-4-yl)piperazine-1-carboxamide
[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]({[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl})amine
1-{3-[4-(3-chlorophenyl)piperazin-1-yl]piperidin-1-yl}-2-(methylsulfanyl)ethan-1-one
2-(1-{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}piperidin-2-yl)pyridine
(2R,6R)-4-(2-amino-2-methylpropanoyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
5-{[(1S,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}-N-propylpyrimidin-2-amine
ethyl 4-benzyl-1-[(2-methoxyphenyl)methyl]piperidine-4-carboxylate
1-(1,2,4-oxadiazol-3-ylmethyl)-N-[2-(pyridin-3-yloxy)phenyl]piperidine-3-carboxamide
ethyl 4-{[3-(naphthalen-1-yl)-1H-pyrazol-4-yl]methyl}piperazine-1-carboxylate
2-methyl-5-{4-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]piperazin-1-yl}-2,3-dihydropyridazin-3-one
(1S,5R)-3-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]acetamide