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8-{[4-(furan-2-yl)phenyl]methyl}-1-(2-methoxyethyl)-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-{[3-(dimethylamino)pyrrolidin-1-yl]methyl}-N,8-dimethyl-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
11-[(8-methoxyquinolin-2-yl)methyl]-3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecane
2-({4-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]phenyl}sulfanyl)ethan-1-ol
1-(5-ethyl-1,2-oxazole-3-carbonyl)-3-[2-(4-fluorophenyl)ethyl]piperidine
(3aS,6aS)-2-{3-fluoro-7-methylimidazo[1,2-a]pyridine-2-carbonyl}-5-propyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-{[(4-fluorophenyl)methyl]sulfanyl}-N-[(3R,4R)-3-hydroxypiperidin-4-yl]propanamide
(1R,7S)-3-[(3,4-dimethylphenyl)methyl]-6-(3-oxopiperazine-1-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
4-{2-[2-(4,5-dimethylfuran-2-yl)-1H-imidazol-1-yl]ethyl}pyridine
N-benzyl-N-(cyclobutylmethyl)-1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
2-(2-butoxy-5-methylphenyl)-6-(pyrrolidine-1-carbonyl)pyrazine
(3S,4R)-4-(2-methoxyphenyl)-1-(6-oxo-1,6-dihydropyridine-3-carbonyl)pyrrolidine-3-carboxylic acid
2-{3-[1-(oxan-2-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyrazine
2-[4-(2-ethylpyrimidine-5-carbonyl)-1-(furan-3-ylmethyl)piperazin-2-yl]ethan-1-ol
1-(4-cyclohexylphenyl)-3-(pyrimidin-4-ylmethyl)urea
6-ethyl-2-methyl-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}quinoline-4-carboxamide
N-(1-benzothiophen-5-ylmethyl)-1-(2-methoxyethyl)-6-oxopiperidine-3-carboxamide
1-cyclohexyl-4-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-1,4-diazepane
2-methoxy-6-({methyl[2-(morpholin-4-yl)propyl]amino}methyl)phenol
methyl 3-cyclobutaneamido-5-{[(2,3-dimethoxyphenyl)methyl]amino}-1-[2-(pyridin-2-yl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(2R,3R)-3-amino-1'-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-{4-[(2,3-dimethoxyphenyl)methyl]-1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-2-yl}ethan-1-ol
3-{[(1-ethyl-1H-pyrazol-4-yl)methyl]sulfamoyl}-N-[(2S)-1-methoxypropan-2-yl]benzamide
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-4-(piperidin-3-yl)benzamide
N4-methyl-N4-(1,3-thiazol-2-ylmethyl)-5,6,7,8-tetrahydroquinazoline-2,4-diamine
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-1,9-dioxaspiro[5.5]undecan-4-amine
3-ethoxy-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-4-(prop-2-en-1-yloxy)benzamide
4-methoxy-6-(3-{1-[(1-methyl-1H-imidazol-5-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyrimidine
4-({4-methyl-5-[1-(thiophen-2-ylmethyl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
2-{2-[2-(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)-1H-imidazol-1-yl]propyl}pyrazine
2-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-5-fluoropyridine
N-butyl-2-[N-methyl-1-(3,4,7-trimethyl-1H-indol-2-yl)formamido]acetamide
1-(pyridin-2-yl)-4-{[3-(trifluoromethyl)-1H-pyrazol-5-yl]methyl}piperazine
1-[6-methyl-3-(thiomorpholin-4-ylmethyl)quinolin-2-yl]piperidin-3-ol
N-[(3R,4S)-1-[(methylcarbamoyl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]-1-(4-methylphenyl)cyclopropane-1-carboxamide
4-(3-{4-[(4-chlorophenyl)methyl]piperazin-1-yl}-2,2-dimethylpropyl)morpholine
1-ethyl-5-(pyrrolidin-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
4-(1-benzyl-1H-imidazol-2-yl)-N-cyclohexylpiperidine-1-carboxamide
5-(3-{[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]methyl}phenyl)-1H-1,2,3,4-tetrazole
3-[1-(naphthalene-2-carbonyl)piperidin-3-yl]-1-(pyrrolidin-1-yl)propan-1-one
7-{2-[ethyl(3-methylphenyl)amino]ethyl}-2-oxa-7-azaspiro[4.5]decan-8-one
N5-(4-aminopyrimidin-2-yl)-N2-benzyl-N2,7,7-trimethyl-5,6,7,8-tetrahydroquinazoline-2,5-diamine
3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-{[4-(4-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}benzamide
3-{[2-(3-fluorophenyl)-2,3,4,5-tetrahydro-1,5-benzothiazepin-5-yl]methyl}-1,2-dihydroquinolin-2-one
N-{[1-(4-methoxyphenyl)cyclopentyl]methyl}-3-(4-methyl-1,3-thiazol-5-yl)propanamide
7-fluoro-4-[2-(thiophen-2-yl)azetidine-1-carbonyl]-1,2-dihydroquinolin-2-one
4-(3-hydroxy-3-methylbutyl)-N-[2-(4-methyl-1H-imidazol-2-yl)ethyl]benzamide
3-[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-1-[2-(2-methoxyethoxy)phenyl]urea
(2S,4S)-4-amino-N,N-diethyl-1-propylpyrrolidine-2-carboxamide
1-(cyclohexylmethyl)-N-[2-(5-methylthiophen-2-yl)ethyl]-6-oxopiperidine-3-carboxamide