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N-[3-(1,3-benzoxazol-2-yl)propyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-2-(2,3,6-trimethylphenoxy)ethan-1-one
1-(2,2-dimethylpropyl)-3-({[(4-fluorophenyl)methyl](methyl)amino}methyl)-3-hydroxypiperidin-2-one
2-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)-N-[(3S)-2-oxoazepan-3-yl]butanamide
N-(1-cycloheptylpiperidin-3-yl)-1-ethylpiperidine-4-carboxamide
(1-{1-[5-(ethylsulfanyl)thiophene-2-carbonyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methanamine
N-[2-(2-fluorophenyl)ethyl]-1-(methoxymethyl)cyclopropane-1-carboxamide
1-{5-methoxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
5-[2-(2H-1,3-benzodioxol-5-ylmethyl)propyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
[(3-chloropyridin-4-yl)methyl](ethyl)(oxan-2-ylmethyl)amine
(2S,4S)-4-amino-N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-1-methylpyrrolidine-2-carboxamide
N-ethyl-N-(2-hydroxyethyl)-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]acetamide
2-{[2-(ethylsulfanyl)ethyl]amino}-N-(pyrazin-2-yl)acetamide
3-(3-hydroxypiperidine-1-carbonyl)-4,6-dimethyl-1,2-dihydropyridin-2-one
5-ethyl-2,3-dimethyl-N-[2-(morpholin-4-yl)butyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]pyrazolo[1,5-a]pyridine-7-carboxamide
9-(3-ethyl-4,5-dihydro-1,2-oxazole-5-carbonyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
4,4,4-trifluoro-1-[(2R,6S)-6-phenyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]butan-1-one
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-2-propyl-1,3-thiazole-4-carboxamide
2-{1-butyl-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-5-yl}-5-methylpyrazine
methyl 1-ethoxy-2-oxo-8-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-1,8-diazaspiro[4.5]decane-4-carboxylate
(1R,7S)-N-methyl-4-oxo-3-(pentan-3-yl)-N-(pyrazin-2-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
2-[1-(4-methylpyrimidin-2-yl)pyrrolidin-3-yl]benzoic acid
N-methyl-2-(2-oxo-1,2,3,4-tetrahydroquinolin-1-yl)-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(2-methoxyethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-[4-(1-benzylpiperidin-4-yl)piperazin-1-yl]-2-[(4-methyl-1,3-thiazol-2-yl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
1-[4-(3-methoxybenzoyl)piperazin-1-yl]-2-(propan-2-ylsulfanyl)ethan-1-one
ethyl 2-[(3S,4S)-3-hydroxy-4-(morpholin-4-yl)pyrrolidin-1-yl]-1,3-oxazole-4-carboxylate
1-(2-methanesulfonylethyl)-4-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]piperazine
1-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-4-(1-methyl-1H-imidazol-2-yl)-1H-1,2,3-triazole
N-[(1-ethyl-1H-imidazol-5-yl)methyl]-2-{3-oxo-2-azatricyclo[6.3.1.04,12]dodeca-1(12),4,6,8,10-pentaen-2-yl}propanamide
methyl({[3-({1-[4-(1H-pyrazol-1-yl)benzoyl]piperidin-4-yl}oxy)phenyl]methyl})(quinolin-5-ylmethyl)amine
1-(1,3-oxazole-5-carbonyl)-4-[2-(piperidine-1-carbonyl)phenoxy]piperidine
5-{2-azabicyclo[2.2.1]heptane-2-carbonyl}-1-(cyclohexylmethyl)-4-oxo-N-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
N-[2-(dimethylamino)ethyl]-N,5-dimethyl-1-propyl-1H-pyrazole-4-carboxamide
2-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}pyridine-3-carbonitrile
2-methoxy-N-(1-{1-[(5-methylthiophen-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-phenylacetamide
N,4-dimethyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1H-imidazole-5-carboxamide
1-[(2-fluorophenyl)methyl]-5-{4-[(3-methoxyphenyl)methyl]piperazine-1-carbonyl}piperidin-2-one
2-(1-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-yl)ethan-1-ol
1-methyl-4-(2-{1-[(3-methylphenyl)methyl]-1H-1,2,4-triazol-5-yl}ethyl)-1,4-diazepane
3-[4-({3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-1H-pyrazol-1-yl]propanoic acid
6-(4-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)-9H-purine
1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
1-[2-(azepan-1-yl)ethyl]-3-(2-chloro-4-fluorophenyl)-1-methylurea
1-(3-{1,8-dioxa-4,11-diazaspiro[5.6]dodecane-4-carbonyl}phenyl)imidazolidin-2-one
3-{[4-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}pyridine
1-[(4-fluorophenyl)methyl]-4-[(2-hydroxyphenyl)methyl]piperazin-2-one
1-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-4-(4H-1,2,4-triazol-3-yl)piperidine
methyl 3-chloro-4-({[(1-propyl-1H-imidazol-2-yl)methyl]carbamoyl}amino)benzoate