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1-[3-(1H-indazol-1-yl)propyl]-3-[1-(propan-2-yl)-1H-pyrazol-4-yl]urea
3-(4-{5-[3-(methoxymethyl)piperidine-1-carbonyl]pyridin-2-yl}phenyl)propanoic acid
8-(1-benzofuran-5-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-(4-hydroxy-1,2-oxazolidin-2-yl)-2-(4-phenylpiperidin-1-yl)ethan-1-one
N-{2-[7-(2,6-dimethylhept-5-en-1-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-4-methylbenzamide
3-(2-ethylbutyl)-8-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-methyl-N-[(2-methylphenyl)methyl]-N-(oxolan-2-ylmethyl)-3-propyl-1H-pyrazole-5-carboxamide
(1S,5R)-3-[3-(2-methyl-1H-imidazol-1-yl)propyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-[(7R,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
(3E)-1-{4-[4-(thiomorpholin-4-ylmethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}pent-3-en-1-one
3-acetamido-N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]thiophene-2-carboxamide
8-[2-(pyridin-4-yl)acetyl]-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
methyl 3-[3-(aminomethyl)pyrrolidine-1-carbonyl]-5-(cyclobutylmethoxy)benzoate
6-[(diethylamino)methyl]-N-[(dimethyl-1,3-thiazol-5-yl)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-(2-aminoethyl)-N-(isoquinolin-5-ylmethyl)-N-methyl-1H-1,2,3-triazole-4-carboxamide
methyl 3-(2-chlorobenzenesulfonamido)-5-(pent-4-enamidomethyl)benzoate
(2S,4S)-4-amino-1-(2-amino-4-methyl-1,3-benzothiazole-6-carbonyl)-N,N-diethylpyrrolidine-2-carboxamide
1-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}cyclopropan-1-amine
1-[(3R,4S)-3-amino-4-(3-methoxyphenyl)pyrrolidin-1-yl]-2-(4-methyl-1,4-diazepan-1-yl)ethan-1-one
5-acetyl-N-({2-[benzyl(methyl)amino]-2,3-dihydro-1H-inden-2-yl}methyl)thiophene-2-carboxamide
1-(piperidin-1-yl)-2-(4-{[4-(pyridin-2-yl)phenyl]methyl}piperazin-1-yl)ethan-1-one
5-{[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-4-chloro-3-methyl-1H-pyrazole
5-({4-[benzyl(methyl)amino]-6-oxo-1,6-dihydropyridazin-1-yl}methyl)-N,N-dimethylfuran-2-carboxamide
4-(2-fluorophenyl)-2-[5-(propan-2-yl)-4-[4-(propan-2-yl)piperazine-1-carbonyl]-1H-pyrazol-1-yl]pyrimidine
(3S,4R)-4-methyl-1-(4-phenoxybutyl)piperidine-3,4-diol
1-cyclopentyl-4-(2,7,8-trimethylquinoline-4-carbonyl)piperazin-2-one
(1S,9aR)-1-{[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]methyl}-octahydro-1H-quinolizine
4-{2-[(4-methoxyphenyl)methyl]morpholine-4-carbonyl}pyridin-2-amine
N-[3-(3-methoxyphenyl)phenyl]-1-[(6-methylpyridin-2-yl)methyl]piperidine-4-carboxamide
1-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(2-ethyl-1H-imidazol-1-yl)ethan-1-one
[3-({1-[5-fluoro-4-(morpholin-4-yl)pyrimidin-2-yl]pyrrolidin-3-yl}methyl)phenyl]methanol
2-methyl-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
4-(7-chloro-4-hydroxyquinoline-3-carbonyl)piperazine-2-carboxylic acid
N-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-6-oxo-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
3-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]propan-1-one
[(2S,6S)-11-methoxy-4-{[2-(methylsulfanyl)phenyl]methyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
(3R,4S)-1-(1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)-4-(5-methylfuran-2-yl)pyrrolidin-3-amine
4-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-{imidazo[1,2-a]pyridin-3-ylmethyl}pyrimidin-2-amine
{[1-(2-methoxyethyl)-2-(3-methylbutanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)[1-(pyridin-2-yl)ethyl]amine
5-{1-[(3-fluorophenyl)methyl]-4-hydroxypiperidin-4-yl}-N-(2-methoxyphenyl)-1-benzofuran-2-carboxamide
2-[6-chloro-3-(thiomorpholin-4-ylmethyl)imidazo[1,2-a]pyridine-2-carbonyl]-1,2,3,4-tetrahydroisoquinoline
4-{1-[(4-chlorophenyl)methyl]pyrrolidin-3-yl}-1-(1H-pyrazole-4-carbonyl)piperidine
1-(4-{[2-(1-benzothiophen-2-yl)-1H-imidazol-1-yl]methyl}piperidin-1-yl)ethan-1-one
2-{[4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methyl}pyridine
(2E)-3-(2,3-difluorophenyl)-1-[3-(pyrimidin-4-yl)piperidin-1-yl]prop-2-en-1-one
1-[(3,5-dimethylphenyl)methyl]-4-[2-(propylsulfanyl)acetyl]piperazin-2-one
N-[(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)methyl]-3-(2-methoxyphenyl)propanamide
4-{[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]sulfonyl}-1-methyl-1H-imidazole
(3S,9aR)-8-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-(1H-indol-3-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-(3-chloro-4-methoxyphenyl)-3-{1-[2-(4-methylphenoxy)acetyl]piperidin-3-yl}propanamide