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N-{2-methoxy-5-[2-(2-methylpiperidin-1-yl)acetamido]phenyl}benzamide
3-ethyl-8-(pent-2-yn-1-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
7-methyl-2-(quinolin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
2-fluoro-N-[1-({[(1R,2S)-2-phenylcyclohexyl]carbamoyl}methyl)-1H-pyrazol-4-yl]benzamide
3-cycloheptyl-5-[(2-fluorophenyl)methyl]-5-(piperidin-4-yl)imidazolidine-2,4-dione
1-{3-[3-(2-phenylethyl)piperidine-1-carbonyl]phenyl}imidazolidin-2-one
N-ethyl-4-{6-[(2-hydroxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}benzamide
N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-N-methyl-2-propyl-1,3-thiazole-4-carboxamide
N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-3-(1H-1,2,4-triazol-1-yl)propanamide
1-(2-methylpyridin-4-yl)-4-{pyrazolo[1,5-a]pyridine-3-carbonyl}-1,4-diazepane
3-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-1-[2-(oxolan-2-ylmethoxy)phenyl]urea
2-(4-ethyl-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-[1-(3-methylpyridin-2-yl)propan-2-yl]acetamide
1-[3-(2-methylpyrimidin-4-yl)phenyl]-N-(pentan-2-yl)piperidin-4-amine
N-[2-(3-chlorophenyl)ethyl]-3-[(3S,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-(pyridin-2-ylmethyl)piperidin-3-yl]propanamide
1-[2-(4-chlorophenyl)ethyl]-N-(2-{imidazo[1,2-a]pyrimidin-2-yl}ethyl)-6-oxopiperidine-3-carboxamide
2-[3-(2-{[(3-methoxyphenyl)methyl]carbamoyl}ethyl)piperidin-1-yl]pyridine-3-carboxamide
N-{3-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-3-oxopropyl}-4-methylbenzamide
(2S,4S)-1-(cyclohexylmethyl)-N-[(4-methylphenyl)methyl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
1-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-5-oxopyrrolidine-3-carboxylic acid
6-fluoro-4-methyl-2-(2-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine-1-carbonyl}pyrrolidin-1-yl)quinazoline
1-methyl-4-[2-(trifluoromethyl)morpholine-4-carbonyl]-1,2-dihydroquinolin-2-one
methyl 3-[(2-fluoro-4-methoxyphenyl)methyl]-9-[(1-methyl-5-oxopyrrolidin-3-yl)methoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-phenoxy-5-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)pyridine
1-[1-(benzenesulfonyl)cyclopropanecarbonyl]-4-(4-ethyl-1H-pyrazol-5-yl)piperidine
6-[1-(8-chloroquinoline-2-carbonyl)piperidin-3-yl]pyrimidin-4-ol
3-chloro-4-[(1-cyclobutanecarbonylpiperidin-4-yl)oxy]-N-cyclopentylbenzamide
3-(3-hydroxyquinoxalin-2-yl)-1-[2-(pyridin-2-yl)pyrrolidin-1-yl]propan-1-one
methyl 2-chloro-5-[({[5-(2-methoxyethyl)-1,2,4-oxadiazol-3-yl]methyl}carbamoyl)amino]benzoate
3-[5-(1-ethylpiperidin-3-yl)-4-phenyl-1H-imidazol-1-yl]propan-1-ol
2-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-3-(piperidine-1-carbonyl)pyrazine
1-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]-4-(pyridin-4-yl)piperazine
3-{3-[3-(aminomethyl)pyrrolidine-1-carbonyl]phenyl}-2H-chromen-2-one
2-(2-hydroxypropyl)-9-[(4-methoxy-3-methylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
1-ethyl-2-methyl-5-{[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]methoxy}-1H-1,3-benzodiazole
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-{2-[(3-methylpyridin-4-yl)amino]ethyl}benzamide
1-{4-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-3,5-dimethyl-1H-pyrrol-2-yl}ethan-1-one
2-[2-({3-[(3,4-dimethoxyphenyl)amino]piperidin-1-yl}methyl)phenoxy]ethan-1-ol
(1R,5R)-6-(cyclopropylmethyl)-3-(5-methanesulfonyl-2-methylpyrimidin-4-yl)-3,6-diazabicyclo[3.2.2]nonane
N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-3-(4,5,6,7-tetrahydro-2H-indazol-3-yl)propanamide
2-[(3-{[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]sulfamoyl}phenyl)formamido]-N,N-dimethylacetamide
1-(cyclopropylmethyl)-4-{[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
methyl 1-{2-[1-cyclopentyl-3-(3-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]acetyl}piperidine-2-carboxylate
1-cyclohexyl-5-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-N-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
N-({7-chloro-5-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-1-methylcyclopropane-1-carboxamide
4-(4-aminopyrimidin-2-yl)-9-ethyl-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
4-[5-({[(1R,2R,4S)-bicyclo[2.2.1]heptan-2-yl]amino}methyl)-1,2,4-oxadiazol-3-yl]benzoic acid
2-(1,2-benzoxazol-3-yl)-1-[4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]ethan-1-one
N-ethyl-N-(oxan-4-yl)-2-oxo-1,2-dihydroquinoline-4-carboxamide
5-{[(5-methoxy-1-methyl-1H-indol-2-yl)formamido]methyl}thiophene-2-carboxylic acid
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-2,3-dihydro-1-benzofuran-7-carboxamide