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4-fluoro-N-({3-methoxy-4-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]benzene-1-sulfonamide
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-6-(morpholin-4-yl)pyrimidin-4-amine
3-(2-{3-[benzyl(methyl)amino]piperidin-1-yl}-2-oxoethyl)-1,2,3-oxadiazol-3-ium-5-olate
3-chloro-5-(4-methyl-3-phenylpiperazine-1-carbonyl)-1,2-dihydropyridin-2-one
1-ethyl-5-{[4-(thian-4-yl)piperazin-1-yl]methyl}-1H-indole
3-(oxolan-2-ylmethyl)-3-(thiophen-3-ylmethyl)-1-[3-(4H-1,2,4-triazol-4-yl)phenyl]urea
N-[(3R,4S)-4-cyclopropyl-1-(3-methylpyrazin-2-yl)pyrrolidin-3-yl]-2-(2,4-dioxoimidazolidin-1-yl)acetamide
4-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
4-{1-[1-(methoxymethyl)cyclobutanecarbonyl]piperidin-3-yl}-2-methyl-6-(pyrrolidin-1-yl)pyrimidine
(2E)-1-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidin-1-yl]-3-phenylprop-2-en-1-one
2-(3,4-dimethoxyphenyl)-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]acetamide
N3-benzyl-1-cyclopropyl-N5-(naphthalen-1-ylmethyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2,6-dimethyl-5-{[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-3,4-dihydropyrimidin-4-one
4-{6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-2-ethyl-1-(propan-2-yl)piperazine
6-(methoxymethyl)-2-[4-({methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
ethyl 3-benzyl-1-(3-acetamidobenzenesulfonyl)piperidine-3-carboxylate
3-{5-[4-(thiophen-2-yl)butanoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
1-(2,3-dihydro-1H-inden-2-yl)-3-(ethoxymethyl)-5-(oxolan-3-yl)-1H-1,2,4-triazole
1-{3-[benzyl(methyl)amino]piperidin-1-yl}-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
1-ethyl-N-(pyridin-4-ylmethyl)-5-[(thiophen-2-ylmethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-{[4-(pyrimidin-2-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}ethan-1-ol
N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}-3,5-dimethyl-1,2-oxazole-4-sulfonamide
(2,3-dihydro-1-benzofuran-5-ylmethyl)[2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl]amine
N-[(3-chlorophenyl)methyl]-3,5-dimethyl-1-benzofuran-2-carboxamide
2-{4-[6-(4-methyl-1H-pyrazol-1-yl)pyrimidin-4-yl]-1H-pyrazol-1-yl}-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
1-(3-{[(dicyclopropylmethyl)amino]methyl}phenoxy)-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-[3-(aminomethyl)pyrrolidine-1-carbonyl]-2-(4-tert-butylphenoxymethyl)pyrimidin-4-ol
N-benzyl-N-methyl-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
5-[3-(methoxymethyl)piperidine-1-carbonyl]-N-[2-(6-methylpyridin-2-yl)ethyl]pyridin-2-amine
(3S,4R)-1-(2,5-dimethylfuran-3-carbonyl)-4-(4-methoxyphenyl)-N,N-dimethylpyrrolidin-3-amine
1-methyl-4-({5-[3-(thiophen-2-yl)propyl]-1,2,4-oxadiazol-3-yl}methyl)piperazine
N-[2-(1H-pyrazol-4-yl)ethyl]-2-[4-(trifluoromethyl)phenyl]-1,3-thiazole-4-carboxamide
6-(2-fluoro-4-methoxyphenyl)-N-[2-(1H-imidazol-4-yl)ethyl]-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
5-(8-methoxyquinolin-5-yl)pyrazin-2-amine
{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}[2-(1H-pyrazol-4-yl)ethyl]amine
N-[3-(2-oxopyrrolidin-1-yl)phenyl]-1H-indazole-3-carboxamide
1-(carbamoylmethyl)-N-{3-[(pyridin-3-yl)amino]propyl}piperidine-3-carboxamide
N-[4-(3-fluorophenyl)phenyl]-1-[(2-methyl-1H-imidazol-4-yl)methyl]pyrrolidine-2-carboxamide
N-cyclopropyl-4-methoxy-3-({[2-(5-methylfuran-2-yl)ethyl]carbamoyl}amino)benzamide
N'-(2,3-dimethylphenyl)-N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]propanediamide
N-(2H-1,3-benzodioxol-4-ylmethyl)-N-[(4-ethoxyphenyl)methyl]cyclopropanamine
(1S,5R)-6-benzyl-3-[3-(thiophen-2-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{[3-(benzyloxy)phenyl]methyl}-4-(2-methoxyethyl)-1,4-diazepan-5-one
8-methoxy-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-amine
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-1,3,5-trimethyl-1H-pyrazole-4-sulfonamide
4,5,6,7-tetramethyl-2-[1-(piperidin-4-yl)-1H-1,2,3-triazol-4-yl]-1H-1,3-benzodiazole
(2,3-dihydro-1-benzofuran-5-ylmethyl)(methyl)[1-(pyridin-2-yl)propan-2-yl]amine
(1S,5R)-1,3,3-trimethyl-N-[4-(1H-1,2,4-triazol-1-yl)phenyl]-6-azabicyclo[3.2.1]octane-6-carboxamide