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2-(2-chlorophenyl)-1-[4-hydroxy-4-(hydroxymethyl)azepan-1-yl]ethan-1-one
(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-[(4-hydroxyphenyl)methyl]piperidin-3-ol
1-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]methyl}-4-(4-methyl-1H-pyrazol-3-yl)piperidine
3-(azepan-1-ylmethyl)-6,7-dimethoxy-1,2-dihydroquinolin-2-one
4-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]phenol
ethyl 5-({[3-(2-oxopyrrolidin-1-yl)propyl]amino}methyl)-1-(4-phenyl-1,3-thiazol-2-yl)-1H-pyrazole-4-carboxylate
N-[1-(3-chlorophenyl)cyclopropyl]-3-(2,5-dioxoimidazolidin-4-yl)propanamide
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-[5-(phenoxymethyl)-1H-pyrazole-3-carbonyl]piperazine
2-[3-(isoquinolin-5-yl)phenoxy]propanamide
1-[7-(2-cyclohexylethyl)-2,7-diazaspiro[4.5]decan-2-yl]-3-(dimethyl-1,2-oxazol-4-yl)propan-1-one
(3R,4R)-1-(4-chloro-2-methoxybenzoyl)-3,4-dimethylpyrrolidin-3-ol
4-cyclobutyl-N,6-dimethyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}pyrimidin-2-amine
1-cyclohexyl-3-(cyclopropylmethyl)-5-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-{2-[5-(2,6-dimethylphenyl)-4-phenyl-1H-imidazol-1-yl]ethyl}acetamide
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)-1H-indazole-3-carboxamide
2-{4-[1-(oxan-4-yl)piperidine-3-carbonyl]piperazin-1-yl}pyrazine
3-(azepane-1-carbonyl)-N-cycloheptyl-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-ethyl-4-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}piperazine-2,3-dione
2-cyclopentyl-7-[(3,4-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
1-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-3-yl]-2-(pyridin-2-ylsulfanyl)ethan-1-one
1-benzyl-N-ethyl-4-oxo-5-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-1,4-dihydropyridine-3-carboxamide
(3S,4R)-4-(2-methylphenyl)-1-(1-methylpiperidin-4-yl)pyrrolidine-3-carboxylic acid
3-fluoro-N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methylimidazo[1,2-a]pyridine-2-carboxamide
N-({7-chloro-5-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)oxolane-3-carboxamide
N-(pyridin-3-ylmethyl)-3-(1-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)propanamide
2-amino-6-(furan-2-yl)-4-[5-(oxan-2-yl)furan-2-yl]pyridine-3-carbonitrile
3-[4-(thiophen-2-yl)-1H-imidazol-1-yl]pyridin-4-amine
3-[7-(2-cyclohexylethyl)-2,7-diazaspiro[4.5]decane-2-carbonyl]-5,6-dimethyl-1,2-dihydropyridin-2-one
4-(7-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl)morpholine
N-ethyl-N-(2-hydroxyethyl)-1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carboxamide
5-methyl-N-[3-(4-methylbenzenesulfonamido)propyl]-1,2-oxazole-3-carboxamide
(2R,6S)-6-phenyl-2-(prop-2-en-1-yl)-1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}-1,2,3,6-tetrahydropyridine
N-[(1-methylpiperidin-3-yl)methyl]-4-(1H-pyrazol-3-yl)benzamide
1-[2-(3-chlorophenoxy)ethyl]-1-methyl-3-[1-(2-methylpropyl)-1H-pyrazol-5-yl]urea
methyl 5-cyano-6-[(3S,4R)-3-acetamido-4-(propan-2-yl)pyrrolidin-1-yl]-2-methylpyridine-3-carboxylate
5-(2-oxo-2-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl}ethyl)imidazolidine-2,4-dione
1-[(1-cyclopentyl-1H-imidazol-5-yl)methyl]-2-(4-fluorophenyl)piperidine
3-[(4-ethylpiperazin-1-yl)methyl]-3-hydroxy-1-(3-phenylpropyl)piperidin-2-one
6-(2-fluoro-4-methoxyphenyl)-N-(2-methoxyethyl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-[(3R,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-chlorobenzamide
4-ethyl-3-(1-{[4-(propan-2-yl)phenyl]methyl}piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(1,3-dimethyl-1H-pyrazol-5-yl)-2-[3-(4-fluorophenyl)-1H-pyrazol-1-yl]acetamide
6-(1-{[2-(butylsulfanyl)pyrimidin-5-yl]methyl}piperidin-4-yl)-2-methylpyrimidin-4-ol
8-[2-(3-chlorophenyl)-2-hydroxyacetyl]-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
3-({[1-(1-tert-butyl-1H-pyrrole-3-carbonyl)piperidin-3-yl]oxy}methyl)pyridine
(3aR,6aR)-2-methyl-N-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
1-tert-butyl-5-oxo-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidine-3-carboxamide
7-fluoro-3-methyl-N-[1-(1-methyl-1H-imidazol-2-yl)butyl]-1-benzofuran-2-carboxamide
N-[1-(cyclohex-1-en-1-yl)ethyl]-3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)propanamide
[(2S,4R,5R)-4-({[(5-ethylfuran-2-yl)methyl]amino}methyl)-5-(2-fluorophenyl)-1-methylpyrrolidin-2-yl]methanol