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3-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1H-indazole
N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-1-benzothiophene-2-carboxamide
3-[6-amino-2-(butylsulfanyl)pyrimidin-4-yl]-3,9-diazaspiro[5.6]dodecan-10-one
4-[(3S)-3-aminopyrrolidine-1-carbonyl]-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]benzene-1-sulfonamide
N-methyl-2-({[2-(propylsulfanyl)pyrimidin-5-yl]methyl}amino)ethane-1-sulfonamide
2-(2,4-dichlorophenoxy)-N-{[4-(dimethylamino)oxan-4-yl]methyl}acetamide
3-(2-fluorophenyl)-N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-3-phenylpropanamide
2-{4-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]phenyl}-N-methylacetamide
N-[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4,4,4-trifluorobutanamide
2-(2,4-dichlorophenoxy)-N-(2-oxopyrrolidin-3-yl)acetamide
2-{4-[(2-chloro-4-fluorophenyl)methyl]-1-(2-phenylethyl)piperazin-2-yl}ethan-1-ol
1-ethyl-8-{imidazo[1,2-a]pyridine-6-carbonyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-methoxy-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
2-[4-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-1-(thiophen-2-ylmethyl)piperazin-2-yl]ethan-1-ol
(3S,4R)-1-(2-amino-2-methylpropanoyl)-4-(2,3-dimethoxyphenyl)pyrrolidine-3-carboxylic acid
1-(2-benzylmorpholin-4-yl)-3-(thiophen-3-yl)propan-1-one
1-(4,6-dimethoxypyrimidin-2-yl)-4-hydroxypiperidine-4-carboxylic acid
(1R,5R)-6-(2-methoxypyridine-3-carbonyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2-{4-[(2-aminopyrimidin-5-yl)methyl]-1-[(4-methoxy-3-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
2-(dimethylamino)-N-[1-(3-methylbutanoyl)piperidin-4-yl]-2-(4-methylphenyl)acetamide
N-ethyl-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-2-(2-oxopiperidin-1-yl)acetamide
1-{2-[4-(hydroxymethyl)piperidin-1-yl]-5,6,7,8-tetrahydroquinazolin-5-yl}-3-(propan-2-yl)urea
N-[2-(4-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-1-methyl-1H-indole-4-carboxamide
2-(4-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-1-methylpiperazin-2-yl)ethan-1-ol
3-{[({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)amino]methyl}piperidin-3-ol
3-{3-[(2H-1,3-benzodioxol-5-yl)amino]piperidine-1-carbonyl}-6-methyl-1,2-dihydropyridin-2-one
4-methyl-2-(propan-2-yl)-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1,3-thiazole-5-carboxamide
1-(4-carboxy-1,3-oxazol-2-yl)-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylic acid
4-(benzyloxy)-1-{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}piperidine
N-[1-(4-ethoxy-3-fluorophenyl)ethyl]-2-(2-oxopiperidin-1-yl)acetamide
3-(3-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}propyl)-1H-indole
N-(2,3-dihydro-1H-inden-2-yl)-N-methyl-3-oxo-3,4-dihydroquinoxaline-2-carboxamide
2-methyl-1-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}-1H-1,3-benzodiazole
(3aS,6aR)-5-(2,3-dihydro-1-benzofuran-5-ylmethyl)-3-[2-(4-fluorophenyl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
8-(2-amino-6-methoxypyrimidin-4-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(oxolan-3-ylmethyl)cyclopropanamine
N-[(2S,4R,6S)-2-ethyl-6-(2-methylnaphthalen-1-yl)oxan-4-yl]acetamide
2-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-4-(2,6-dimethylpyridin-3-yl)pyrimidine
N-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-1-methyl-N-(2-phenylethyl)piperidin-4-amine
N-[(1-methylpiperidin-3-yl)methyl]-N-(2-phenylethyl)pent-4-enamide
[(4-ethyl-5-{1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
1-ethyl-8-(1H-indol-2-ylmethyl)-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N1,N1-dimethyl-N3-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-1,3-dicarboxamide
3,6,7-trimethyl-N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-1-benzofuran-2-carboxamide
3-fluoro-2-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}pyridine
N,2-dimethyl-N-[3-(oxolan-2-yl)propyl]thieno[2,3-d]pyrimidin-4-amine
N-[(3R,5S)-1-[(4-fluoro-3-methylphenyl)methyl]-5-(methylcarbamoyl)pyrrolidin-3-yl]-1-methyl-1H-imidazole-5-carboxamide
2-ethyl-1-{3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}butan-1-one
2-[methyl(pyridin-3-ylmethyl)amino]-1-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethan-1-one
2-[1-(1-cyclopropanecarbonylpiperidin-4-yl)-1H-1,2,3-triazol-4-yl]propan-2-ol