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(2S)-2-amino-4-[1-(cyclohexylmethyl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]butanoic acid
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-3-(3-hydroxy-3-methylbutyl)benzamide
N2-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-N1-(3-methylpyridin-4-yl)ethane-1,2-diamine
2-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-6-methylpyridine-3-carboxamide
9-[2-(2,5-difluorophenyl)acetyl]-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
3-(4-chlorobenzoyl)-1-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidine
2-ethyl-1-{4-[(2-methylprop-2-en-1-yl)oxy]benzoyl}pyrrolidine
6-(4-methoxyphenyl)-9-(thian-4-yl)-6,9-diazaspiro[4.5]decan-7-one
2-(5-acetylthiophen-3-yl)-1-[4-(furan-2-carbonyl)-1,4-diazepan-1-yl]ethan-1-one
5-[3-(diethylamino)pyrrolidine-1-carbonyl]-N-(propan-2-yl)pyrimidin-2-amine
1-(3-fluorophenyl)-3-(1-{1-[2-(2-oxopyrrolidin-1-yl)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
1-[(6-chloropyridin-3-yl)methyl]-4-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}piperazine
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-2-fluoro-N-methyl-5-sulfamoylbenzamide
1-{1-[(2,3-difluorophenyl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
1-{[(3R,4R)-1-{[6-(dimethylamino)pyridin-3-yl]methyl}-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}piperidin-4-ol
1-cyclopropanecarbonyl-4-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}piperidine
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-6-methylpyridine-3-carboxamide
1-[(3aR,5S,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]-2-(2-amino-4,6-dimethylpyrimidin-5-yl)ethan-1-one
4-cyclobutaneamido-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]benzamide
3-{[3-(azepan-1-yl)-2-hydroxypropyl]sulfamoyl}-N-(propan-2-yl)benzamide
N-(1-{7-[2-(cyclohex-1-en-1-yl)acetyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)propanamide
5-[2-(dimethylamino)-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
(3S,4R)-1-{[2-(2-methoxyphenyl)pyrimidin-5-yl]methyl}-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
3-[2-(4-methoxyphenyl)ethyl]-5-methyl-5-{1-[3-(pyridin-3-yl)propanoyl]piperidin-4-yl}imidazolidine-2,4-dione
2-ethyl-4-methyl-N-[4-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]-1,3-oxazole-5-carboxamide
2-cyclopropyl-8-[6-methyl-2-(propan-2-yl)pyrimidin-4-yl]-2,8-diazaspiro[5.5]undecan-3-one
6-(aminomethyl)-2-methyl-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}pyrimidin-4-amine
3-[(3R,4S)-1-(4-chloro-2-methylbenzoyl)-4-(dimethylamino)piperidin-3-yl]propan-1-ol
1-(diethylamino)-3-(2-methoxy-5-{[4-(pyridin-3-yloxy)piperidin-1-yl]methyl}phenoxy)propan-2-ol
2-(4-cyclobutyl-6-methylpyrimidin-2-yl)benzamide
N-{2H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-ethyl-N-methyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
2-amino-6-cyclobutyl-4-(2,6-dimethoxyphenyl)pyridine-3-carbonitrile
2-({1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]piperidin-4-yl}oxy)pyrimidine
(1R,3S)-3-methoxy-7-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}-7-azaspiro[3.5]nonan-1-ol
4-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazine-1-carbonyl]-2-(pyrrolidin-1-yl)-5,6,7,8-tetrahydroquinazoline
1-ethyl-4-[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]pyrrolidin-2-one
1-(2-chlorobenzenesulfonyl)-2-(3-methoxypropyl)piperidine
1-(1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-4-phenylpiperidin-4-yl)ethan-1-one
4,5-dimethyl-6-[4-(pyridin-4-ylmethyl)piperazin-1-yl]pyrimidine
ethyl({[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl})(oxolan-2-ylmethyl)amine
1-({4-methyl-5-[1-(pyridin-4-ylmethyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]propan-1-one
1-(piperidin-1-yl)-3-[2-({[2-(pyridin-4-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
1-(cyclohexylmethyl)-N-(2-methoxyethyl)-6-oxo-N-(pyridin-4-ylmethyl)piperidine-3-carboxamide
5-(3-acetylphenoxymethyl)-N-(2-hydroxypropyl)-1H-pyrazole-3-carboxamide
4-{3-[(2,6-difluorophenyl)methyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl}piperazin-2-one
4-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]butanamide
4-{4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-methylpyridine
3-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]-1-[4-(propylsulfanyl)phenyl]urea
4-[3-(furan-2-yl)-1H-pyrazol-1-yl]-1-(1,3-thiazol-2-yl)piperidine-4-carboxylic acid