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N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
5-chloro-6-{4-[(4-methylphenyl)methyl]-3-oxopiperazin-1-yl}pyridine-3-carboxylic acid
(1-{[1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methanol
1-(pyridin-2-yl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]piperidine-3-carboxamide
3-(2-chlorophenyl)-N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-5-methyl-1,2-oxazole-4-carboxamide
3-(1-{4-[(methylcarbamoyl)methyl]phenyl}-1H-imidazol-2-yl)benzoic acid
N-({2-[benzyl(methyl)amino]-2,3-dihydro-1H-inden-2-yl}methyl)-4,4,4-trifluorobutanamide
N-[1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]cyclobutanecarboxamide
6-[2-chloro-4-(pyrrolidin-1-ylmethyl)phenoxy]pyridine-3-carbonitrile
methyl[(3-methyl-1,2-oxazol-5-yl)methyl]{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}amine
1-[(4-chlorophenyl)methyl]-N-(pyridin-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
5-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-3,4-dihydropyrimidin-4-one
N-{[5-methyl-7-(2-methylquinolin-6-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}pyrazolo[1,5-a]pyrimidine-2-carboxamide
6-[2-(aminomethyl)-5-fluoro-2,3-dihydro-1-benzofuran-7-yl]-N-cyclopentylpyridazin-3-amine
N-(2-{1-[(4,6-dimethylpyrimidin-2-yl)methyl]piperidin-2-yl}ethyl)acetamide
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-1-(3-hydroxyphenyl)-N-methyl-5-oxopyrrolidine-3-carboxamide
2-(3-{3-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-4-yl]phenyl}-1H-pyrazol-1-yl)ethan-1-ol
2-(2-methyl-1,3-thiazol-4-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)acetamide
1-(1-cyclopropylethyl)-5-(2-fluoro-6-methoxyphenyl)-3-methyl-1H,4H-pyrazolo[3,4-d]imidazole
6-fluoro-N-methyl-2-(1-methyl-1H-pyrazol-4-yl)-N-[2-(1H-pyrazol-1-yl)ethyl]quinoline-4-carboxamide
3-(3-hydroxy-3-methylbutyl)-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]benzamide
N-butyl-3-(4-methylpiperazine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-[4-(3-methoxypropyl)piperazine-1-carbonyl]-1-(pyridin-4-ylmethyl)pyrrolidin-2-one
3-[1-(6-amino-5-methylpyridin-3-yl)-1H-1,3-benzodiazol-2-yl]propanoic acid
N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
2-(2,3-difluoro-4-methylphenyl)-1-(prop-2-en-1-yl)-1H-imidazole
3-{[(2-chloro-3,4-dimethoxyphenyl)methyl]amino}-N-cyclopentyl-5-(phenylsulfamoyl)benzamide
2-methyl-5-[2-(3-methyl-1H-pyrazol-4-yl)phenyl]-1,3,4-thiadiazole
1-{3-[4-(adamantan-1-yl)piperazin-1-yl]-3-oxopropyl}-1,2-dihydropyridin-2-one
N-cycloheptyl-2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}acetamide
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-N-methyl-2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetamide
N-[(4-methoxypyridin-2-yl)methyl]-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetamide
1-phenyl-N-[(1-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}piperidin-3-yl)methyl]methanesulfonamide
3-(1H-1,3-benzodiazol-1-yl)-1-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]propan-1-one
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-6-oxo-1-(2-phenylethyl)piperidine-3-carboxamide
N-ethyl-N-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-2,2-dimethyloxan-4-amine
(4aS,8aR)-6-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-1-(3-methylbutyl)-decahydro-1,6-naphthyridin-2-one
4-(2-methoxyphenoxy)-1-(3-methoxypyrazin-2-yl)piperidine-4-carboxylic acid
(2S)-N-[1-benzyl-6-(propan-2-yloxy)-1H-indazol-3-yl]-6-oxopiperidine-2-carboxamide
N5,N5-dimethyl-N6-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
(3aS,7aR)-2-[3-(3-hydroxy-3-methylbutyl)benzoyl]-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
8-(2-methoxy-2-methylpropanoyl)-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
1-butyl-5-(2-{[(3-methoxyphenyl)methyl]amino}ethyl)pyrrolidin-2-one
2-{2-[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-2-oxoethyl}-6-methyl-2,3-dihydropyridazin-3-one
4-{1-[2-(pyrrolidin-1-yl)benzoyl]piperidin-3-yl}benzoic acid
N-{3-[methyl(phenyl)amino]propyl}-[1,2,4]triazolo[4,3-a]pyridine-7-carboxamide
N-[(4-fluorophenyl)methyl]-1-methyl-5-[(pyridin-3-ylmethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
5-[3-(4-fluorophenoxymethyl)piperidine-1-carbonyl]-1H-1,3-benzodiazole
2-[3-(1-benzofuran-2-yl)-1H-pyrazol-1-yl]-N-(2-ethyl-2H-1,2,3-triazol-4-yl)acetamide
5-({[(1-ethyl-1H-pyrazol-4-yl)methyl](methyl)carbamoyl}amino)-2-methoxy-N-methylbenzamide