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2-[2-ethoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]-5-(trifluoromethyl)pyridine
2-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decan-4-ylmethyl]benzoic acid
3-[(3R,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]-N-(1,3-thiazol-2-yl)propanamide
methyl 2-(2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamido)acetate
5-{2-[(2-methylprop-2-en-1-yl)oxy]benzoyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonitrile
ethyl 1-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-4-(3-phenylpropyl)piperidine-4-carboxylate
3-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]-1-[3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]urea
(3R,5S)-1-(2-methylpropyl)-5-(morpholin-4-ylmethyl)-N-(oxolan-2-ylmethyl)piperidine-3-carboxamide
2-{[2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]methyl}-1H-1,3-benzodiazole
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-3-(benzylsulfanyl)propan-1-one
N-{[7-(1,3-benzothiazol-2-yl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-5-(methoxymethyl)furan-2-carboxamide
1-{2-[3-(pyridin-3-yl)azetidin-1-yl]pyrimidin-4-yl}pyrrolidin-3-ol
1-(3-methylpyridin-2-yl)-4-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)piperazine
5-{[4-(4-methoxyphenyl)-2-methylpiperazin-1-yl]methyl}-2,1,3-benzothiadiazole
N,N-dimethyl-2-[(1S,5R)-7-oxo-3-(1-phenylcyclopropanecarbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
4-[7-(5-cyclopropyl-1,2-oxazole-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]morpholine
1-{2-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-2-oxoethyl}azepan-2-one
N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carboxamide
3-{2-[(4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
7-methyl-2-[2-(methylsulfanyl)propyl]-1H-1,3-benzodiazole
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-2-(7-fluoro-2-methyl-1H-indol-3-yl)acetamide
4-methoxy-N-(2-methoxyethyl)-2-[(1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidin-4-yl)oxy]benzamide
5-cyclopropanecarbonyl-1'-[(2,3-difluorophenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-{4-[(4-methyl-1H-pyrazol-1-yl)methyl]piperidine-1-carbonyl}-6-phenyl-1,2-dihydropyridin-2-one
1-(4-aminopyrimidin-2-yl)-4-(thiophene-3-carbonyl)-1,4-diazepane-6-carboxylic acid
N2-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-5-fluoro-N4,N4-dimethylpyrimidine-2,4-diamine
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylspiro[2.5]octane-1-carboxamide
(2R,6R)-11-methoxy-4-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-cyclobutyl-3-(2-hydroxyphenyl)-3-(4-hydroxyphenyl)propanamide
N-(2-methoxyethyl)-3-{octahydro-1H-pyrido[1,2-a]piperazine-2-sulfonyl}benzamide
1-(1-methyl-1H-imidazole-2-carbonyl)-3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
4-cyclobutyl-6-methyl-2-{3-methyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}pyrimidine
N-(1,3-benzoxazol-2-ylmethyl)-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
(3R,4R)-1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-ol
3-chloro-N-[2-(dimethylamino)ethyl]-4-{[1-(2-hydroxypropanoyl)piperidin-4-yl]oxy}benzamide
3-(3-methyl-1-phenyl-1H-pyrazol-5-yl)-1-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}urea
(3S,4S)-4-cyclopropyl-1-[2-(1H-1,2,4-triazol-1-yl)benzoyl]pyrrolidine-3-carboxylic acid
4-[2,2-dimethyl-3-(4-methyl-3-phenylpiperazin-1-yl)propyl]morpholine
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-ethyl-N-methylacetamide
N-cyclopropyl-5-{[4-(dimethylamino)phenyl]methyl}-1-[2-(4-methoxyphenyl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-{3-[(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]phenyl}ethan-1-amine
4-(2,6-dimethylpyridin-3-yl)-N-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]pyrimidin-2-amine
3-[3-(furan-2-yl)-1H-pyrazol-1-yl]-5-(pyrrolidine-1-sulfonyl)benzoic acid
5-methyl-4-[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]pyrimidin-2-amine
1-methyl-4-({methyl[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amino}methyl)-1H-pyrrole-2-carbonitrile
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(propan-2-yloxy)propyl]acetamide
1-{2-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-{1-[3-(methoxymethyl)benzoyl]piperidin-2-yl}ethan-1-ol
1-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
2-methoxy-5-({[(8-methoxyquinolin-5-yl)methyl](methyl)amino}methyl)benzoic acid