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3-(dimethyl-1,2-oxazol-4-yl)-N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]propanamide
N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-6-oxo-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
4-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyrimidin-2-amine
1-(2,3-dihydro-1H-inden-5-yl)-3-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}urea
ethyl 1-[(2E)-4-methylpent-2-enoyl]-4-(oxan-2-ylmethyl)piperidine-4-carboxylate
N,2-dimethyl-4-oxo-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide
4-[1-(2-fluorophenyl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl]butanoic acid
2-{1-[(6-methylpyridin-2-yl)methyl]-4-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl}ethan-1-ol
(3S,4S)-4-(4-fluorophenyl)-1-[(3-methyl-1H-indol-2-yl)methyl]piperidin-3-ol
methyl 4-{4-[6-(dimethylamino)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperazin-1-yl}benzoate
N-(2-methoxyethyl)-4-oxo-N-(thiophen-2-ylmethyl)-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
7-(4-chloro-1H-pyrazole-3-carbonyl)-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-[4-(1-methyl-1H-pyrazol-5-yl)phenyl]pyridine-4-carboxamide
(3R,5S)-N-[2-(1-methylpyrrolidin-2-yl)ethyl]-1-(naphthalen-2-ylmethyl)-5-[3-(trifluoromethyl)phenoxymethyl]piperidine-3-carboxamide
(2R,6R)-4-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-triene-6-carboxylic acid
3-(3-methoxybenzoyl)-1-[(3-methyl-1H-pyrazol-5-yl)methyl]piperidine
(4aR,8aR)-4a-hydroxy-7-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-N,N-dimethyl-decahydro-2,7-naphthyridine-2-carboxamide
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-[2-(methylsulfanyl)ethyl]benzamide
4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidine
ethyl 4-(2,3,4,5-tetrahydro-1-benzoxepine-4-amido)piperidine-1-carboxylate
{1-[1-(3-phenyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methanol
2-{1-[(2-ethylpyrimidin-4-yl)methyl]piperidin-4-yl}-1,3-benzoxazole
5-(2-chlorophenyl)-N-[(3S,4R)-4-ethoxyoxolan-3-yl]furan-2-carboxamide
2-methyl-4-(3-{2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carbonyl}phenyl)butan-2-ol
N-butyl-N-(thiophen-3-ylmethyl)-1,8-naphthyridine-2-carboxamide
(3S,4S)-N-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]-4-methoxy-1-(propan-2-yl)pyrrolidin-3-amine
5-(2-fluorophenoxymethyl)-N-[(6-hydroxypyrimidin-4-yl)methyl]-1H-pyrazole-3-carboxamide
2-amino-3-ethyl-N-[(3-methyloxetan-3-yl)methyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
2-[4-(benzyloxy)butanoyl]-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
N-methyl-2-[(1S,6R)-4-oxo-3,9-diazabicyclo[4.2.1]nonan-3-yl]-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
N-(1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperidin-4-yl)methanesulfonamide
methyl 3-{[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]carbamoyl}propanoate
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[3-(methylsulfanyl)propyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
2-methyl-N-(1-{1-[3-(1,2-oxazolidin-2-yl)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
1-{[4-(benzyloxy)-2-methoxyphenyl]methyl}-4-(1,2,4-oxadiazol-3-yl)piperidine
N-{1-[1-(3-methoxybenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}oxolane-3-carboxamide
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}propanamide
N-[4-(1H-indol-2-yl)phenyl]-1-(3-methoxypropanoyl)pyrrolidine-2-carboxamide
2-[2-methyl-3-({[(1-methyl-3-phenyl-1H-pyrazol-5-yl)methyl]amino}methyl)-1H-indol-1-yl]acetamide
N-[(5-chloro-2-methoxyphenyl)methyl]-N-ethyl-2-(methylamino)pyridine-3-carboxamide
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]quinoline-3-carboxamide
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-3-(3,4-dimethoxyphenyl)propanamide
2-methyl-N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}-1-benzofuran-5-carboxamide
3-{[4-(aminomethyl)-1H-1,2,3-triazol-1-yl]methyl}-N-[2-(4-fluorophenyl)ethyl]piperidine-1-carboxamide
N-(2-methoxyethyl)-N-{[6-methyl-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-2-(thiophen-3-yl)acetamide
2-[3-(2-phenylethyl)piperidin-1-yl]-5-(piperidine-1-carbonyl)pyridine
(3S,4R)-3-ethyl-4-methyl-1-(2-methyl-4-phenyl-1,3-thiazole-5-carbonyl)piperidin-4-ol
(1S,5R)-3-(3-acetylbenzoyl)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(cyclohexylmethyl)-N-ethyl-5-(2-fluorophenoxymethyl)-1H-pyrazole-3-carboxamide
5-(4-chloro-3,5-dimethylphenoxymethyl)-N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1,2-oxazole-3-carboxamide