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N-{3-oxo-3-[(1S,5R)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propyl}methanesulfonamide
[3-({ethyl[(1-ethyl-1H-pyrazol-4-yl)methyl]amino}methyl)-2,4,6-trimethylphenyl]methanol
4-[(4-hydroxy-5-methoxypyridin-2-yl)methyl]-3-methyl-1-(2-methylpropyl)piperazin-2-one
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-2-(2-ethyl-4-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetamide
7-[(2,3-difluorophenyl)methyl]-2-(pyrazine-2-carbonyl)-2,7-diazaspiro[4.5]decane
N-(oxolan-2-ylmethyl)-3-{1-[3-(pyridin-2-yl)propanoyl]piperidin-4-yl}propanamide
N-[(3R,4S)-1-cyclopentyl-4-cyclopropylpyrrolidin-3-yl]-2-[4-(hydroxymethyl)phenyl]acetamide
5-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridine-6-carbonyl]-2-(pyrrolidin-1-yl)pyrimidine
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(5-methylpyrazine-2-carbonyl)piperidine-4-carboxamide
N-{[(propan-2-yl)carbamoyl]methyl}-2-(1H-pyrazol-1-yl)butanamide
N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
6-{[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amino}pyridine-3-carboxamide
7-(5-chloro-2-methoxyphenyl)-4-(2,2-dimethyloxane-4-carbonyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-tert-butyl-5-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-1,3,4-oxadiazole
N-[(3R,7S,8aS)-3-[(1S)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3,5-dichlorobenzamide
N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]-3-(pyridin-3-yl)propanamide
2-(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidin-1-yl)pyridine-3-carboxamide
3-[(3S,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(4-chlorophenyl)urea
N-[(3-chlorophenyl)methyl]-3-{1-[2-(1H-1,2,4-triazol-1-yl)propanoyl]piperidin-4-yl}propanamide
1-{[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(thiophene-2-carbonyl)piperazine
N-(propan-2-yl)-1-[(1s,4s)-4-[2-(pyridin-2-ylsulfanyl)acetamido]cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-(2-methylpropyl)-1-[1-(pyrazine-2-carbonyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
1-{2-amino-4-[(2-methoxyethyl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}-3-(1H-pyrrol-1-yl)propan-1-one
2-methyl-4-[4-(pyridin-3-ylmethyl)piperazine-1-carbonyl]-1,2-dihydrophthalazin-1-one
3-[1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]-1-[4-(propylsulfamoyl)phenyl]urea
N-{[1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-4-hydroxyazepan-4-yl]methyl}pyrrolidine-1-carboxamide
N-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-1-[2-(2-methoxyphenyl)ethyl]-2,6-dimethyl-4-oxo-1,4-dihydropyridine-3-carboxamide
3-(2,5-dimethylphenyl)-1-({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-1-methylurea
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-4-hydroxy-2-(pyridin-2-yl)pyrimidine-5-carboxamide
N-[2-(2,4-dimethoxyphenyl)ethyl]-3-(pyridin-4-yl)propanamide
N-{[(3S,4S)-3-hydroxy-1-(5-methoxyfuran-2-carbonyl)piperidin-4-yl]methyl}pyrrolidine-1-carboxamide
2-ethyl-N-(5-fluoro-2-methoxyphenyl)-2,5-dihydro-1H-pyrrole-1-carboxamide
3-[2-({[3-(4-fluorophenyl)oxolan-3-yl]methyl}(methyl)amino)ethyl]-1H-indol-5-ol
(4aS,7aR)-1-(3-cyclopentylpropanoyl)-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{[(butan-2-yl)(cyclopentyl)amino]methyl}-1-methyl-1,2-dihydroquinolin-2-one
N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
(1S,5R)-3-[2-(4-chloro-2-methylphenoxy)acetyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{2-[(2-butyl-6-methylpyrimidin-4-yl)amino]ethyl}-4-hydroxy-2-methylpyrimidine-5-carboxamide
(2S,4R)-4-amino-1-[3-(1,3-benzothiazol-2-yl)propanoyl]-N-ethylpyrrolidine-2-carboxamide
1-(2-methoxyacetyl)-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]piperidine-4-carboxamide
3-{2-oxo-2-[4-(pyridin-2-ylmethyl)piperazin-1-yl]ethyl}-4-(3-phenylpropyl)piperazin-2-one
1-[(4-methylphenyl)methyl]-4-{2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanoyl}piperazin-2-one
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-(thiophen-3-ylmethyl)cyclopropanamine
2-(2H-1,3-benzodioxol-5-yl)-1-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-9-yl]ethan-1-one
2-[(2-chlorophenyl)methyl]-N-ethylmorpholine-4-carboxamide
(1R,9aR)-1-{10,13-dioxa-4,5,6-triazatricyclo[7.4.0.03,7]trideca-1(9),2,5,7-tetraen-4-ylmethyl}-octahydro-1H-quinolizin-1-ol
4-methoxy-N-[1-(1-{spiro[2.3]hexane-1-carbonyl}piperidin-4-yl)-1H-pyrazol-5-yl]benzamide
4-[(3-hydroxyphenyl)methyl]-1-(2-phenylethyl)-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
N-[(1-tert-butyl-5-oxopyrrolidin-3-yl)methyl]-N-methyl-2-[(prop-2-en-1-yl)amino]benzamide
3-[5-(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]propan-1-ol