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(2S,4R)-1-[(4-chlorophenyl)methyl]-N-(2-methoxyethyl)-4-({[3-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
1-{2-[2-(3-{[methyl(quinolin-8-ylmethyl)amino]methyl}phenoxy)ethyl]piperidin-1-yl}-2-phenylethan-1-one
N-[(2,2-dimethyl-1-phenylcyclopropyl)methyl]-3-propyl-1H-pyrazole-5-carboxamide
4-(1H-imidazol-1-yl)-1-[(2-methyl-1-benzothiophen-3-yl)methyl]piperidine-4-carboxylic acid
N-[1-(3-cyanopyridin-2-yl)piperidin-4-yl]-2-(2,5-dioxoimidazolidin-1-yl)acetamide
N-(3-methoxy-4-methylphenyl)-4-[(1-methylpiperidin-3-yl)methyl]piperazine-1-carboxamide
N-{[1-(morpholin-4-yl)cycloheptyl]methyl}-2-oxo-1-phenylpyrrolidine-3-carboxamide
4-[5-(3-benzyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-1-methylpiperazin-2-one
N-[(2-amino-1,3-thiazol-4-yl)methyl]-4-(4-oxo-3,4-dihydroquinazolin-3-yl)butanamide
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-3-[4-(3-methylphenyl)piperazin-1-yl]propanamide
methyl 2-{1-[2-(2,3-difluorophenoxymethyl)-1,3-oxazol-4-yl]-N-methylformamido}acetate
1-[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]-3-[(3S,4R)-1-(pyridin-2-ylmethyl)-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]propan-1-one
N-(6-phenoxypyridin-3-yl)-1-(1,2,3-thiadiazole-4-carbonyl)piperidine-4-carboxamide
2-[3-(4-fluoro-2-methoxyphenyl)phenoxy]acetamide
3-(2-{[(3-methyl-1H-pyrazol-5-yl)methyl]amino}phenyl)-1,3-oxazolidin-2-one
5-(1,3-benzoxazol-2-yl)-N-[2-(dimethylamino)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-(1-tert-butyl-1H-pyrrole-3-carbonyl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
2-(1-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}piperidin-4-yl)-N-methylacetamide
4-phenyl-1-(3-propyl-1H-pyrazole-5-carbonyl)piperidine-4-carbonitrile
5-cyclopropyl-1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-[1-(6-methylpyridin-2-yl)propan-2-yl]-1H-pyrazole-4-carboxamide
5-(azocan-1-yl)-1-(prop-2-en-1-yl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
4-{[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl}thiomorpholine
8-[2-(2-ethylphenoxy)ethyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-(3-phenylpropyl)-8-[2-(1H-1,2,4-triazol-1-yl)propanoyl]-2,8-diazaspiro[4.5]decan-3-one
1-{4-[4-(3,6,7-trimethyl-1-benzofuran-2-carbonyl)piperazin-1-yl]phenyl}ethan-1-one
3-[(2-ethylbutyl)amino]-5-(phenylsulfamoyl)-N-(pyridin-3-ylmethyl)benzamide
(4aS,7aR)-1-(3-methyl-1H-pyrazole-5-carbonyl)-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{4-fluoro-2-[1-(2-methoxy-2-methylpropyl)-1H-imidazol-2-yl]phenyl}-3,5-dimethyl-1H-pyrazole
1-(3-methylpyridin-4-yl)-4-(2-propoxybenzoyl)-1,4-diazepane
2-[3-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)piperidin-1-yl]pyrimidine
3-methyl-1-{1-[2-(pyrrolidin-1-yl)benzoyl]piperidin-4-yl}butan-1-ol
1-[1'-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
3-(1-propyl-1H-pyrazol-5-yl)-1-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]urea
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(quinolin-8-ylmethyl)pyrrolidine-3-carboxylic acid
6-(2,5-dimethylfuran-3-yl)-N-(2-hydroxypropyl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
7-(5-phenoxyfuran-2-carbonyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
[(3S,5R)-5-[(dimethylamino)methyl]-1-(2-methoxy-4-methylbenzenesulfonyl)piperidin-3-yl]methanol
4-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-1,2-dihydroquinazolin-2-one
N-[(2,4-dimethoxyphenyl)methyl]-3-(1-ethylpiperidin-3-yl)propanamide
N,5-dimethyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1-propyl-1H-pyrazole-4-carboxamide
2-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-1,3-benzoxazole
1-[6-(4-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-2-(methoxymethyl)piperidine
3-(3-methylbutyl)-8-(oxolan-3-ylmethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
methyl 8-[(2-chloro-4,5-dimethoxyphenyl)methyl]-2-oxo-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate
N-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
N-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-2-{2-[(dimethylamino)methyl]-4-(pyridin-3-yl)phenoxy}acetamide
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-[1-(pyridin-4-ylmethyl)piperidin-4-yl]pyrimidin-2-amine
(2R,6S)-4-(1-{5-cyclopropyl-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}piperidin-4-yl)-2,6-dimethylmorpholine
4-benzyl-1-(2-phenylethyl)-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one