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N-(propan-2-yl)-6-[3-(1H-pyrazol-5-yl)piperidin-1-yl]pyrimidin-4-amine
4-phenyl-N-(3-{4-[4-(pyridin-4-ylmethyl)piperazin-1-yl]piperidin-1-yl}phenyl)butanamide
2-(dimethylamino)-N-{1-[1-(1H-indole-5-carbonyl)piperidin-4-yl]-2-phenylethyl}-N-methylacetamide
1-(1-benzylpiperidin-4-yl)-N-(2-methylprop-2-en-1-yl)piperidine-3-carboxamide
2-cyclopropyl-9-[5-oxo-1-(prop-2-en-1-yl)pyrrolidine-3-carbonyl]-2,9-diazaspiro[5.5]undecan-3-one
(1R,9aR)-1-[({[5-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-3-yl]methyl}amino)methyl]-octahydro-1H-quinolizin-1-ol
1-(4-fluorophenyl)-N-[2-(4-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]cyclopropane-1-carboxamide
methyl(quinolin-2-ylmethyl)[1-(thiophen-2-yl)ethyl]amine
7-(3-chlorophenyl)-4-(5-methylpyrazine-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-ethyl-6-methyl-5-{2-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]-2-oxoethyl}-3,4-dihydropyrimidin-4-one
N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-(pyridin-2-yl)acetamide
2-cyclohexyl-5-({4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}methyl)pyrimidine
3-{1-[2-(3,4-dimethyl-6-oxo-1,6-dihydropyridazin-1-yl)acetyl]piperidin-3-yl}benzoic acid
3-(4-ethoxyphenyl)-3-{[3-(1H-pyrazol-1-yl)phenyl]formamido}propanoic acid
ethyl 1-[3-({[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)-6,7-dimethoxyquinolin-2-yl]piperidine-3-carboxylate
1-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-(5-methylpyridin-2-yl)piperidin-4-ol
5-propyl-N-[2-(4H-1,2,4-triazol-4-yl)ethyl]-1,2-oxazole-3-carboxamide
N-(cyclohex-1-en-1-ylmethyl)-2-ethyl-4-methyl-1,3-oxazole-5-carboxamide
5-(2-phenylazetidine-1-carbonyl)-2-(pyridin-3-yl)pyrimidin-4-ol
2-[4-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)piperazin-1-yl]-1,3-benzothiazole
methyl 3-[(3S,4R)-1-[(3-chlorophenyl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]propanoate
5-({2-oxo-1,2-dihydrospiro[indole-3,4'-piperidine]-1'-yl}carbonyl)pyridine-2-carbonitrile
2-(2-chloro-4-fluorophenyl)-N-[(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)methyl]acetamide
N-benzyl-2-(2-methoxyphenyl)-N-(1,3-thiazol-2-ylmethyl)acetamide
1-(2-phenylethyl)-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
1-[1-(4-chlorophenyl)cyclopropanecarbonyl]-4-[(2-fluorophenyl)methyl]-1,4-diazepan-5-one
4-(5-chloro-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1-cyclopentylpyrrolidin-2-one
1-cyclopentyl-N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]piperidine-3-carboxamide
2-methoxy-N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}-5-sulfamoylbenzamide
2-(6-phenoxypyridin-3-yl)-1H-1,3-benzodiazole-5-carbonitrile
1-(2-{1-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]piperidin-2-yl}ethyl)pyrrolidin-2-one
2-(naphthalen-2-yloxy)-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}acetamide
1-(4-chloro-3-methylphenyl)-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
2-methyl-7-{2-[(4-methylphenyl)methyl]benzoyl}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-4-(1H-imidazol-1-yl)butan-1-one
4-[(2-fluorophenyl)methyl]-1-[4-(thiophen-2-yl)butanoyl]-1,4-diazepan-5-one
3-chloro-N-(2-methoxyethyl)-4-{[1-(4,4,4-trifluorobutyl)piperidin-4-yl]oxy}benzamide
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-1-(pyrimidin-2-yl)piperidin-4-amine
N-[(2-chloro-6-fluorophenyl)methyl]-N-ethyl-3-(4-hydroxyphenyl)-1H-pyrazole-5-carboxamide
5-{1-[(2-methyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-4-phenyl-1H-imidazol-5-yl}pyrimidine
(1S,4S)-2-(3-chloro-4-methoxyphenyl)-5-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-2,5-diazabicyclo[2.2.1]heptan-3-one
3-{1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]azetidin-3-yl}pyridine
N-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-5-cyclopropyl-1-[4-(furan-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]oxane-4-carboxamide
3-{methyl[3-(1H-pyrazol-1-yl)propyl]sulfamoyl}-N-(oxolan-3-yl)benzamide
6-methyl-2-propyl-N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}pyrimidin-4-amine
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
4-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]benzene-1-sulfonamide
1-cyclohexyl-5-[(2-methyl-1,3-thiazol-4-yl)methyl]-1H-1,2,4-triazole
[(3S,5R)-5-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(5-methyl-1,3-benzoxazol-2-yl)piperidin-3-yl]methanol