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N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N,1-dimethyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-(oxolan-2-ylmethyl)-2-(3-phenylpropyl)-1,3-benzoxazole-5-carboxamide
2-amino-N-[2-(dimethylamino)ethyl]-N-[(3-methylthiophen-2-yl)methyl]acetamide
(1S,5R)-6-(3,5-difluorobenzoyl)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-[(3-acetylphenyl)methyl]-N-[3-(3-fluorophenyl)phenyl]piperidine-4-carboxamide
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-amine
(2S,4R)-4-amino-N-ethyl-1-[4-(trifluoromethyl)benzoyl]pyrrolidine-2-carboxamide
3-(2,3-dihydro-1,4-benzodioxin-6-yl)-4-{[2-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-1-methyl-1H-pyrazole
(2R,3R,6R)-3-(4-fluorophenyl)-5-[5-(methoxymethyl)furan-2-carbonyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-4-methylpentan-1-one
4-methyl-N-[2-(7-{[4-(propan-2-yloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]benzamide
(3S,5S)-N-[(2-chlorophenyl)methyl]-1-(2,3-dihydro-1H-inden-2-yl)-5-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)pyrrolidin-3-amine
2-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyrimidine
N-[5-carbamoyl-2-(2-methylpiperidin-1-yl)phenyl]-2-methoxypyridine-3-carboxamide
(1S,6R)-3-[3-oxo-3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
2-(morpholin-4-yl)-2-(pyridin-3-yl)-N-[2-(thiophen-2-yl)ethyl]acetamide
N-(1,3-benzothiazol-2-ylmethyl)-4-hydroxy-N-methyl-2-(pyridin-4-yl)pyrimidine-5-carboxamide
(5S,9aS,9bS)-5-(9H-fluoren-2-yl)-2-(1-methylpiperidin-4-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-(cyclopropylmethyl)-5-methyl-4-{[2-(pyridin-2-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
N-methyl-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
3-{2-[4-(2-hydroxyethyl)piperazin-1-yl]-2-oxoethyl}-4-[(4-methylphenyl)methyl]piperazin-2-one
N-cyclohexyl-4-[3-(4-methyl-1,3-thiazol-5-yl)propanamido]piperidine-1-carboxamide
1-[(5-chlorothiophen-2-yl)methyl]-3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
5-(4-benzoylpiperidine-1-carbonyl)-1-(pyridin-2-ylmethyl)piperidin-2-one
1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]urea
2-{[(2-chlorophenyl)methyl]sulfanyl}-1-[(3R,5R)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidin-1-yl]ethan-1-one
{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]methylamine
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-N-(2-methoxyethyl)-N-methyl-1H-pyrazole-4-carboxamide
(4aS,8aR)-6-(ethanesulfonyl)-1-[2-(5-methylfuran-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-(2-phenylethyl)-1,2-oxazole-3-carboxamide
2-[2-(pyrrolidin-1-yl)ethyl]-1-(1,3-thiazol-4-ylmethyl)piperidine
1-(6-cyanopyridin-2-yl)-4-(2-fluorophenoxy)piperidine-4-carboxylic acid
4-[1-(cyclopent-1-ene-1-carbonyl)piperidin-3-yl]-5-phenyl-2-(pyridin-4-yl)pyrimidine
6-(3-chlorophenyl)-N-(2-methoxyethyl)-N-(propan-2-yl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
4-ethyl-5-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,3-thiazol-2-amine
[(4-chloro-3-fluorophenyl)methyl](methyl)[2-(2-methyl-1H-imidazol-1-yl)ethyl]amine
1-(3-aminoazepan-1-yl)-4-(thiophen-2-yl)butan-1-one
4-(4-benzyl-3-ethyl-5-oxo-1,4-diazepan-1-yl)-4-oxobutanamide
3-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)formamido]-N-(4-methylphenyl)propanamide
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(pyridin-2-yl)acetamide
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-{3-[4-(trifluoromethyl)phenyl]-1H-pyrazol-1-yl}acetamide
N-[(4-fluorophenyl)methyl]-5-(4-formylpiperazin-1-yl)-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-(4-methyl-1,3-thiazol-5-yl)-N-[(3-methylphenyl)(thiophen-2-yl)methyl]propanamide
N-methyl-2-(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)-5H,6H,7H-cyclopenta[d]pyrimidin-4-amine
2-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]-2,7-diazaspiro[4.5]decane
N-(1-methyl-1H-pyrazol-4-yl)-3-({3-methyl-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl}methyl)benzamide
2-oxo-2-(thiophen-2-yl)-N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]acetamide
3-tert-butyl-1-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}urea
5-[4-(hydroxymethyl)piperidin-1-yl]-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
1-[1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)piperidin-4-yl]-1,4-diazepan-5-one