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5-(6-methoxy-2H-1,3-benzodioxol-5-yl)-1-[(2S)-1-methoxypropan-2-yl]-4-phenyl-1H-imidazole
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanamide
1-(1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)-4-[3-(trifluoromethyl)phenyl]piperazine
2-ethyl-4-{[2-(methylsulfanyl)phenyl]methyl}-1-(propan-2-yl)piperazine
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(pyrrolidin-1-yl)butanamide
1-{4-[1-(difluoromethyl)-3-methyl-1H-pyrazol-4-yl]phenyl}-3-ethylurea
N-[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
N-(1-carbamoylcycloheptyl)-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-3-phenoxypropanamide
1-(adamantan-1-yl)-4-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperazine
3-[2-oxo-2-(piperidin-1-yl)ethyl]-4-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-one
(2S)-1-{[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}pyrrolidine-2-carboxamide
{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}bis(prop-2-en-1-yl)amine
N-[2-(3-chlorophenyl)ethyl]-2-[(6-{[(4-fluorophenyl)methyl](methyl)amino}pyridazin-3-yl)oxy]acetamide
6-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N-ethyl-N-methylpyrimidin-4-amine
2-(1-{1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
(3S,9aR)-3-(1H-imidazol-4-ylmethyl)-8-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[4-(3-fluorophenyl)phenyl]-4-[3-(methoxymethyl)pyrrolidin-1-yl]piperidine
4-{5-[2-(morpholin-4-yl)ethyl]-1,2,4-oxadiazol-3-yl}-1H-indole
N-{2-[5-(2-methoxypyrimidin-5-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}pyridin-3-amine
3-{5-[methoxy(phenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-{2-[4-(trifluoromethyl)phenyl]ethyl}propanamide
N-(2-chloro-6-methylphenyl)-3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carboxamide
{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl){[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}amine
1-{2-[2-({3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)phenoxy]ethyl}-1H-imidazole
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-(4-methylbenzoyl)pyrrolidin-3-yl]methanol
N-[(1-ethylpyrrolidin-2-yl)methyl]-4-(pyridin-2-yl)pyrimidin-2-amine
1-{4-[3-(ethoxymethyl)-1-(1-methylpiperidin-4-yl)-1H-1,2,4-triazol-5-yl]thiophen-2-yl}ethan-1-one
(1S,5R)-6-{3-fluoro-7-methylimidazo[1,2-a]pyridine-2-carbonyl}-1,3,3-trimethyl-6-azabicyclo[3.2.1]octane
(3aR,7aS)-2-[(1-benzyl-1H-imidazol-5-yl)methyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
N-(1,3-dimethyl-1H-pyrazol-5-yl)-2-{3-[(E)-2-phenylethenyl]-1H-indazol-1-yl}acetamide
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(pyrimidin-2-ylsulfanyl)acetamide
N-[3-(4-{[(2-benzyl-1,3-thiazol-4-yl)methyl]amino}piperidin-1-yl)phenyl]pyridine-4-carboxamide
(1S,4S)-2-(2H-1,3-benzodioxol-5-yl)-5-[(8-methoxyquinolin-2-yl)methyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
2-methyl-5-[3-(2-methylphenyl)piperidine-1-carbonyl]-1H-1,3-benzodiazole
6-butyl-2-{2-[(2-methylpiperidin-1-yl)methyl]phenyl}-3,4-dihydropyrimidin-4-one
3-({2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}methyl)pyridin-2-amine
[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](2-methoxyethyl){[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}amine
1-(5-methoxy-2-{[(1-phenylcyclopropyl)amino]methyl}phenoxy)-3-(4-methylpiperazin-1-yl)propan-2-ol
N-[(3-ethoxy-4-methoxyphenyl)methyl]-N-methyl-2-(2-oxopiperidin-1-yl)acetamide
2-ethyl-8-({4-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)-2,8-diazaspiro[4.5]decan-3-one
N-(butan-2-yl)-4-methyl-3-(2-oxoimidazolidin-1-yl)-N-(thiophen-3-ylmethyl)benzamide
(1S,5R)-6-(cyclobutylmethyl)-3-{4-[(2-hydroxyethyl)(methyl)amino]benzoyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
4-(1-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-1H-imidazol-2-yl)quinoline
N-{2-methyl-3-[(1,3-thiazol-2-yl)carbamoyl]phenyl}-1-(propan-2-yl)piperidine-4-carboxamide
N-[(1-cyclopentylpiperidin-4-yl)methyl]-1-(furan-2-ylmethyl)piperidin-4-amine
3-(4-hydroxyphenyl)-N-methyl-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1H-pyrazole-5-carboxamide
2-{methyl[(3-methylpyridin-2-yl)methyl]amino}-2-[4-(1H-pyrazol-5-yl)phenyl]acetic acid
methyl 2-{3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}pyridine-3-carboxylate
3-(5-{2-[4-(propan-2-yl)morpholin-2-yl]acetyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)propanoic acid
3-[(3R,4S)-1-(5-methyl-1H-indazole-3-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol