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8-(2-methyl-1,3-thiazole-4-carbonyl)-2-(oxolan-2-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
N-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-N-methyl-1-(pyrimidin-2-yl)piperidin-4-amine
N-[2-(furan-2-yl)ethyl]-3-{imidazo[1,2-a]pyridin-2-yl}propanamide
N-[2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)ethyl]imidazo[1,2-a]pyridine-3-carboxamide
(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-{[(4-chlorophenyl)methyl]amino}-1-(propan-2-yl)pyrrolidine-2-carboxamide
6-methyl-4-{1-methyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaene
5-(pyridin-4-yl)-N-(thiophen-3-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
1-[4-(ethylcarbamoyl)pyridin-2-yl]-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
1-(4-{[(1-ethylcyclobutyl)methyl]amino}-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
1-{2-[2-(2-methylphenyl)pyrrolidin-1-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one
4-{butyl[2-(2,2,6,6-tetramethylpiperidin-4-yl)ethyl]amino}butan-1-ol
1-(1-cyclopropyl-1H-pyrrole-2-carbonyl)-4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-1,4-diazepan-6-ol
5-methanesulfonyl-N-(3-phenylpropyl)-4-(piperidin-3-yl)pyrimidin-2-amine
1-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
4-[(3S)-3-hydroxy-3-phenylpropyl]-1-(3-methoxyphenyl)piperazin-2-one
1-{1-ethyl-5-[2-(2-fluorophenyl)benzoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}pyrrolidine
2-[4-(hydroxymethyl)phenyl]-2-{4-[(3-methoxyphenyl)methyl]-3-oxopiperazin-1-yl}acetic acid
2-methoxyethyl 4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepane-1-carboxylate
2-(1-ethylpiperidin-4-yl)-N-[2-(3-fluorophenyl)-2-hydroxyethyl]acetamide
2-(6-methoxynaphthalen-2-yl)-4-(2-propylpyridine-4-carbonyl)morpholine
(3R)-3,4,4-trimethyl-1-[5-(piperidine-1-carbonyl)pyridin-2-yl]pyrrolidin-3-ol
4-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}benzene-1-sulfonamide
6-{6-amino-1H-pyrrolo[2,3-b]pyridin-4-yl}-N-(propan-2-yl)pyridazin-3-amine
3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]-1-(2-propyl-2,5-dihydro-1H-pyrrol-1-yl)propan-1-one
2-[2-(pyrrolidin-1-yl)-6-(trifluoromethyl)pyrimidin-4-yl]-1,2,3,4-tetrahydroisoquinolin-4-ol
(3aS,6aS)-2-[(3-chloro-4,5-dimethoxyphenyl)methyl]-5-(2-hydroxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N,N-dimethyl-5-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}thiophene-2-carboxamide
3-amino-1-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}propan-1-one
2-[3-(phenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyridine
3-(3,3-diphenylpiperidine-1-carbonyl)piperidine-1-carboxamide
N,2,5,6-tetramethyl-N-{[1-(morpholin-4-yl)cyclohexyl]methyl}pyrimidin-4-amine
4-{2-[(cyclopropylmethyl)sulfanyl]acetyl}-1-(3,5-dimethylphenyl)piperazin-2-one
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-(3-phenylpropyl)propanamide
8-cyclopentyl-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
N-[2-chloro-5-(diethylcarbamoyl)phenyl]-6-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
(4aR,7aS)-1-butyl-4-(2-methoxy-5-methylbenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(4,6-dimethylpyridin-2-yl)methyl]-5-methanesulfonyl-N-methyl-4-(piperidin-3-yl)pyrimidin-2-amine
4-[4-(2-methoxyacetamido)-1H-pyrazol-1-yl]-N-[3-(pyridin-3-yloxy)propyl]benzamide
N-[(3R,5S)-1-cyclopropanecarbonyl-5-(diethylcarbamoyl)pyrrolidin-3-yl]-5-methylpyrazine-2-carboxamide
5-{[(2,3-dimethoxyphenyl)methyl]amino}-N,N-dimethyl-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]-1,2,5-thiadiazole-3-carboxamide
N3-[1-(4-fluorophenyl)ethyl]-N5-methyl-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
4-{2-[2-(3-ethyl-1,2-oxazol-5-yl)-1H-imidazol-1-yl]ethyl}benzene-1-sulfonamide
ethyl[(1-ethylpyrrolidin-3-yl)methyl][(1-methyl-1H-imidazol-2-yl)methyl]amine
3-(2-fluorophenyl)-1-{4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}propan-1-one
6-[(5-acetamidothiophen-2-yl)methyl]-N-methyl-N-[2-(4-methylphenoxy)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
2-(3-methoxypropyl)-8-[(2-methyl-1,3-thiazol-4-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-(2,3-dihydro-1H-inden-4-yl)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}benzamide
N-{[7-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-phenyl-1,2-oxazole-5-carboxamide
N-[(5-fluoro-1H-indol-2-yl)methyl]-N-methyl-2-(pyrrolidin-3-yl)benzamide