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3,6-dimethyl-N-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
1-[(3-chlorophenyl)methyl]-4-[(4R)-3-methyl-1,3-thiazolidine-4-carbonyl]piperazine
N-(2-fluoro-5-methylphenyl)-4-[3-(2-methylpropyl)morpholin-4-yl]-4-oxobutanamide
(4-{2-phenyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}morpholin-2-yl)methanamine
3-[2-(2,4-difluorophenyl)ethyl]-1-(furan-3-carbonyl)piperidine
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetamide
N-{2-[1-(2-methylpropyl)piperidin-3-yl]ethyl}-1,3-thiazole-5-carboxamide
4-(4-chloro-2-hydroxybenzoyl)-1-(2-methylphenyl)piperazin-2-one
N-(oxolan-2-ylmethyl)-3-(1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)propanamide
4-{2-[benzyl(methyl)carbamoyl]ethyl}-N-(3,4-dimethylphenyl)piperidine-1-carboxamide
N-butyl-N-[(2-fluorophenyl)methyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
(3R,5S)-N3-ethyl-N3-[(1-methyl-1H-pyrazol-4-yl)methyl]-N5-(6-methylpyridin-3-yl)piperidine-3,5-dicarboxamide
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-4-(3-hydroxy-3-methylbutyl)benzamide
3-{1-[(1,2-dimethyl-1H-indol-3-yl)methyl]piperidin-4-yl}-N-[(1-ethylpyrrolidin-2-yl)methyl]propanamide
8-chloro-2-(furan-2-yl)-4-[3-(methoxymethyl)pyrrolidine-1-carbonyl]quinoline
(1S,5R)-3-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-butyl-3-(3-methoxyphenyl)-N-[(2-methylphenyl)methyl]-1H-pyrazole-5-carboxamide
1-{[7-chloro-2-(2-methoxyphenyl)quinolin-3-yl]methyl}piperidin-4-ol
2-hydroxy-N-[(5-methoxy-1H-indol-2-yl)methyl]-4-(methylsulfanyl)butanamide
1-methyl-5-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
(3aS,6aS)-2-cyclopentyl-5-(5-methyl-1,3,4-thiadiazol-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
6-(1-methyl-1H-imidazol-2-yl)-N-[1-(thiophen-2-yl)propan-2-yl]pyridazin-3-amine
2-({[(3R,4R)-4-(hydroxymethyl)-1-[(2-methoxy-4-methylphenyl)methyl]pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
4,6-dimethyl-13-(3-phenyl-1,2-oxazol-5-yl)-3,7,8,10-tetraazatricyclo[7.4.0.02,7]trideca-1,3,5,8-tetraen-11-one
3-{4-[(dimethylamino)methyl]phenyl}-5-[(propan-2-yl)sulfamoyl]benzoic acid
2-({[3-(2-ethyl-1H-imidazol-1-yl)propyl]amino}methyl)-6-methylquinolin-4-ol
N'-(2,3-dimethylphenyl)-N-[2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)ethyl]propanediamide
3-(4-tert-butylbenzoyl)-1-(1H-imidazol-2-ylmethyl)piperidine
methyl (2S,4S,5R)-5-(2-fluorophenyl)-1-methyl-4-[(1-phenylcyclopropyl)carbamoyl]pyrrolidine-2-carboxylate
5-[4-(1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-N-benzyl-1-cyclopropyl-4-oxo-1,4-dihydropyridine-3-carboxamide
8-[(4-methoxyphenyl)methyl]-1-(2-methylpropyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl)benzamide
(1R,5R)-6-(1H-1,3-benzodiazole-2-carbonyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
1-methyl-1-[3-(1-methyl-1H-imidazol-2-yl)propyl]-3-{2-methyl-[1,2,4]triazolo[1,5-a]pyridin-8-yl}urea
[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl](2,3-dihydro-1,4-benzodioxin-6-ylmethyl)methylamine
(3S,4S)-1-{[2-(difluoromethoxy)phenyl]methyl}-4-(morpholin-4-yl)pyrrolidin-3-ol
1-[4-({3-[2-(4-fluorophenyl)pyrrolidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)phenyl]-1H-1,2,4-triazole
4-{1-[2-(2,3-difluoro-6-methoxyphenyl)-1H-imidazol-1-yl]butan-2-yl}morpholine
3-[(4-tert-butyl-1H-1,2,3-triazol-1-yl)methyl]-1-(2,3-dihydro-1-benzofuran-5-carbonyl)piperidine
N-[(1R,3R)-3-aminocyclopentyl]-2-(ethylamino)-4-methyl-1,3-thiazole-5-carboxamide
1-{3-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
(3S,4R)-1-(carbamoylmethyl)-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
4-[(2,3-difluorophenyl)methyl]-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
N-(1-benzylpiperidin-4-yl)-1-[4-(3-methoxyphenyl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carboxamide
1-{2-[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]-2-oxoethyl}azepan-2-one
5-(1H-indol-1-ylmethyl)-N-[3-(morpholin-4-yl)propyl]-1H-pyrazole-3-carboxamide
5-[4-(2-methylphenoxy)piperidine-1-carbonyl]-1-[3-(morpholin-4-yl)propyl]piperidin-2-one
3-(3-hydroxy-1,2-oxazol-5-yl)-1-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decan-4-yl]propan-1-one
N-[(3R,4S)-4-cyclopropyl-1-[2-methyl-5-(trifluoromethyl)benzoyl]pyrrolidin-3-yl]acetamide
6-methoxy-2-oxo-N-(2,2,2-trifluoroethyl)-1,2,3,4-tetrahydroquinoline-4-carboxamide