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2-(5-fluoro-2-methylphenyl)-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]acetamide
4-ethyl-3-[(1-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]acetyl}piperidin-4-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
7-chloro-4-[1-ethyl-3-(4-methyl-1,4-diazepane-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[(3R,4S)-4-cyclopropyl-1-(3-sulfamoylbenzoyl)pyrrolidin-3-yl]acetamide
ethyl 3-{[3-(morpholin-4-yl)piperidine-1-carbonyl]amino}propanoate
1-ethyl-8-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{1-[4-(3-chlorophenyl)-5-({[3-(trifluoromethyl)phenyl]methyl}sulfanyl)-4H-1,2,4-triazol-3-yl]ethyl}-2-(1-methyl-1H-pyrrol-3-yl)acetamide
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-4-(1H-pyrazol-3-yl)benzamide
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-3-(4,5,6,7-tetrahydro-2H-indazol-3-yl)propanamide
N-[4-(4-{[1-(1H-indol-1-yl)propan-2-yl]amino}piperidin-1-yl)phenyl]pyrazine-2-carboxamide
5-ethyl-N-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
4-cyclopentyl-N-(oxan-2-ylmethyl)pyrimidin-2-amine
2-(2,5-dimethylphenoxy)-N-(2-methanesulfonamidoethyl)propanamide
2-({2-[bis(pyridin-3-ylmethyl)carbamoyl]phenyl}amino)acetic acid
1-{2-[7-(cyclopropylmethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-2-oxoethyl}imidazolidine-2,4-dione
N-{2-[(6-ethyl-4-methylquinolin-2-yl)amino]ethyl}acetamide
1-(4-{3-[4-(3-chlorophenyl)piperazin-1-yl]piperidin-1-yl}-4-oxobutyl)pyrrolidin-2-one
2-({3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}methyl)phenol
N-methyl-4-[4-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-1,3-thiazol-2-amine
4-ethyl-3-[(1-{[2-(ethylamino)pyrimidin-5-yl]methyl}piperidin-4-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[2-(2-chlorophenyl)ethyl]-5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
1-[(4S,4aS,8aS)-4-hydroxy-4-phenyl-decahydroquinolin-1-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
5-fluoro-2-{1-[3-(2-phenylethyl)-1,2-oxazole-5-carbonyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
1-{2-[4-(adamantan-1-yl)piperazin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N4-{[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
4-oxo-4-phenyl-N-[1-(2-phenylethyl)piperidin-3-yl]butanamide
2-[5-(1H-1,3-benzodiazol-2-yl)-3-(oxan-4-yl)-1H-1,2,4-triazol-1-yl]acetic acid
(2S,4R)-1-{[4-(benzyloxy)phenyl]methyl}-4-[(4-fluorophenyl)sulfanyl]-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]pyrrolidine-2-carboxamide
(4aR,8aR)-1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-6-[(2E)-3-phenylprop-2-en-1-yl]-decahydro-1,6-naphthyridine
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2-methoxy-6-methylbenzamide
3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)propanamide
(1-{[2-cyclohexylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}piperidin-3-yl)methanol
N-[3-(3-fluorophenyl)phenyl]-1-[(2S)-pyrrolidine-2-carbonyl]piperidine-4-carboxamide
N-cyclopentyl-N'-methyl-N'-[2-(oxan-2-yl)ethyl]butanediamide
1-[1'-(3,6-dimethylpyrazin-2-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
5-[(5-hydroxyadamantan-2-yl)amino]-1-methyl-N-[2-(piperidin-1-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(1S,5R)-3-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(1-cyclopentylpiperidin-3-yl)methyl]-1-methyl-N-[2-(piperidin-1-yl)ethyl]-1H-pyrazole-5-carboxamide
{[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}({[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl})amine
2-[4-methoxy-3-(methoxymethyl)phenyl]-6-methyl-1H-1,3-benzodiazole
6-[(4aR,8aR)-7-cyclopentanecarbonyl-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-N,N-dimethylpyridine-2-carboxamide
1-(methoxymethyl)-N-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]cyclobutane-1-carboxamide
2-(2-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-ylmethyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl)pyrimidine
3-cyclopropyl-1-phenyl-5-[2-(trimethyl-1H-pyrazol-4-yl)ethyl]-1H-1,2,4-triazole
2-(3-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine-1-carbonyl}piperidin-1-yl)acetamide
N-{2-[1-({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-4-yl]ethyl}acetamide
4-[(3,4-dimethoxyphenyl)methyl]-2-[(4-fluorophenyl)methyl]morpholine
(2R)-N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]pyrrolidine-2-carboxamide
2-benzyl-9-[4-(1H-pyrazol-4-yl)butanoyl]-2,9-diazaspiro[5.5]undecan-3-one
(3S,4S)-1-[6-(dimethylamino)pyrazin-2-yl]-4-methylpiperidine-3,4-diol