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3-[5-(quinoxalin-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
(3R,4R)-1-(dimethyl-1,3-thiazol-2-yl)-3,4-dimethylpyrrolidin-3-ol
1-[4-(2-hydroxyethyl)piperazin-1-yl]-2-(2-methyl-1H-1,3-benzodiazol-5-yl)ethan-1-one
3-{[(6-methoxypyridin-3-yl)methyl][(5-methylthiophen-2-yl)methyl]amino}propan-1-ol
N-{[4-(2-fluoro-5-methoxyphenyl)phenyl]methyl}cyclopropanamine
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-3-(2-methoxyphenyl)-N-methylpropanamide
2,6-diamino-4-[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]-5,6,7,8-tetrahydroquinoline-3-carbonitrile
(4aR,7aS)-1-{2-[4-(methylamino)piperidin-1-yl]pyrimidin-4-yl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(2-fluorophenyl)methyl]-6-oxo-N-[(3-propyl-1,2-oxazol-5-yl)methyl]piperidine-3-carboxamide
1-{2-[4-(4-methoxyphenoxy)piperidin-1-yl]-2-oxoethyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
methyl 2-[(3-chloro-4-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}phenyl)formamido]acetate
1-{3-[(3R,4S)-3-(dimethylamino)-4-propylpyrrolidin-1-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[3-(4-{[4-(2-chlorophenyl)piperazin-1-yl]methyl}phenoxy)propyl]-3,5-dimethyl-1,2-oxazole-4-sulfonamide
2-[2-amino-6-(pyrrolidin-1-yl)pyrimidin-4-yl]benzoic acid
4-(1-{3-methyl-3H-[1,2,3]triazolo[4,5-b]pyridine-6-carbonyl}piperidin-4-yl)-6-(pyrrolidin-1-yl)pyrimidine
(1-{5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-yl}pyrrolidin-3-yl)methanol
2-(3-{[(1-methanesulfonylpiperidin-4-yl)amino]methyl}-2-methyl-1H-indol-1-yl)acetamide
1-[3-({[(trimethylpyrazin-2-yl)methyl]amino}methyl)pyridin-2-yl]piperidin-3-ol
2-{[2-(2-chloro-4-fluorophenyl)-1H-imidazol-1-yl]methyl}pyridine
1-(3-fluorophenyl)-3-{1-[1-(oxolan-2-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
N4-[2-(1H-imidazol-2-yl)ethyl]-N2,N2-dimethyl-5,6,7,8-tetrahydroquinazoline-2,4-diamine
6-(2-methyl-1,3-thiazol-4-yl)-2-[4-(morpholin-4-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
3-[2-(3-propyl-1H-pyrazole-5-carbonyl)-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-1-yl]pyridine
(4aS,7aR)-1-(3-methoxypropyl)-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3S,4S)-1-(2-phenylpyrimidine-5-carbonyl)-4-(propan-2-yloxy)pyrrolidin-3-ol
8-{6-chloroimidazo[1,2-a]pyrimidine-2-carbonyl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-{1-[1-(5-phenylpentanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}oxolane-3-carboxamide
ethyl 1-[2-(4-methoxyphenyl)ethyl]-5-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-{8-methylimidazo[1,2-a]pyridin-3-yl}-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]acetamide
N-{2-[5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-2-oxopiperidin-1-yl]ethyl}pyridine-3-carboxamide
2-{5-[2-(3-chloro-1,2-oxazol-5-yl)ethyl]-1-(2,3-dihydro-1H-inden-4-yl)-1H-1,2,4-triazol-3-yl}acetamide
4-{1-[1-(1-ethylpiperidine-2-carbonyl)piperidin-4-yl]piperidine-4-carbonyl}morpholine
ethyl 4-[({2-[2-hydroxy-3-(pyrrolidin-1-yl)propoxy]-4-methoxyphenyl}methyl)amino]piperidine-1-carboxylate
N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]oxane-2-carboxamide
4-(2-chlorobenzenesulfonyl)-7-(2-methylphenyl)-9-(oxolan-3-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-1-[3-(1H-pyrazol-1-yl)phenyl]piperidin-4-amine
(1S,5R)-3-(anthracene-9-carbonyl)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
6-[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]-9H-purine
2-{[1-(2-chloro-6-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}pyridine
N-[1-(1-cyclopropylethyl)-3-methyl-1H-pyrazol-5-yl]-2-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazol-1-yl]acetamide
2-(4-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-(2-methylpropyl)piperazin-2-yl)ethan-1-ol
(4aS,7aR)-1-[3-(3,4-dimethylphenyl)propanoyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{4-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]piperazin-1-yl}-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
(2R,6R)-4-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
2-ethoxy-5-(2-{methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}pyrimidin-4-yl)benzoic acid
1-(1-methyl-1H-indole-6-amido)-1,2,3,4-tetrahydronaphthalene-1-carboxylic acid
N-({3-[1-(dimethylamino)ethyl]phenyl}methyl)-N-(pyridin-2-ylmethyl)cyclopropanamine
2-[4-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)phenoxymethyl]pyridine
3-(2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamido)propanamide
3-[2-fluoro-4-(pyrrolidin-1-ylmethyl)phenoxy]-6-(1-methyl-1H-imidazol-2-yl)pyridazine