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N-{4-[(3-propylmorpholin-4-yl)methyl]phenyl}acetamide
4-(furan-3-ylmethyl)-3-(2-{4-[(3-methylphenyl)sulfanyl]piperidin-1-yl}-2-oxoethyl)piperazin-2-one
3-(6-methoxynaphthalene-2-carbonyl)-1-(thian-4-yl)piperidine
8-cyclopropanecarbonyl-2-(4-methyl-1,3-oxazole-5-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-(benzyloxy)-8-[2-(4-phenylpiperidin-1-yl)acetyl]-1,8-diazaspiro[4.5]decan-2-one
2,4-dimethyl-N-[1-(thian-4-yl)piperidin-4-yl]-1,3-thiazole-5-carboxamide
N5-[(2,4-dimethoxyphenyl)methyl]-N2,N2-dimethyl-5,6,7,8-tetrahydroquinazoline-2,5-diamine
N-[(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)methyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
N-[(1R,3R)-3-aminocyclopentyl]-5-phenyl-1H-pyrrole-2-carboxamide
4-benzyl-3-[1-(2-methylpyrimidin-4-yl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
4-(5-{[3-(2-hydroxyethyl)-4-[1-(propan-2-yl)piperidin-4-yl]piperazin-1-yl]methyl}thiophen-2-yl)-2-methylbut-3-yn-2-ol
15-methyl-13-oxo-N-(oxolan-2-ylmethyl)-9-(pyridin-3-yl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide
3-(5-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)pyridine
4-(5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-sulfonyl}pyridin-2-yl)morpholine
[(3S,5R)-1-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidin-3-yl]methanol
1-(5-fluoro-2-methylbenzoyl)-4-(2-methylpyridin-4-yl)-1,4-diazepane
7-acetamido-2-(2-methoxyphenyl)-1-methyl-N-[1-(pyridin-3-yl)propan-2-yl]-1H-1,3-benzodiazole-5-carboxamide
N-[1-(3-methoxyphenyl)-5-oxopyrrolidin-3-yl]-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
1-{1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]azetidin-3-yl}piperidine
1-{[4-(1-phenoxypropan-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperidin-4-ol
(3R,4R)-4-cyclobutyl-3-methyl-1-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-4-ol
1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-3-(thiophen-2-yl)propan-1-one
3-(azepane-1-carbonyl)-1-methyl-5-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}-4,5,6,7-tetrahydro-1H-indazole
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-(2-methoxyacetyl)piperidine-3-carboxamide
3-ethyl-5-[1-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1H-imidazol-2-yl]-1,2-oxazole
(3S,4S)-1-(3-fluoropyridin-2-yl)-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-({[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)piperidin-2-one
2-[(4-chlorophenyl)methyl]-8-[3-(dimethylamino)propyl]-2,8-diazaspiro[4.5]decan-3-one
N-[(3R,4S)-4-cyclopropyl-1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]pyrrolidin-3-yl]-2-methanesulfonamidoacetamide
N-{[2-(dimethylamino)-7-methoxyquinolin-3-yl]methyl}-4-methoxy-N-(2-methoxyethyl)benzamide
1-[(5-ethylfuran-2-yl)methyl]-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-4-carboxamide
5-(4-cyclopentylpiperazine-1-carbonyl)-1-(2-methylpropyl)-4-oxo-N-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
4-(cyclopropanesulfonyl)-1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-1,4-diazepane
5-acetyl-N,N-bis(prop-2-en-1-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
methyl (2S,4S)-1-[(3,4-difluorophenyl)methyl]-4-propanamidopyrrolidine-2-carboxylate
N-ethyl-3-({[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]carbamoyl}amino)-2-methylbenzamide
(benzylsulfamoyl)({5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl})amine
1-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}-2-(dimethylamino)ethan-1-one
8-(6-ethyl-2-methylpyrimidin-4-yl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
N-{3-[(2,6-dimethylphenyl)carbamoyl]phenyl}-1H-1,3-benzodiazole-5-carboxamide
4-(azepane-1-carbonyl)-2-(1-ethyl-1H-pyrazol-4-yl)-7,8-dimethylquinoline
2-[(1S,5R)-6-[(3,5-dimethyl-1-benzofuran-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
methyl 1-({[1-(cyclopropylmethyl)-1H-indazol-3-yl]carbamoyl}methyl)-1H-pyrazole-3-carboxylate
(2S,4R)-N-cyclopropyl-1-(1-ethylpiperidin-4-yl)-4-[(4-fluorophenyl)sulfanyl]pyrrolidine-2-carboxamide
5-[3-(2-chlorophenyl)-5-methyl-1,2-oxazol-4-yl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
1-propanoyl-N-[2-(pyridin-3-yloxy)phenyl]piperidine-3-carboxamide
N,N-dimethyl-4-[3-(morpholine-4-carbonyl)piperidin-1-yl]piperidine-1-sulfonamide
6-(2-chlorophenyl)-N-ethyl-7-methyl-8-oxo-N-propyl-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-1,9-dioxaspiro[5.5]undecan-4-amine
(3S,4S)-1-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(pyrrolidin-1-yl)pyrrolidin-3-ol