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4-(2-methylphenyl)-N-(3-sulfamoylphenyl)-1,4-diazepane-1-carboxamide
(4aS,8aR)-1-(3-methoxypropyl)-6-(3-methoxypyrazin-2-yl)-decahydro-1,6-naphthyridin-2-one
3-(4-benzyl-4-hydroxypiperidine-1-carbonyl)-N,N-dimethylpiperidine-1-carboxamide
N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}-4-(pyridin-3-yl)pyrimidin-2-amine
6-[2-(4-methylpentyl)morpholine-4-carbonyl]-2,3-dihydropyridazin-3-one
2-[(2-aminopyridin-3-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-[1-(4-ethoxyphenyl)ethyl]-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
N-(2-hydroxyethyl)-N-[(2E)-3-phenylprop-2-en-1-yl]pyrazolo[1,5-a]pyridine-2-carboxamide
5-({[1-(furan-2-ylmethyl)piperidin-3-yl]methyl}carbamoyl)thiophene-2-carboxylic acid
N-({5-[(3-ethoxyphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
N3-cyclohexyl-1-cyclopropyl-N5-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-[4-(3-methylphenyl)piperazin-1-yl]-N-[(1-methylpiperidin-3-yl)methyl]acetamide
6-methoxy-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]pyrimidin-4-amine
N-[3-(5-amino-1-methyl-1H-pyrazol-4-yl)phenyl]acetamide
N-{[1-(dimethylamino)cyclohexyl]methyl}-5-(3,4,5-trimethoxyphenyl)-1,2,4-triazin-3-amine
9-(2-hydroxy-5-methylbenzoyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
7-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-2-methyl-2,7-diazaspiro[4.5]decane
4-(1H-1,3-benzodiazol-1-yl)-1-(thiophene-2-carbonyl)piperidine-4-carboxylic acid
methyl 3-(2-methoxybenzamido)-5-[(phenylformamido)methyl]benzoate
3-{[(1-{[4-(1H-imidazol-1-yl)phenyl]methyl}piperidin-4-yl)oxy]methyl}pyridine
3-[1-(1-ethylpiperidin-4-yl)-1H-pyrazol-5-yl]-1-(3-fluorophenyl)urea
3-(4-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}piperazin-1-yl)-1,2-dihydropyrazin-2-one
4-(4-fluorophenyl)-1-(1-methylazepane-2-carbonyl)piperidin-4-ol
(2S,4R)-N-ethyl-4-(2-hydroxy-4-methylbenzamido)-1-[3-(methylsulfanyl)propyl]pyrrolidine-2-carboxamide
(4aS,8aR)-6-(2-aminopyrimidin-4-yl)-1-[2-(cyclohex-1-en-1-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
3-chloro-N-cyclopentyl-4-({1-[2-(1H-pyrazol-1-yl)acetyl]piperidin-4-yl}oxy)benzamide
[(2,3-difluoro-6-methoxyphenyl)methyl](methyl)[(1-methylpyrrolidin-2-yl)methyl]amine
2-{4-[(4-tert-butylphenyl)methyl]piperazin-1-yl}pyridine-3-carboxamide
1-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propan-1-one
1-[(2-chloro-6-fluorophenyl)methyl]-3-(2-methoxyethyl)-5-(5-methoxyfuran-2-yl)-1H-1,2,4-triazole
N-{1-[1-(2,5-dimethylbenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopropanecarboxamide
N-cyclopropyl-2-(2-oxopiperidin-1-yl)-N-(1,3-thiazol-2-ylmethyl)acetamide
ethyl 3-[(2-methylphenyl)methyl]-1-(phenylcarbamoyl)piperidine-3-carboxylate
5-acetyl-N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methylthiophene-2-carboxamide
(4aS,7aR)-N-ethyl-6,6-dioxo-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
ethyl 3-[(3-chlorophenyl)methyl]-1-(5-ethyl-1,2-oxazole-3-carbonyl)piperidine-3-carboxylate
5-{1-[2-(2,5-dimethoxyphenyl)acetyl]pyrrolidin-2-yl}thiophene-2-carboxamide
4-(2-methyl-1-benzofuran-7-carbonyl)-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
10-[(3S,4R)-4-hydroxy-4-methyl-3-(2-methylpropyl)piperidine-1-carbonyl]-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraen-9-one
3-(3-fluorophenyl)-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]benzamide
2-[1-(cyclopropylmethyl)-4-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperazin-2-yl]ethan-1-ol
N-[2-(2-methoxyphenyl)ethyl]-2-(4-{4-[(oxolan-2-ylmethyl)amino]piperidin-1-yl}phenyl)acetamide
N-benzyl-4-chloro-1-methyl-N-[(4-methyl-1,3-thiazol-5-yl)methyl]-1H-pyrazole-3-carboxamide
2-[1-(2,2-dimethylpropyl)-4-[(1-methyl-1H-indol-3-yl)methyl]piperazin-2-yl]ethan-1-ol
3-[(3S,7S,8aS)-3-[(benzyloxy)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-chloro-4-methylphenyl)urea
4-(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidin-4-yl)thiomorpholine
9-(2-aminopyridine-4-carbonyl)-2-(2-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
4-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]-1-phenyl-1H-pyrazole
{1-[(3-chloro-5-fluorophenyl)methyl]-3-[(dimethylamino)methyl]piperidin-3-yl}methanol