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6-[(3-phenyl-1H-pyrazol-5-yl)methyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
N-methyl-N-[(3-methylpyridin-4-yl)methyl]-3-(1,2-oxazinan-2-yl)propanamide
8-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
(2R,3R)-3-[methyl(thiophen-2-ylmethyl)amino]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
3-(carbamoylmethoxy)-N-{1-[(3-chlorophenyl)methyl]-1H-pyrazol-5-yl}benzamide
N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-9H-purin-6-amine
6-ethyl-N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}-2-oxo-1,2-dihydropyridine-4-carboxamide
1-({3-[2-hydroxy-3-(4-methylpiperazin-1-yl)propoxy]-4-methoxyphenyl}methyl)azetidin-3-ol
3-({[1-(hydroxymethyl)cyclopropyl]carbamoyl}methyl)-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
1-[1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidin-3-yl]-4-[3-(trifluoromethyl)phenyl]piperazine
8-(2-methylpyrimidin-4-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
(3aR,6aS)-2-ethyl-5-[4-methyl-2-(methylamino)-1,3-thiazole-5-carbonyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[5-(3,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-2-(4-fluorophenyl)piperidine
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-(2-methoxyphenyl)propanamide
4-(2-fluorophenoxy)-1-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
ethyl 2-(1-{1-[(3-methoxyphenyl)methyl]-6-oxopiperidin-3-yl}-N-methylformamido)acetate
ethyl 1-(3-methylbutyl)-5-[3-(pyrazin-2-yl)propanoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
ethyl({[2-(piperidin-1-yl)pyrimidin-5-yl]methyl})[2-(1H-pyrazol-1-yl)ethyl]amine
(3S,4S)-1-[3-(2-amino-1,3-thiazol-4-yl)propanoyl]-4-cyclopropylpyrrolidine-3-carboxylic acid
(2R,6R)-1-(1H-imidazole-2-carbonyl)-2,6-bis(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
N-({1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]piperidin-3-yl}methyl)naphthalene-1-carboxamide
(2S,4S)-4-{[(2,4-difluorophenyl)methyl]amino}-N-(propan-2-yl)-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(3-methylphenyl)acetamide
N-[(3S,5S,9R)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]-3-fluoro-4-methylbenzamide
1-[2-(4-cycloheptylpiperazin-1-yl)ethyl]-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
N-[(2-chlorophenyl)methyl]-3-[(3S,4R)-1-(2-methylpropyl)-4-(morpholin-4-yl)piperidin-3-yl]propanamide
N-{[4-hydroxy-1-(pyrazine-2-carbonyl)azepan-4-yl]methyl}morpholine-4-carboxamide
2-hydroxy-N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}-4-methylbenzamide
1-{3-[4-(difluoromethoxy)phenyl]phenyl}-1H-pyrazole
4-{1-[(3-methyl-1,2-oxazol-5-yl)methyl]-1H-imidazol-2-yl}-2,1,3-benzoxadiazole
1-{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-[3-(trifluoromethyl)phenyl]piperazine
5-[2-(ethanesulfonyl)acetyl]-N-phenyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
1-[(3-methylpyridin-2-yl)methyl]-4-[3-(thiophen-2-yl)-1H-pyrazole-4-carbonyl]piperazine
N-[(4-chlorophenyl)methyl]-2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxybenzamide
methyl 6-[(2,4-dimethylphenyl)methyl]-2-[(2-methoxyethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-(2-oxo-2-{4-[2-(pyridin-4-yl)ethyl]piperazin-1-yl}ethyl)-2,3-dihydro-1,3-benzoxazol-2-one
[3-({1-[(3-chloro-5-fluoro-4-methoxyphenyl)methyl]pyrrolidin-3-yl}methyl)phenyl]methanol
4-[4-(butylamino)piperidin-1-yl]-N-(1-phenylethyl)benzamide
1-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-2-[2-(1H-imidazol-1-yl)ethyl]piperidine
1-(4-ethylpiperazin-1-yl)-3-[3-({methyl[(4-methylphenyl)methyl]amino}methyl)phenoxy]propan-2-ol
N-cyclopropyl-N-{[2-(dimethylamino)-7-methylquinolin-3-yl]methyl}naphthalene-1-carboxamide
6-(2-aminoethyl)-N-(furan-3-ylmethyl)-N-methylpyrimidin-4-amine
N-{[4-fluoro-3-(trifluoromethyl)phenyl]methyl}-2,2-dimethylcyclopropane-1-carboxamide
(2S,4R)-N-ethyl-1-(1,2-oxazole-3-carbonyl)-4-(thiophene-3-amido)pyrrolidine-2-carboxamide
6-[4-(propan-2-yl)phenyl]-1,3,8-triazatricyclo[7.4.0.02,7]trideca-2(7),8-dien-4-one
ethyl 4-[5-amino-2-(2-methoxyphenyl)-1-methyl-1H-1,3-benzodiazole-7-amido]piperidine-1-carboxylate
N-benzyl-2-(morpholin-2-yl)-N-(2,2,2-trifluoroethyl)acetamide
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}propanamide
{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(2-methoxyethyl)methylamine