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5-[4-(4-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-N-ethylpyrimidin-2-amine
4-[(3-methoxyphenyl)methyl]-1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-1,4-diazepan-5-one
2-(methylamino)-N-[2-(1-methylpyrrolidin-2-yl)ethyl]pyridine-3-carboxamide
2-{1-[1-(piperidin-1-yl)cyclohexanecarbonyl]pyrrolidin-2-yl}pyridine
N-{[7-(4,6-dimethylpyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-5-(methoxymethyl)furan-2-carboxamide
{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}(methyl)[(4-methyl-1,3-thiazol-2-yl)methyl]amine
2-(dimethylamino)-N-(2-hydroxyethyl)-2-(4-methylphenyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]acetamide
(4aS,7aR)-1-[(4-methoxyphenyl)methyl]-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}[2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl]amine
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-methyl-N-(1,2-oxazol-3-ylmethyl)piperidine-3-carboxamide
1-(1H-1,2,3-benzotriazol-4-yl)-3-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]urea
2-(3,4-dimethylphenoxy)-1-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]ethan-1-one
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-ethyl-1-methyl-1H-pyrazole-5-carboxamide
3-[6-(cyclopentylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]-6-methylpyridin-2-amine
2-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]acetamide
1-{4-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-3-phenylpropan-1-ol
{4-[(3-fluorophenyl)methyl]-1-(4-methoxypyrimidin-2-yl)piperidin-4-yl}methanol
N-(1,3-dihydro-2-benzofuran-5-yl)-2-(2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-4-(thiophen-2-yl)phenoxy)acetamide
4-(1H-indol-2-ylmethyl)-9-methoxy-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(1R,3S)-1,3-dihydroxy-N-[3-(trifluoromethyl)phenyl]-7-azaspiro[3.5]nonane-7-carboxamide
(2S)-N-[(5-chloro-3-methyl-2-phenyl-1H-indol-7-yl)methyl]-5-oxopyrrolidine-2-carboxamide
N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-2-(furan-2-yl)-2-oxoacetamide
7-fluoro-3-methyl-N-[1-(thiophen-3-yl)propan-2-yl]-1-benzofuran-2-carboxamide
3-{3-[5-(furan-2-yl)-4-phenyl-1H-imidazol-1-yl]propoxy}pyridine
3-methyl-1-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-1,2-dihydroquinoxalin-2-one
3-(1,4-dioxan-2-ylmethyl)-1-[4-(2-methoxyphenoxy)phenyl]urea
dimethyl({[4-methyl-5-(1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl)-4H-1,2,4-triazol-3-yl]methyl})amine
3-{1-[(8-methoxy-2H-chromen-3-yl)methyl]piperidin-4-yl}-1-(morpholin-4-yl)propan-1-one
(3S,4R)-1-{imidazo[1,2-a]pyridine-2-carbonyl}-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
N-butyl-N-(furan-2-ylmethyl)-2-methanesulfonamidopropanamide
N-[(4-fluorophenyl)(pyridin-4-yl)methyl]-2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]-N-{[2-(trifluoromethoxy)phenyl]methyl}acetamide
(3R,4R)-1-(2,1,3-benzothiadiazol-5-ylmethyl)-4-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidin-3-ol
N-{5-[({[4-(hydroxymethyl)oxan-4-yl]methyl}carbamoyl)amino]-2-methoxyphenyl}-2-methoxyacetamide
N-[3-(1H-1,3-benzodiazol-2-yl)propyl]-1-ethyl-6-oxopiperidine-3-carboxamide
N-{3-[(3S,4R)-3-ethyl-4-hydroxy-4-methylpiperidin-1-yl]-3-oxopropyl}-3-methoxybenzamide
3-({[2-(3-phenoxyphenyl)ethyl]amino}methyl)pyrrolidin-3-ol
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[(3,4-difluorophenyl)methyl]-1,3-oxazole-4-carboxamide
N-[2-methoxy-2-(thiophen-2-yl)ethyl]-5,6,7,8-tetrahydroquinoline-3-carboxamide
2-(propan-2-yl)-4-({4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)pyrimidine
3-(2-chlorophenyl)-3-(3-hydroxyphenyl)-N-methyl-N-[(3-methylpyridin-4-yl)methyl]propanamide
methyl({[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}){[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}amine
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-4-methyl-N-(2-methylpropyl)-1H-imidazole-2-carboxamide
4-(4-{[3-(2-hydroxyethyl)-4-[(2-methylphenyl)methyl]piperazin-1-yl]methyl}phenyl)-2-methylbut-3-yn-2-ol
N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}-2-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)acetamide
(1R,3S)-3-amino-N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)cyclohexane-1-carboxamide
N-{2-methoxy-4-[3-(pyridin-3-yl)propanamido]phenyl}butanamide
4-{[5-(3,5-dimethyl-4,5-dihydro-1,2-oxazol-5-yl)-1,2,4-oxadiazol-3-yl]methyl}-1-propylpiperidine
2-amino-4-[methyl(pyridin-3-ylmethyl)amino]quinazoline-6-carboxylic acid
N-[2-(4-ethyl-1,3-thiazol-2-yl)ethyl]-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide