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5-(1-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)-5-(3-phenylpropyl)imidazolidine-2,4-dione
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-[2-(1H-indol-1-yl)ethyl]propanamide
(2-{5-[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}phenyl)methanol
3-(3-fluorophenyl)-4-(2-methyl-1-benzofuran-5-carbonyl)piperazin-2-one
N-cyclopropyl-1-[3-(4-fluorophenyl)phenyl]piperidin-4-amine
4-(2,5-dimethoxyphenyl)-3-[(4-hydroxyphenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
8-(2,3-dihydro-1H-inden-2-yl)-1-(2-methoxyethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(9H-fluorene-9-carbonyl)-3-(hydroxymethyl)piperidin-3-ol
1-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-2-(4-methylphenoxy)ethan-1-one
(1R,5R)-6-[3-(4-fluorophenoxy)propyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-(3-phenylpyrrolidin-1-yl)acetamide
1-[(3-methyl-1,2-oxazol-5-yl)methyl]-3-(3-methylbut-2-en-1-yl)piperidine-3-carboxylic acid
4-ethyl-3-(piperidin-3-yl)-1-{[6-(trifluoromethyl)pyridin-3-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
(3R,9aR)-3-(2-methylpropyl)-8-(quinolin-5-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methylquinoxaline-6-carboxamide
methyl 2-{[5-(4-fluorophenyl)-4-[1-(2-methoxypyridine-3-carbonyl)piperidin-3-yl]pyrimidin-2-yl]sulfanyl}acetate
N-[1-(4-methoxyphenyl)-5-oxopyrrolidin-3-yl]-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
1-[4-(propylsulfamoyl)phenyl]-3-[2-(1,3-thiazol-2-yl)ethyl]urea
propan-2-yl 4-chloro-3-(2,5-dihydro-1H-pyrrole-2-amido)benzoate
methyl 2-[8-(furan-3-ylmethyl)-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-N-[3-(propan-2-yloxy)propyl]-1H-pyrazole-4-carboxamide
2-{1-[(3-methylphenyl)methyl]-5-(3-oxo-1,2,3,4-tetrahydroquinoxalin-6-yl)-1H-1,2,4-triazol-3-yl}acetamide
4-[5-fluoro-2-(2-fluoro-3-methylphenyl)pyrimidin-4-yl]morpholine
2-[(3,4-dimethoxyphenyl)methyl]-N,N-bis(prop-2-en-1-yl)-1,3-benzoxazole-6-carboxamide
3-chloro-N-cyclopentyl-4-{[1-(6-oxo-1,6-dihydropyridazine-3-carbonyl)piperidin-4-yl]oxy}benzamide
2-[4-(2H-1,3-benzodioxol-4-ylmethyl)-1-[(2-methylphenyl)methyl]piperazin-2-yl]ethan-1-ol
N-methyl-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]-2-[(4S)-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]acetamide
1-[2-(2-ethoxyethoxy)phenyl]-3-[(3R,4R)-3-hydroxypiperidin-4-yl]urea
1-(2-methyloxolane-2-carbonyl)-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
[2-(dimethylamino)-1-phenylethyl]({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl})amine
N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}imidazo[1,2-a]pyridine-3-carboxamide
N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2,3-dihydro-1-benzofuran-2-carboxamide
2-chloro-N-methyl-5-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}benzamide
2-[2-(6-fluoroquinolin-2-yl)-1H-imidazol-1-yl]-1-(piperazin-1-yl)ethan-1-one
6-(2-propyl-1H-imidazol-1-yl)naphthalen-2-ol
N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-{[4-(pyridin-2-yl)phenyl]methyl}cyclopropanamine
ethyl 3-[(2-fluorophenyl)methyl]-1-[4-(2-oxopiperidin-1-yl)butanoyl]piperidine-3-carboxylate
N-({8-[(2-methoxyphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)furan-3-carboxamide
2-(2-{[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
(1-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}-4-(2-phenylethyl)piperidin-4-yl)methanol
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-1-(difluoromethyl)-1H-pyrazole-3-carboxamide
2-(4-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl)ethan-1-ol
1-(cyclopropylmethyl)-N-[3-(3-fluorophenyl)phenyl]piperidine-4-carboxamide
1-[(3,5-dimethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylic acid
2-{[5-(1,5-dimethyl-1H-pyrazol-4-yl)-4-(1-phenylethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]methylamine
N-(4-{[3-(morpholin-4-yl)piperidin-1-yl]sulfonyl}phenyl)acetamide
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]cyclohex-1-ene-1-carboxamide
N-(1-butyl-3-methyl-1H-pyrazol-5-yl)-4-(pyrimidin-2-yloxy)piperidine-1-carboxamide
N-[(2S)-1-methoxypropan-2-yl]-3-[methyl(thian-4-yl)sulfamoyl]benzamide